Small-molecule Inhibitors of Peptidases

Main names are emphasised. All names are links to the respective Summary pages.

(   1   2   3   4   5   6   7   9   <   A   B   C   D   E   F   G   H   I   J   K   L   M   N   O   P   Q   R   S   T   U   V   W   X   Y   Z   [   {  


(
(+)-2-[4-[(-1-acetimidoyl-4-piperidinyl)oxy]- 3-(7-amidino-2-naphthyl)propionic acid DX-9065a
(2-benzyl-3-mercaptopropanoyl)-L-alanylglycinamide (2-benzyl-3-mercaptopropanoyl)-L-alanylglycinamide
(2S)-5-amino-2-[(1-n-propyl-1H-imidazol-4-yl)methyl]pentanoic acid UK-396082
(3R)-amino-(2S)-hydroxyheptanoyl-l-Ala-l-Leu-l-Val-l-Phe-OMe small-molecule inhibitors of metallopeptidases
(3S,4S)-3-amino-4-mercapto-6-phenyl-hexane-1-sulfonic acid (3S,4S)-3-amino-4-mercapto-6-phenyl-hexane-1-sulfonic acid
(4R)-3-[(2S)-3-mercapto-2-methylpropanoyl]-4-thiazolidinecarboxylic acid YS-980
(4S)-4-[4-cyano-2-(methylsulfonyl)phenyl]-3,6-dimethyl-2-oxo-1-[3-(trifluorometh yl)phenyl]-1,2,3,4-tetrahydropyrimidine-5-carbonitrile BAY 85-8501
(5-(1R)-4-cyclohexyl-1-[2-(hydroxyamino)-2-oxoethyl]butyl-1,2,4-oxadiazole-3-carboxamide) UK-383,367
(acyloxy)methyl ketone acyloxymethane derivatives
(CYGAK)(2) CYGAK2
(N-[2(S)-(mercapto-methyl)-3-(2-methylphenyl)-4-oxopropyl]-L-methionine SCH 42354
(R)-4-cyclopropyl-7,8-difluoro-5-(4-(trifluoromethyl)phenylsulfonyl)-4,5-dihydro-1H-pyrazolo[4,3-c]quinoline ELND006
(R)-4-cyclopropyl-8-fluoro-5-(6-(trifluoromethyl)pyridin-3-ylsulfonyl)-4,5-dihydro-2H-pyrazolo[4,3-c]quinoline ELND007
(S)-1-((S)-1-(4-phenylbutanoyl)-pyrrolidine-2-carbonyl)pyrrolidine-2-carbonitrile KYP-2047
(S)-2-((S)-2-(3,5-difluorophenyl)-2-hydroxyacetamido)-N-((S,Z)-3-methyl-4- oxo-4,5-dihydro-3H-benzo[d][1,2]diazepin-5-yl)propanamide BMS-433796
(S)-2-amino-3-(4-hydroxy-3-nitrophenyl)-N-((S,E)-5-phenyl-1-(phenylsulfonyl)pent-1-en-3-yl)propanamide SAK-1
(S)-3-(benzyloxycarbonyl-(S)-leucyl-(S)-leucylamino)-5-methyl-2-oxo-N-(2,4-dimethylphenyl)hexanamide BSc4999
(S)-3-amino-4-mercaptobutyl sulfonic acid EC33
(S)-Alanylpyrrolidine-boronic acid (Ala-boroPro) boron-containing inhibitors of serine peptidases
(S,S)-2-[2-(3,5-difluorophenyl)acetylamino]-N-(1-methyl-2-oxo-5-phenyl-2,3-dihydro-1Hbenzo[e][1,4]diazepin-3-yl)-propionamide compound E
1
1,2-epoxy-3-(p-nitrophenoxy) propane EPNP
1,3-diazetidine-2,4-dione azetidin-2-one derivative inhibitors of serine peptidases
1,5-dansyl-L-glutamyl-L-glycyl-L-arginine chloromethylketone halomethane inhibitors of serine peptidases
1-[3-(acetylsulfanyl)-2-methylpropanoyl]prolylphenylalanine alacepril
1-chloro-3-amino-4-phenyl-butanone-2 1-chloro-3-amino-4-phenyl-butanone-2
1-naphthalenesulfonyl-IW-CHO (NaphthaCHO) aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
1-naphthalenesulfonyl-lle-Trp-CHO NapSul-Ile-Trp-CHO
141W94 amprenavir
15-oxospiramilactone polyphenol inhibitors of cysteine peptidases
15apt S01.217-binding aptamer
15fTBA S01.217-binding aptamer
15TGT S01.217-binding aptamer
16R ML188
1G244 1G244
2
2(S)-benzyl-3-[hydroxy(1"(R)-aminoethyl)phosphinyl]propanoyl-l-tyrosine 7B
2,4-dichlorocinnamic acid hydroxamate 2,4-dichlorocinnamic acid hydroxamate
2,4-dichlorocinnamyl hydroxamate 2,4-dichlorocinnamyl hydroxamate
2,6-dimethyl-benzoic acid 3-benzyloxycarbonylamino-4-carbamoyl-2-oxo-butyl ester MV026630
2-(3-mercaptopropyl)pentanedioic acid 2-(3-mercaptopropyl)pentanedioic acid
2-(4-phenoxyphenylsulfonylmethyl)thiirane SB-3CT
2-[3-methyl[1-(2-naphthoyl)piperidin-4-yl]aminocarbonyl)-2-naphthyl]-1- (1-naphthyl)-2-oxoethylphosphonic acid RWJ-355871
2-amino-4-methylsulfonyl butane thiol PC18
2-amino-pentan-1,5-dithiol (EC27) EC27
2-aminobenzylstatine derivative pseudopeptide threonine peptidase inhibitor
2-benzyl-3,4-epithiobutanoic acid 2-benzyl-3,4-epithiobutanoic acid
2-benzyl-3,4-iminobutanoic acid 2-benzyl-3,4-iminobutanoic acid
2-benzyl-3-iodopropanoic acid 2-benzyl-3-iodopropanoic acid
2-benzyl-3-mercaptopropanoic acid SQ 14,603
2-benzyl-4-oxo-5,5,5-trifluoropentanoic acid haloketone inhibitor of metallopeptidase
2-mercaptoacetyl-L-leucyl-L-phenylalanine 2-mercaptoacetyl-L-leucyl-L-phenylalanine
2-mercaptoacetyl-L-phenylalanyl-L-leucine 2-mercaptoacetyl-L-phenylalanyl-L-leucine
2-mercaptoacyl-dipeptides 2-mercaptoacyl-dipeptides
2-mercaptomethyl-3-guanidinoethylthiopropanoic acid 2-mercaptomethyl-3-guanidinoethylthiopropanoic acid
