CHEBI:38637 - tyrosine kinase inhibitor

ChEBI IDCHEBI:38637
ChEBI Nametyrosine kinase inhibitor
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DefinitionAny protein kinase inhibitor that interferes with the action of tyrosine kinase.
Last Modified27 February 2025
SubmitterMarcus Ennis
Wikipedia
ChEBI Ontology
Outgoing Relation(s)
tyrosine kinase inhibitor (CHEBI:38637) is a protein kinase inhibitor (CHEBI:37699)
Incoming Relation(s)
1-NA-PP1 (CHEBI:52310) has role tyrosine kinase inhibitor (CHEBI:38637)
1-NM-PP1 (CHEBI:52309) has role tyrosine kinase inhibitor (CHEBI:38637)
4,5-dianilinophthalimide (CHEBI:53110) has role tyrosine kinase inhibitor (CHEBI:38637)
afatinib (CHEBI:61390) has role tyrosine kinase inhibitor (CHEBI:38637)
afatinib dimaleate (CHEBI:76003) has role tyrosine kinase inhibitor (CHEBI:38637)
axitinib (CHEBI:66910) has role tyrosine kinase inhibitor (CHEBI:38637)
BE-23372M (CHEBI:65473) has role tyrosine kinase inhibitor (CHEBI:38637)
biochanin A (CHEBI:17574) has role tyrosine kinase inhibitor (CHEBI:38637)
bosutinib (CHEBI:39112) has role tyrosine kinase inhibitor (CHEBI:38637)
bosutinib hydrate (CHEBI:68533) has role tyrosine kinase inhibitor (CHEBI:38637)
brigatinib (CHEBI:232810) has role tyrosine kinase inhibitor (CHEBI:38637)
butein (CHEBI:3237) has role tyrosine kinase inhibitor (CHEBI:38637)
cabozantinib (CHEBI:72317) has role tyrosine kinase inhibitor (CHEBI:38637)
cabozantinib malate (CHEBI:72319) has role tyrosine kinase inhibitor (CHEBI:38637)
canertinib (CHEBI:61399) has role tyrosine kinase inhibitor (CHEBI:38637)
dasatinib (anhydrous) (CHEBI:49375) has role tyrosine kinase inhibitor (CHEBI:38637)
dasatinib monohydrate (CHEBI:70839) has role tyrosine kinase inhibitor (CHEBI:38637)
DCC-2036 (CHEBI:62166) has role tyrosine kinase inhibitor (CHEBI:38637)
emodin (CHEBI:42223) has role tyrosine kinase inhibitor (CHEBI:38637)
emodin(1−) (CHEBI:77659) has role tyrosine kinase inhibitor (CHEBI:38637)
genistein (CHEBI:28088) has role tyrosine kinase inhibitor (CHEBI:38637)
herbimycin (CHEBI:5674) has role tyrosine kinase inhibitor (CHEBI:38637)
hydroxy-2-naphthalenyl-methyl phosphonic acid trisacetoxymethylester (CHEBI:75391) has role tyrosine kinase inhibitor (CHEBI:38637)
imatinib (CHEBI:45783) has role tyrosine kinase inhibitor (CHEBI:38637)
imatinib methanesulfonate (CHEBI:31690) has role tyrosine kinase inhibitor (CHEBI:38637)
lapatinib (CHEBI:49603) has role tyrosine kinase inhibitor (CHEBI:38637)
leflunomide (CHEBI:6402) has role tyrosine kinase inhibitor (CHEBI:38637)
masitinib (CHEBI:63450) has role tyrosine kinase inhibitor (CHEBI:38637)
melemeleone B (CHEBI:66690) has role tyrosine kinase inhibitor (CHEBI:38637)
neratinib (CHEBI:61397) has role tyrosine kinase inhibitor (CHEBI:38637)
nilotinib (CHEBI:52172) has role tyrosine kinase inhibitor (CHEBI:38637)
nintedanib (CHEBI:85164) has role tyrosine kinase inhibitor (CHEBI:38637)
nintedanib esylate (CHEBI:85170) has role tyrosine kinase inhibitor (CHEBI:38637)
pazopanib (CHEBI:71219) has role tyrosine kinase inhibitor (CHEBI:38637)
pazopanib hydrochloride (CHEBI:71217) has role tyrosine kinase inhibitor (CHEBI:38637)
PD173955 (CHEBI:49791) has role tyrosine kinase inhibitor (CHEBI:38637)
piceatannol (CHEBI:28814) has role tyrosine kinase inhibitor (CHEBI:38637)
picropodophyllotoxin (CHEBI:75251) has role tyrosine kinase inhibitor (CHEBI:38637)
ponatinib (CHEBI:78543) has role tyrosine kinase inhibitor (CHEBI:38637)
ponatinib hydrochloride (CHEBI:191940) has role tyrosine kinase inhibitor (CHEBI:38637)
PP121 (CHEBI:50915) has role tyrosine kinase inhibitor (CHEBI:38637)
radicicol (CHEBI:556075) has role tyrosine kinase inhibitor (CHEBI:38637)
regorafenib (CHEBI:68647) has role tyrosine kinase inhibitor (CHEBI:38637)
regorafenib hydrate (CHEBI:68646) has role tyrosine kinase inhibitor (CHEBI:38637)
Remibrutinib (CHEBI:746867) has role tyrosine kinase inhibitor (CHEBI:38637)
SKLB-677 (CHEBI:140875) has role tyrosine kinase inhibitor (CHEBI:38637)
sorafenib (CHEBI:50924) has role tyrosine kinase inhibitor (CHEBI:38637)
teriflunomide (CHEBI:68540) has role tyrosine kinase inhibitor (CHEBI:38637)
vandetanib (CHEBI:49960) has role tyrosine kinase inhibitor (CHEBI:38637)
WZ4002 (CHEBI:61400) has role tyrosine kinase inhibitor (CHEBI:38637)
EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434) is a tyrosine kinase inhibitor (CHEBI:38637)
EC 2.7.10.2 (non-specific protein-tyrosine kinase) inhibitor (CHEBI:76617) is a tyrosine kinase inhibitor (CHEBI:38637)
Synonyms  Source
tyrosine kinase inhibitorsChEBI
protein tyrosine kinase inhibitorChEBI
TKI inhibitorChEBI
TKI inhibitorsChEBI
protein tyrosine kinase inhibitorsChEBI
tyrphostinsChEBI
Manual XrefsDatabases
Tyrosine-kinase_inhibitorWikipedia