2-mercaptomethyl-5-guanidinopentanoic acid SQ 24,798
2-MPPA 2-(3-mercaptopropyl)pentanedioic acid
2-naphthoyl-Lys-Lys-ArgH Naph-KKR-H
2-phenylethaneboronic acid 2-phenylethaneboronic acid
2-PMPA PMPA
24F hydroxamate-containing inhibitors of metallopeptidases
27apt S01.217-binding aptamer
2cPE (proinhibitor) compound 2c
2F12 small-molecule inhibitors of cysteine peptidases
3
3-(4-5-[(2R,6S)-2,6-dimethyltetrahydro-1(2H)-pyridinyl]pentyl-3-oxo-3,4-di hydro-2-quinoxalinyl)-4-hydroxybenzenecarboximidamide PD-198961
3-(4-[2-(E)-styrylphenoxy]butanoyl-l-4-hydroxyprolyl)-thiazolidine SUAM-14746
3-2-Mercaptoethyl)biphenyl-2,3-dicarboxylic acid E2072
3-[(2S,4S)-4-[4-(3-methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]pyrrolidin-2-ylcarbonyl]thiazolidine teneligliptin
3-acetyl-2-aminoquinolin-4-one 3-acetyl-2-aminoquinolin-4-one
3-amidinophenylalanine derivatives (S01.302 inhibitors) 3-amidinophenylalanine derivatives (S01.302 inhibitors)
3-amino-2-hydroxy-4-phenylbutanoylvalylisoleucine 3-amino-2-hydroxy-4-phenylbutanoylvalylisoleucine
3-but-2-ynyl-5-methyl-2-piperazin-1-yl-3,5-dihydro-4H-imidazo[4,5-d]pyridazin-4-one tosylate E3024
3-mercaptopropanoyl-L-proline mercaptoacyl amino acids
3-oxo-beta-sultam beta-sultams
3-TAPAP 3-TAPAP
3-thienylalanine-ornithyl-proline 3-thienylalanine-ornithyl-proline
351A MK351A
4
4"-acetaminophenyl 4-guanidinobenzoate hydrochloride AGB
4,4"-phosphinicobis(butane-1,3-dicarboxylic acid) phosphorus-containing inhibitors of metallopeptidases
4-(2-aminoethyl)benzenesulfonylfluoride AEBSF
4-(4-benzylphenyl)thiazol-2-amine ARM1
4-(dimethylamino)-N-[7-(hydroxyamino)-7-oxoheptyl]benzamide suberone derivative
4-(guanidinomethyl)phenylacetyl-Arg-Val-Arg-4-amidinobenzylamide inhibitor 24
4-[1-[[bis-(4-methyl-phenyl)-methy]-carbamoyl]-3-(2-ethoxy-benzyl)-4-oxo-azetidine-2-yloxy]-benzoic acid BCEAB
4-amino-5-mercaptopentanoic acid (Glu-thiol); Glu-thiol
4-aminophenylboronic acid boron-containing inhibitors of serine peptidases
4-APBA boron-containing inhibitors of serine peptidases
4-chloro-3-ethoxy-7-guanidinoisocoumarin 4-chloro-3-ethoxy-7-guanidinoisocoumarin
4-fluoro-1-(4-fluoro-(4-fluorophenyl)phenylalanyl)-2-pyrrolidinecarbonitrile denagliptin
4-guanidinomethyl-phenylacetyl-Arg-Tle-Arg-4-amidinobenzylamide MI-1148
4-hydroxy-2-nonenal (HNE) 4-hydroxy-2-nonenal (HNE)
4-methyl-1-(S)-(5-[(3-oxo-3,4-dihydro-2H-benzo[1,4]oxazin-6-ylmethyl)-carbamoyl]-pyrazolo[1,5-a]pyrimidine-7-carbonyl-amino)-indan-5-carboxylic acid small-molecule inhibitors of metallopeptidases
4862F 4862F
5
5,7,4-trihydroxyflavone apigenin
5-(4-phenoxyphenyl)-5-[4-(2-pyrimidinyl)-1-piperazinyl]barbituric acid 5-(4-phenoxyphenyl)-5-[4-(2-pyrimidinyl)-1-piperazinyl]barbituric acid
5-benzamido-2-benzyl-4-oxopentanoic acid 5-benzamido-2-benzyl-4-oxopentanoic acid
5-caffeoylquinic acid 5-caffeoylquinic acid
5-nitro-8-hydroxyquinoline nitroxoline
5-oxo-1,2,4-oxadiazole-related compounds 5-oxo-1,2,4-oxadiazole-related compounds
5-oxoprolinal 5-oxoprolinal
5-S-5-benzamido-4-oxo-6-phenylhexanoyl-L-proline 5-S-5-benzamido-4-oxo-6-phenylhexanoyl-L-proline
5S,6S penem 5S,6S penem
6
6,7-dihydroxy-2H-chromen-2-one esculetin
6-diazo-5-oxo-D-norleucine 6-diazo-5-oxo-D-norleucine
6-diazo-5-oxo-L-norleucylglycine 6-diazo-5-oxo-L-norleucylglycine
7
7-amino-3-(2-bromoethoxy)-4-chloroisocoumarin 7-amino-3-(2-bromoethoxy)-4-chloroisocoumarin
7-amino-4-chloro-3-methoxy isocoumarin JLK-6
7-but-2-ynyl-9-(6-methoxy-pyridin-3-yl)-6-piperazin-1-yl-7,9-dihydro-purin-8-one ER-319711
7-hydroxyflavone polyphenol inhibitors of cysteine peptidases
7B 7B
9
9-ethyloxyimino-9H-indeno[1,2-b]pyrazine-2,3-dicarbonitrile 9-ethyloxyimino-9H-indeno[1,2-b]pyrazine-2,3-dicarbonitrile
<
Bj-PRO-5a
[
[(S)-4-(2,4-difluoro-5-pyrimidin-5-yl-phenyl)-4-methyl-5,6-dihydro-4H-[1,3]thiazin-2-ylamine] LY2811376
[2-[3-[[(1-benzoyl-4-piperidinyl)methylamino]carbonyl]-2-naphthalenyl]-1-(1-naphthalenyl)-2-oxoethyl]-phosphonic acid cathepsin G inhibitor I
[N-(S)-(1-carboxy-3-phenylpropyl)- (S)-leucyl-(S)-tryptophan] CLT
A
A-183 peptide inhibitors of serine peptidases
A-357300 A-357300
A-705239 A-705239
A-705253 A-705253
A-74704 A-74704
A-77003 A-77003
A-790742 A-790742
A-792611 A-792611
A-80987 A-80987
A-84538 A-84538
A70450 A70450
A90720A A90720A
AAE581 AAE581
AAPACK Ac-Ala-Ala-Pro-AlaCH2Cl
AAPFcmk Suc-Ala-Ala-Pro-Phe-CH(2)Cl
aaptamine small-molecule inhibitors of threonine peptidases
aaptamine aaptamine
AB192 AB192
ABBA ABBA
ABS 130 2,4-dichlorocinnamic acid hydroxamate
ABS 252 thiol inhibitors of metallopeptidases
ABT-279 ABT-279
ABT-341 ABT-341
ABT-378 lopinavir
ABT-450 ABT-450
ABT-493 glecaprevir
ABT-518 ABT-518
ABT-538 ritonavir
Ac-Ala-Ala-Pro-Ala-CMK Ac-Ala-Ala-Pro-AlaCH2Cl
Ac-Ala-Ala-Pro-AlaCH2Cl Ac-Ala-Ala-Pro-AlaCH2Cl
Ac-Ala-Ala-Pro-CHN2 diazo inhibitors of serine peptidases
Ac-Ala-Ala-Pro-Val-CMK Ac-Ala-Ala-Pro-Val-CMK
Ac-Ala-Lys-boroArg boron-containing inhibitors of serine peptidases
Ac-Arg-Glu-Lys-Arg peptidyl boronic acid boron-containing inhibitors of serine peptidases
Ac-Arg-Glu-Lys-boroArg pinanediol boron-containing inhibitors of serine peptidases
Ac-Asp-Glu-Val-Asp-glyoxal aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
Ac-Asp-Glu-Val-Asp-H Ac-Asp-Glu-Val-Asp-H
Ac-Asp-Met-Gln-Asp-H aldehyde or ketone C14.GNW inhibitors
Ac-Asp-PheY(PO2-CH2)(L)Ala-Ala-NH2 RXP401
Ac-Asp-Val-Ala-Asp-CH(2)F Ac-Asp-Val-Ala-Asp-CH(2)F
Ac-DEVD-CHO Ac-Asp-Glu-Val-Asp-H
Ac-DEVD-glyoxal aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
Ac-DLeu-LLLRVK-Amba C23
Ac-DMQD-CHO aldehyde or ketone C14.GNW inhibitors
Ac-DMQD-CHO aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
Ac-DNLD-CHO aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
Ac-DPMSSTYIEELGKREVTIPPKYRELLA-NH2 calpastatin peptide
Ac-DVAD-fmk Ac-Asp-Val-Ala-Asp-CH(2)F
Ac-Ile-Glu-Thr-Asp-H Ac-Ile-Glu-Thr-Asp-H
ac-KR-H aldehyde- or ketone-related inhibitors of serine peptidases
Ac-LAAQ(mm)-FMK Ac-Leu-Ala-Ala-Gln(Me2)-FMK
Ac-LEHD-CHO aldehyde or ketone C14.GNW inhibitors
Ac-Leu-Ala-Ala-Gln(Me2)-FMK Ac-Leu-Ala-Ala-Gln(Me2)-FMK
Ac-Leu-Ala-Ala-Gln(Me2)-pMK Ac-Leu-Ala-Ala-Gln(Me2)-pMK
Ac-Leu-Asp-Glu-Ser-Asp-H aldehyde or ketone C14.GNW inhibitors
Ac-Leu-Leu-Arg-H leupeptin
Ac-Leu-Leu-Met-H ALLM
Ac-Leu-Leu-Nle-H ALLN
Ac-Leu-Phe-Phe-Glu-FMK Ac-Leu-Phe-Phe-Glu-FMK
Ac-LVK-CHO aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
Ac-NA-Val-Sta-Glu-NA-NH2 LP-149
Ac-PRLNvs Ac-Pro-Arg-Leu-AsnVS
Ac-Pro-Arg-Leu-AsnVS Ac-Pro-Arg-Leu-AsnVS
Ac-Pro-Thr-Ser-Tyr-CH(2)Cl halomethane inhibitors of serine peptidases
Ac-Ser-Leu-Asn-Phe-PSI(CH(OH)-CH2)-Pro-Ile-Val-OME JG-365
Ac-tLeu-Asp-H small-molecule inhibitors of cysteine peptidases
Ac-Trp-Glu-His-Asp-H Ac-Trp-Glu-His-Asp-H
Ac-Tyr-Val-Ala-Asp-chloromethylketone Ac-YVAD-CMK
Ac-Tyr-Val-Ala-Asp-H Ac-Tyr-Val-Ala-Asp-H
Ac-Val-Glu-Ile-Asp-H aldehyde or ketone C14.GNW inhibitors
Ac-VEID-CHO aldehyde or ketone C14.GNW inhibitors
Ac-WEHD-CHO Ac-Trp-Glu-His-Asp-H
Ac-YVAD-CHO Ac-Tyr-Val-Ala-Asp-H
Ac-YVAD-CMK Ac-YVAD-CMK
AC1NX476 small-molecule inhibitors of aspartic peptidases
acacetin polyphenol inhibitors of cysteine peptidases
acetorphan (prodrug) thiorphan
N-acetyl-L-leucyl-L-leucyl-D,L-argininaldehyde leupeptin
acetylaminoacetaldehyde aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
ACH-1625 small-molecule serine peptidase inhibitors
ACH-2684 ACH-2684
acivicin acivicin
aclacinomycin A aclacinomycin A
ACT-077825 MK-8141
ACT-178882 MK-1597
actinonin actinonin
active metabolite M8 nelfinavir
acyl sulfonamide S29.001 inhibitors acyl sulfonamide S29.001 inhibitors
acylating inhibitors of cysteine peptidases acylating inhibitors of cysteine peptidases
acylating inhibitors of serine peptidases acylating inhibitors of serine peptidases
acyloxymethane derivatives acyloxymethane derivatives
acyloxymethylketone C25.001 inhibitor acyloxymethylketone C25.001 inhibitor
Ada-Ahx3-L3VS Ada-Ahx3-L3VS
AdaAhx(3)L(3)VS Ada-Ahx3-L3VS
adapentpronitrile aldehyde- or ketone-related inhibitors of serine peptidases
AE-3763 AE-3763
AEBSF AEBSF
aeruginosin aeruginosin
AG-1343 nelfinavir
AG-1776 AG-1776
AG1776 KNI-764
AG3340 Prinomastat
AG7088 rupintrivir
AG7404 AG7404
agaricoglyceride A unclassified small-molecule inhibitors of peptidases
AGB AGB
ageladine A ageladine A
Agenerase amprenavir
AGM-1470 fumagillin
AGM-1470 TNP-470
ahpatinin pseudo-peptide bond inhibitors of aspartic peptidases
AHU377 (prodrug of M13.001 inhibitor LBQ657) LBQ657
AJN-230 AJN-230
AK275 AK275
AK295 AK295
AL-11 (M01.011 ligand) peptide inhibitors of metallopeptidase
Ala-Ala-Phe-CH(2)Cl Ala-Ala-Phe-CH(2)Cl
Ala-Gly-Lys-Lys-Asp-Asp-Asp-Asp-Pro-Pro-Glu bifunctional aspartic peptidase inhibitor (Bacillus sp.)
Ala-Met-Asn peptide inhibitors of metallopeptidase
alacepril alacepril
alatrioprilat small-molecule inhibitors of metallopeptidases
aldehyde inhibitors of calpains aldehyde inhibitors of calpains
aldehyde or ketone C14.GNW inhibitors aldehyde or ketone C14.GNW inhibitors
aldehyde or ketone inhibitors of metallopeptidases aldehyde or ketone inhibitors of metallopeptidases
aldehyde, glyoxal or ketone inhibitors of aspartic peptidases aldehyde, glyoxal or ketone inhibitors of aspartic peptidases
aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
aldehyde- or ketone-related inhibitors of serine peptidases aldehyde- or ketone-related inhibitors of serine peptidases
aldehyde-like S09.003 inhibitors aldehyde-like S09.003 inhibitors
aliskiren aliskiren
alkalo-thermophilic Bacillus inhibitor bifunctional aspartic peptidase inhibitor (Bacillus sp.)
allicin allicin
ALLM ALLM
ALLN ALLN
allophenylnorstatine-containing inhibitors pseudo-peptide bond inhibitors of aspartic peptidases
allyl (5S,6S)-6-[(R)-acetoxyethyl]-penem-3-carboxylate 5S,6S penem
allyl sulfone vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases
alogliptin alogliptin
aloxistatin E64d
alpha,beta-unsaturated benzo[1,4]diazepin-2-one methyl ester alpha,beta-unsaturated benzo[1,4]diazepin-2-one methyl ester
alpha-ketoamide proteasome inhibitor aldehydes
alpha-ketoamide calpain inhibitors alpha-ketoamide calpain inhibitors
alpha-ketoamide inhibitors of C01.036 alpha-ketoamide inhibitors of C01.036
alpha-ketoamide inhibitors of cysteine peptidases alpha-ketoamide inhibitors of cysteine peptidases
alpha-ketoamide inhibitors of serine peptidases alpha-ketoamide inhibitors of serine peptidases
alpha-lipoic acid thiol inhibitors of metallopeptidases
alpha-MAPI MAPI microbial alkaline proteinase inhibitor
alpha-mercapto-beta-amino acyl dipeptides alpha-mercapto-beta-amino acyl dipeptides
ALS 1-0635 ALS 1-0635
AM-409 small-molecule inhibitors of metallopeptidases
AM114 boronic-chalcone proteasome inhibitor AM114 boronic-chalcone proteasome inhibitor
AM146 small-molecule inhibitors of cysteine peptidases
AM4299 AM4299
AMAC AMAC
amastatin amastatin
AMCHA tranexamic acid
AMG-126737 AMG-126737
AMG-8718 small-molecule inhibitors of aspartic peptidases
amino acid sulfonate sulfur-containing inhibitors of serine peptidases
aminoacetonitrile C01.036 inhibitors aminoacetonitrile C01.036 inhibitors
aminoglycoside aminoglycoside
trans-4-(aminomethyl)cyclohexane carboxylic acid tranexamic acid
amprenavir amprenavir
AMS-36 AMS-36
An-1 small-molecule inhibitors of metallopeptidases
anabaenopeptin cyclic peptide inhibitors of serine peptidases
anabaenopeptin 679 anabaenopeptin G
anabaenopeptin 908 anabaenopeptin G
anabaenopeptin B anabaenopeptin G
anabaenopeptin C anabaenopeptin G
anabaenopeptin F anabaenopeptin G
anabaenopeptin G anabaenopeptin G
anabaenopeptin H anabaenopeptin G
anabaenopeptin I anabaenopeptin G
anabaenopeptin J anabaenopeptin G
anacardic acid small-molecule inhibitors of metallopeptidases
anagliptin anagliptin
ancovenin ancovenin
angiotensin II angiotensin II
angiotensin IV angiotensin IV
angiotensin-receptor-neprilysin inhibitor LBQ657
anilide inhibitor anilide inhibitor
antibiotic TA myxovirescin
antipain antipain
AOMK acyloxymethane derivatives
APC 2059 APC 2059
APC-366 APC-366
APC2848 APC2848
APC3316 vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases
APC3328 APC3328
APG12 small-molecule inhibitors of aspartic peptidases
APG19 small-molecule inhibitors of aspartic peptidases
API (Bacillus licheniformis) aspartic protease inhibitor (Bacillus licheniformis)
apigenin apigenin
apixaban apixaban
APMSF APMSF
apratastat apratastat
apstatin apstatin
Aptivus tipranavir
AQ-E5 small-molecule serine peptidase inhibitors
ARDP0006 ARDP0006
Arg-Arg-Gly-Cys peptide inhibitors of metallopeptidase
Arg-Lys-Asp-Val-Tyr thymopentin
Arg-Pro-Pro Arg-Pro-Pro
argatroban argatroban
arginine- or lysine-based inhibitor of aspartic peptidase arginine- or lysine-based inhibitor of aspartic peptidase
arginine- or lysine-based inhibitor of metallopeptidase arginine- or lysine-based inhibitor of metallopeptidase
arginine- or lysine-based inhibitors of cysteine peptidases arginine- or lysine-based inhibitors of cysteine peptidases
arginine- or lysine-based inhibitors of serine peptidases arginine- or lysine-based inhibitors of serine peptidases
argyrin A argyrin A
argyrin F peptide inhibitors of threonine peptidases
ARH067637 ARH067637
ARI-3099 ARI-3099
ARI-3531 ARI-3531
ARI-4175 small-molecule serine peptidase inhibitors
Aristra fondaparinux
Arixtra fondaparinux
ARM1 ARM1
ARNI LBQ657
ARP-100 small-molecule inhibitors of metallopeptidases
ARP101 ARP101
arphamenine A arphamenine A
arphamenine B arphamenine B
arylomycin arylomycin
arylomycin A2 arylomycin A2
arylomycin C16 arylomycin
arylomycin M131 arylomycin
arylsulfone inhibitors of metallopeptidases arylsulfone inhibitors of metallopeptidases
AS-101 compound AS-101 compound
AS111793 AS111793
AS2761325 small-molecule inhibitors of cysteine peptidases
AS2863995 small-molecule inhibitors of cysteine peptidases
Asp-Leu-Tyr-Asp-Gly-Trp-Lys-His-Glu-Ala-Glu-Cys-Ile aspartic protease inhibitor (Bacillus licheniformis)
Asp-Psi[PO(2)CH(2)]-LeuOH phosphorus-containing inhibitors of metallopeptidases
ASP4000 ASP4000
ASP8497 ASP8497
aspartic protease inhibitor (Bacillus licheniformis) aspartic protease inhibitor (Bacillus licheniformis)
assemblin dimerization inhibitor assemblin dimerization inhibitor
asteropterin asteropterin
astilbin (C60.006 inhbitor) polyphenol inhibitors of cysteine peptidases
asunaprevir asunaprevir
AT-125 acivicin
atazanavir atazanavir
ATBI bifunctional aspartic peptidase inhibitor (Bacillus sp.)
auranofin metal-containing inhibitor of cysteine peptidase (general)
aurintricarboxylic acid aurintricarboxylic acid
avagacestat BMS-708163
AVE-7688 ilepatril
avoralstat avoralstat
AX8819 AX8819
AZ-4217 small-molecule inhibitors of aspartic peptidases
AZ11557272 AZ11557272
AZ12606133 AZ12606133
AZ3971 small-molecule inhibitors of aspartic peptidases
azapeptide epoxides azapeptide epoxides
azapeptide halomethylketone peptidyl halomethane inhibitors of cysteine peptidases
azapeptide inhibitors of cysteine peptidases azapeptide inhibitors of cysteine peptidases
azapeptide inhibitors of hepacivirin azapeptide inhibitors of hepacivirin
azapeptide inhibitors of metallopeptidases azapeptide inhibitors of metallopeptidases
azapeptide inhibitors of serine peptidases azapeptide inhibitors of serine peptidases
azapro-3 azapro-3
AZD 0837 ARH067637
AZD-9668 AZD9668
AZD1236 AZD1236
AZD1446 AZD1446
AZD3293 lanabecestat
AZD3839 AZD3839
AZD4996 small-molecule inhibitors of cysteine peptidases
AZD5248 AZD5248
AZD6564 arginine- or lysine-based inhibitors of serine peptidases
AZD7986 small-molecule inhibitors of cysteine peptidases
AZD8165 AZD8165
AZD9668 AZD9668
AZD9684 AZD9684
AZD9819 small-molecule serine peptidase inhibitors
azepanone inhibitor of serine peptidase aldehyde- or ketone-related inhibitors of serine peptidases
azepanone inhibitors of cysteine peptidases azepanone inhibitors of cysteine peptidases
azetidin-2-one derivative inhibitors of cysteine peptidases azetidin-2-one derivative inhibitors of cysteine peptidases
azetidin-2-one derivative inhibitors of serine peptidases azetidin-2-one derivative inhibitors of serine peptidases
azido-Phe-Leu-Leu-4-aminomethyl-Phe-methyl vinyl sulfone LU-102
azidobestatin bestatin
aziridine derivatives aziridine derivatives
aziridinyl inhibitors of cysteine peptidases aziridinyl inhibitors of cysteine peptidases
AZM551248 small-molecule inhibitors of metallopeptidases
B
b-AP15 b-AP15
B27 peptide calpastatin peptide
B27-HYD B27-HYD
baceridin peptide inhibitors of threonine peptidases
bacitracin A bacitracin A
baicalin baicalin
BAL0019193 BAL0019193
balicatib balicatib
BAPA BAPA
batimastat batimastat
BAY 1142524 small-molecule serine peptidase inhibitors
BAY 59-7939 rivaroxaban
BAY 85-8501 BAY 85-8501
BAY-129566 BAY-129566
BAY-8040 small-molecule serine peptidase inhibitors
BB-1101 hydroxamate-containing inhibitors of metallopeptidases
BB-1101 BB-1101
BB-1909 hydroxamate-containing inhibitors of metallopeptidases
BB-2116 hydroxamate-containing inhibitors of metallopeptidases
BB-2293 hydroxamate-containing inhibitors of metallopeptidases
BB-2516 marimastat
BB-3103 BB3103
BB-94 batimastat
BB3103 BB3103
BCEAB BCEAB
BCH-2763 BCH-2763
BCX-3607 BCX-3607
BCX7353 small-molecule serine peptidase inhibitors
BDA-410 BDA-410
BDM14471 hydroxamate-containing inhibitors of metallopeptidases
BDM43079 small-molecule inhibitors of metallopeptidases
BDM43124 small-molecule inhibitors of metallopeptidases
BDM44768 small-molecule inhibitors of metallopeptidases
BE-1433 small-molecule inhibitors of metallopeptidases
BE113 small-molecule serine peptidase inhibitors
BE114 small-molecule serine peptidase inhibitors
BEA369 small-molecule inhibitors of aspartic peptidases
begacestat begacestat
belactosin A belactosin A
belactosin C belactosin A
beloranib beloranib
benarthin benarthin
benazepril (prodrug form) benazeprilat
benazeprilat benazeprilat
bengamide bengamide
benzamidine benzamidine
benzamidine derivatives benzamidine derivatives
benzoxazinones benzoxazinones
benzyloxycarbonyl-methionyl-2(S)-cyanopyrrolidine benzyloxycarbonyl-methionyl-2(S)-cyanopyrrolidine
benzylsuccinate benzylsuccinic acid
benzylsuccinic acid benzylsuccinic acid
benzylsulfonyl fluoride PMSF
benzylsulfonyl-D-Arg-Pro-4-amidinobenzylamide BAPA
benzylsulfonyl-d-arginine-proline-4-amidinobenzylamide peptide inhibitors of serine peptidases
benzylsulfonyl-D-Ser-Ser-4-amidinobenzylamide CJ-463
berenil (S01.151 inhibitor; M02.006 activator) berenil (S01.151 inhibitor; M02.006 activator)
bestatin bestatin
bestatin analogue SL-387 bestatin
bestatin dimethylaminoethyl ester LYP
bestatin, sulfur-containing analogues bestatin
beta-aminoacylpiperidine derivatives beta-aminoacylpiperidine derivatives
beta-lactam inhibitors of serine peptidases beta-lactam inhibitors of serine peptidases
beta-secretase inhibitors memapsin-2 inhibitors
beta-sultams beta-sultams
betrixaban betrixaban
betulinic acid betulinic acid
beverimat beverimat
BI 201302 small-molecule serine peptidase inhibitors
BI 201335 faldaprevir
BI-1356 linagliptin
BI-8S S01.217-binding aptamer
BIBR 1048 dabigatran
BIBR-953ZW prodrug dabigatran
BIBT986 BIBT986
bifunctional aspartic peptidase inhibitor (Bacillus sp.) bifunctional aspartic peptidase inhibitor (Bacillus sp.)
bifunctional aspartic protease inhibitor (Bacillus sp.) bifunctional aspartic peptidase inhibitor (Bacillus sp.)
BIL-DMK diazomethane inhibitor of cysteine peptidases BIL-DMK diazomethane inhibitor of cysteine peptidases
BILN-2061 BILN-2061
biotinyl-Arg-Gln-Arg-Arg-CH(2)Cl halomethane inhibitors of serine peptidases
bis-benzamidine benzamidine derivatives
bis[ethyl(2R, 3R)-3-[(S)-methyl-1-[4-(2,3,4-trimethoxyphenyl-methyl) piperazin-1-ylcarbonyl] butyl-carbonyl]oxiran-2-carboxylate]sulfate NCO-700
Bj-PRO-5a Bj-PRO-5a
BML-PI116-0005 Z-Leu-Leu-CHO
BMS-186282 BMS-186282
BMS-189090 BMS-189090
BMS-189664 BMS-189664
BMS-232632 atazanavir
BMS-262084 BMS-262084
BMS-275291 BMS-275291
BMS-289948 BMS-289948
BMS-299897 BMS-299897
BMS-363131 BMS-363131
BMS-433796 small-molecule inhibitors of aspartic peptidases
BMS-433796 BMS-433796
BMS-477118 saxagliptin
BMS-561389 razaxaban
BMS-561392 BMS-561392
BMS-562247 apixaban
BMS-56247 small-molecule serine peptidase inhibitors
BMS-605339 BMS-605339
BMS-650032 asunaprevir
BMS-708163 BMS-708163
BMS-740808 BMS-740808
BMS-890068 small-molecule serine peptidase inhibitors
BMS-906024 small-molecule inhibitors of aspartic peptidases
BMS-962212 small-molecule serine peptidase inhibitors
BMS186716 omapatrilat
BMS189921 BMS189921
BMV037 small-molecule inhibitors of threonine peptidases
BN 82204 BN 82204
BN82270 BN 82204
BNA-His-CAL-DCI PD125967
BO43 small-molecule serine peptidase inhibitors
Boc-(D)Val-Leu-(L)boroArg boron-containing inhibitors of serine peptidases
Boc-(R)-Leu-(S)-Pro-(S,S)-Azi(OBn)2 aziridine derivatives
Boc-(S)-Leu-(R)-Pro-(S,S)-Azi(OBn)2 aziridine derivatives
Boc-Asp(OMe)-CH(2)F (BAF) peptidyl halomethane inhibitors of cysteine peptidases
Boc-Asp(OMe)fluoromethane peptidyl halomethane inhibitors of cysteine peptidases
Boc-Asp-CMK Boc-Asp-CMK
Boc-Ile-Glu-Thr-Asp-H Ac-Ile-Glu-Thr-Asp-H
Boc-Val-Ile-(S)-4-amino-3-oxo-2, 2-difluoropentanoyl-Val-Ile-OMe aldehyde, glyoxal or ketone inhibitors of aspartic peptidases
boceprevir boceprevir
BOP 5-benzamido-2-benzyl-4-oxopentanoic acid
boro-Leu dipeptide boron-containing inhibitors of threonine peptidases
boron-containing inhibitors of aspartic peptidases boron-containing inhibitors of aspartic peptidases
boron-containing inhibitors of cysteine peptidases boron-containing inhibitors of cysteine peptidases
boron-containing inhibitors of metallopeptidases boron-containing inhibitors of metallopeptidases
boron-containing inhibitors of serine peptidases boron-containing inhibitors of serine peptidases
boron-containing inhibitors of threonine peptidases boron-containing inhibitors of threonine peptidases
bortezomib bortezomib
BP13944 small-molecule serine peptidase inhibitors
BP2109 small-molecule serine peptidase inhibitors
BPP 9alpha teprotide
bradykinin-potentiating peptides bradykinin-potentiating peptides
Brecanavir GW0385
Brecanvir GW0385
bromoacetyl, difluoroketone inhibitor of gamma-secretase bromoacetyl, difluoroketone inhibitor of gamma-secretase
bromoacetyl-D-arginine bromoacetyl-D-arginine
bromocriptine small-molecule serine peptidase inhibitors
BSc2118 BSc2118
BSc4999 BSc4999
BSF 409425 BSF 409425
BSI-IV small-molecule inhibitors of aspartic peptidases
BTZ bortezomib
Bu-2743E Bu-2743E
BU-32 BU-32
butabindide butabindide
BVM beverimat
BX528 BX528
BX5633 DX-9065a
Bz-Leu-Leu-Leu-COCHO Z-Leu-Leu-Leu-ketoaldehyde
Bz-Pro-Phe-boroArg-OH boron-containing inhibitors of serine peptidases
BZF961 small-molecule serine peptidase inhibitors
BzLLLCOCHO Z-Leu-Leu-Leu-ketoaldehyde
BZS benzylsuccinic acid
C
C000000956 small-molecule inhibitors of aspartic peptidases
C1239-PEG-Poly R small-molecule serine peptidase inhibitors
C20 C20
C23 C23
C2I C2I
CA030 epoxide inhibitors of cysteine peptidases
CA074 CA074
CA074 methyl ester CA074
CA074OMe CA074
CAA0225 CAA0225
CAA0255 small-molecule inhibitors of cysteine peptidases
Cabin-A1 peptide inhibitors of cysteine peptidases
Cabin-A2 peptide inhibitors of cysteine peptidases
caffeic acid phenyl ester caffeic acid phenyl ester
calpain inhibitor 2 ALLM
calpain inhibitor 3 MDL28170
calpain inhibitor I ALLN
calpain inhibitor II ALLM
calpain inhibitor III MDL28170
calpain inhibitor IV Z-Leu-Leu-Tyr-FMK
calpain inhibitor IV calpain inhibitor IV
calpain inhibitor VI calpain-inhibitors
calpain inhibitor VI SJA6017
calpain inhibitor XI AK295
calpain-inhibitors calpain-inhibitors
calpastatin peptide calpastatin peptide
calpeptin calpeptin
camostat mesilate camostat mesilate
candoxatril candoxatril
candoxatrilat candoxatril
CAPE caffeic acid phenyl ester
capsidin capsidin
captopril (XM02.001) captopril (XM02.001)
capzimin capzimin
carbamate or thiocarbamate inhibitors of serine peptidases carbamate or thiocarbamate inhibitors of serine peptidases
carboxylate-containing inhibitors of metallopeptidases carboxylate-containing inhibitors of metallopeptidases
carfilzomib carfilzomib
carmaphycin A carmaphycin A
carmaphycin B small-molecule inhibitors of threonine peptidases
carmaphycin B epoxide inhibitors of threonine peptidases
carmegliptin carmegliptin
carnostatine carnostatine
CAS108383-58-0 hydroxamate-containing inhibitors of metallopeptidases
caspase dimerization inhibitor caspase dimerization inhibitor
CAT0059 CAT0059
CAT811 CAT811
cathepsin G inhibitor I cathepsin G inhibitor I
cathepsin L inhibitor II Z-FY-CHO
cathepsin L inhibitor IV (Calbiochem) NapSul-Ile-Trp-CHO
cathepsin L inhibitor IV (Calbiochem) Z-Phe-Phe-fluoromethane
cathepsin L inhibitor Katunuma CLIK148
cathestatin epoxide inhibitors of cysteine peptidases
cavinafungin small-molecule serine peptidase inhibitors
CB 7969312 CB7969312
CB-12181 CB-12181
CB7967495 CB7967495
CB7969312 CB7969312
CBI CA074
CCT CCT
CD10847 small-molecule inhibitors of cysteine peptidases
CDDO small-molecule serine peptidase inhibitors
CDDO-Me CDDO-Me
CE-0266 CE-0266
CE-1037 CE-1037
celastrol celastrol
CEP-18770 delanzomib
CEP1612 CEP1612
cepafungin I small-molecule inhibitors of threonine peptidases
cephem derivative inhibitors of serine peptidases cephem derivative inhibitors of serine peptidases
CFZ carfilzomib
CGH728 CGH728
CGI1 cathepsin G inhibitor I
CGP 53820 CGP 53820
CGP-60536 aliskiren
CGP38560 CGP38560
CGS 14824 benazeprilat
CGS 24592 CGS 24592
CGS 25966 CGS 25966
CGS 26303 CGS 26303
CGS 26393 CGS 26393
CGS 30084 CGS 30084
CGS 34043 CGS 34043
CGS 35066 CGS 35066
CGS 35601 CGS 35601
CGS 37808 (prodrug) CGS 35601
CGS27023A CGS27023A
CH 1091 arginine- or lysine-based inhibitors of serine peptidases
CH 1500022 small-molecule inhibitors of aspartic peptidases
CH 248 arginine- or lysine-based inhibitors of serine peptidases
CH-2856 FE999024
CH-4215 FE999026
CH-5450 CH-5450
CH-66 CH-66
CH1104I CH1104I
CHA 5-caffeoylquinic acid
chelating inhibitors of metallopeptidases chelating inhibitors of metallopeptidases
chelating inhibitors of threonine peptidases chelating inhibitors of threonine peptidases
CHF5074 (gamma-secretase modulator) CHF5074 (gamma-secretase modulator)
chlorambucil chlorambucil
chlorambucil-L-Pro chlorambucil
chlorogenic acid 5-caffeoylquinic acid
p-chloromercuribenzoate PCMB
chloromethylketone halomethane inhibitors of serine peptidases
CHR-2797 (proinhibitor) CHR-79888
CHR-2863 CHR-2863
CHR-79888 CHR-79888
chromone chromone
chrysin polyphenol inhibitors of cysteine peptidases
chymostatin chymostatin
CI CI
CI-1028 LB30057
CI-1031 UK-356,202
CI-906 quinapril
cilastatin cilastatin
cilazapril cilazapril
cilazaprilat cilazapril
ciluprevir BILN-2061
cinnabaramides A-G (proteasome inhibitors) lactam inhibitors of proteasomes
CIP-13F CIP-13F
CIPPC small-molecule serine peptidase inhibitors
circinamide circinamide
CJ-1737 CJ-1737
CJ-463 CJ-463
CJ-672 CJ-672
CJ-697 3-amidinophenylalanine derivatives (S01.302 inhibitors)
CJ-730 3-amidinophenylalanine derivatives (S01.302 inhibitors)
CKD-731 fumagillin
CKD-732 CKD-732
clasto-lactacystin beta-lactone clasto-lactacystin beta-lactone
ClCH2CO-DL-(N-OH)Leu-Ala-Gly-NH2 ClCH2CO-DL-(N-OH)Leu-Ala-Gly-NH2
ClCH2CO-DL-(N-OH)Leu-OCH3 ClCH2CO-DL-(N-OH)Leu-OCH3
CLIK-060 CLIK-060
CLIK-066 CLIK-066
CLIK-071 CLIK-071
CLIK-072 CLIK-072
CLIK-088 CLIK-088
CLIK-112 CLIK-112
CLIK-121 CLIK-121
CLIK-162 CLIK-162
CLIK-163 CLIK-163
CLIK-164 CLIK-164
CLIK-166 CLIK-166
CLIK-181 CLIK-181
CLIK-185 CLIK-185
CLIK-187 CLIK-187
CLIK-195 CLIK-195
CLIK-60 CLIK-060
CLIK148 CLIK148
clioquinol clioquinol
clitocybin D clitocybin D
CLP Cys-Leu-Pro-Gly-His-Trp-Gly-Phe-Pro-Ser-Cys
CLT CLT
CMT-3 (M10.GNW-inhibitor) CMT-3 (M10.GNW-inhibitor)
cn-716 cn-716
CNP520 CNP520
COL-3 COL-3
compound 1 SB-3CT
Compound 1 AG7404
compound 2477 small-molecule inhibitors of cysteine peptidases
compound 2c compound 2c
compound 38u small-molecule inhibitors of cysteine peptidases
compound 49c (A01.023) inhibitor compound 49c (A01.023) inhibitor
compound 4cc small-molecule inhibitors of metallopeptidases
compound E compound E
compound Ii1 IDE inhibitor 1
compound s9 aziridine derivatives
converstatin peptide inhibitors of metallopeptidase
Coversyl arginine perindopril
CP-108,420 CP-108,420
CP-271485 CP-271485
CP-544439 CP-544439
CP-69,799 CP-69,799
CP-71,362 CP-71,362
CP-72,647 CP-72,647
CP-80,794 pseudo-peptide bond inhibitors of aspartic peptidases
CP-80794 CP-80794
CP-81,282 CP-81,282
CP113972 CP113972
CP1B-[4-23] calpastatin peptide
CPI-2081 CPI-2081
Cpp-Ala-Ala-Phe-pAb Cpp-Ala-Ala-Phe-pAb
Cpp-Leu-Trp Cpp-Leu-Trp
CRA-013783 L-235
CRA-2059 CRA-2059
CRA-9249 CRA-9249
Crixivan indinavir
crocapeptin (Chondromyces crocatus) peptide inhibitors of serine peptidases
CS peptide calpastatin peptide
CS-622 temocapril
CSI-75 CSI-75
CSN5i-3 small-molecule inhibitors of metallopeptidases
CT1418 hydroxamate-containing inhibitors of metallopeptidases
CTS-1027 RS-130830
CTS-1027 CTS-1027
CTS-21166 CTS-21166
CTS21166 CTS-21166
CU-2010 CU-2010
CU-2020 CU-2020
curcumin curcumin
CVS-3983 CVS-3983
CVS4441 aldehyde- or ketone-related inhibitors of serine peptidases
CWHM-117 small-molecule inhibitors of aspartic peptidases
CX295 AK295
cyanopeptolin cyanopeptolin
cyanopeptolin 954 cyanopeptolin
cyanopyrrolidide NVP-DPP728
cyanostatin A cyanostatin A
cyanostatin B cyanostatin B
cyclic peptide inhibitors of serine peptidases cyclic peptide inhibitors of serine peptidases
cyclic peptide inhibitors of threonine peptidases cyclic peptide inhibitors of threonine peptidases
cyclic sulfamide cyclic sulfamide
cyclic sulfamide gamma-secretase inhibitor gamma-secretase inhibitors
cyclic urea pseudo-peptide bond inhibitors of aspartic peptidases
cyclotheonamide E4 cyclotheonamide E4
cyclotheonellazole small-molecule serine peptidase inhibitors
CYGAK2 CYGAK2
Cyklokapron tranexamic acid
CYLA cysteic-leucyl-argininal
Cys-Leu-Pro-Gly-His-Trp-Gly-Phe-Pro-Ser-Cys Cys-Leu-Pro-Gly-His-Trp-Gly-Phe-Pro-Ser-Cys
Cys-Val-Thr-Pro-Ala-Leu-Arg peptide inhibitors of metallopeptidase
cystargamide B epoxide inhibitors of serine peptidases
cystargolide A lactam inhibitors of proteasomes
cystargolide B lactam inhibitors of proteasomes
cysteic-leucyl-argininal cysteic-leucyl-argininal
D
D-2-methyl-3-mercaptopropanoyl-L-Pro captopril (XM02.001)
D-420720 D-420720
d-alpha-aminopimelyl(1,1,1-trifluoro-3- amino)butan-2-one d-alpha-aminopimelyl(1,1,1-trifluoro-3- amino)butan-2-one
d-alpha-aminopimelyl(1,1,1-trifluoro-3-amino)butan-2-one halomethane inhibitors of serine peptidases
D-Arg-Oic-Pro-D-Ala-Phe(p-Me)-NH2 FM 19
D-His-Pro-Phe-His-Leu*Leu-Val-Tyr H.77
D-penicillamine D-penicillamine
D-Phe-Pro-Arg-CH(2)Cl PPACK
D-Phe-Pro-D-Arg-D-Thr-CONH2 D-Phe-Pro-D-Arg-D-Thr-CONH2
D-Val-Gly-Arg-CH(2)Cl D-Val-Gly-Arg-CH(2)Cl
D24 small-molecule inhibitors of metallopeptidases
D6R hexa-D-arginine
D9R nona-d-arginine amide
DA-1229 evogliptin
Dab-Pip Dab-Pip
dabigatran dabigatran
dabigatran etexilate dabigatran
daglutril SLV306
Daglutril SLV306
daidzein polyphenol inhibitors of serine peptidases
DAMPAQ-22 PAQ-22
DANLME DANLME
danoprevir danoprevir
daphnodorin daphnodorin
DAPT DAPT
Darexaban YM150
darunabir darunavir
darunavir darunavir
DC07090 small-molecule inhibitors of cysteine peptidases
DCG-04 biotinylated epoxide DCG-04 biotinylated epoxide
DCH 2,4-dichlorocinnamic acid hydroxamate
DCI DCI
DD2 assemblin dimerization inhibitor
dec-RRLL-chloromethylketone dec-RRLL-chloromethylketone
Dec-RVKR-CMK furin inhibitor 1
decanoyl-Arg-Val-Lys-Arg-chloromethane furin inhibitor 1
decanoyl-PTANA-CHO small-molecule serine peptidase inhibitors
delanzomib delanzomib
delaprilat delaprilat
deldeprevir small-molecule serine peptidase inhibitors
denagliptin denagliptin
DENKI PL265
DFK167 DFK167
DFP DFP
DG-051 DG-051
DG026 small-molecule inhibitors of metallopeptidases
DG35-VIII DG35-VIII
DH-12a small-molecule inhibitors of metallopeptidases
DHT1 small-molecule inhibitors of cysteine peptidases
1,3-di-(N-benzyloxycarbonyl-L-leucyl-L-leucyl)aminoacetone 1,3-di-(N-benzyloxycarbonyl-L-leucyl-L-leucyl)aminoacetone
diacyl hydroxamate hydroxamate-containing inhibitors of cysteine peptidases
diazo inhibitors of aspartic peptidases diazo inhibitors of aspartic peptidases
diazo inhibitors of cysteine peptidases diazo inhibitors of cysteine peptidases
diazo inhibitors of metallopeptidases diazo inhibitors of metallopeptidases
diazo inhibitors of serine peptidases diazo inhibitors of serine peptidases
diazo inhibitors of threonine peptidases diazo inhibitors of threonine peptidases
diazoacetyl-D,L-norleucine methyl ester DANLME
DIC19 calpastatin peptide
3,4-dichloroisocoumarin (DCI) DCI
didemnaketal B didemnaketal B
diethyl p-nitrophenyl phosphate phosphorus-containing inhibitors of serine peptidases
difluoroalcohol inhibitor of gamma-secretase gamma-secretase inhibitors
difluoroketone inhibitor of gamma-secretase gamma-secretase inhibitors
diisopropyl fluorophosphate (DFP) DFP
diisopropyl phosphonofluoridate DFP
diminazene aceturate berenil (S01.151 inhibitor; M02.006 activator)
dinghupeptin A small-molecule serine peptidase inhibitors
dipeptide boronic acid (DPBA) proteasome inhibitor boron-containing inhibitors of threonine peptidases
diphenyl 1-amino-2-phenylethylphosphonate phosphorus-containing inhibitors of serine peptidases
diphenyldiazomethane diazo inhibitors of aspartic peptidases
diprotin diprotin
diprotin A diprotin
diprotin B diprotin
disulfiram small-molecule inhibitors of cysteine peptidases
DIZE berenil (S01.151 inhibitor; M02.006 activator)
DJT06001 small-molecule serine peptidase inhibitors
DKFZ-633 peptide inhibitors of serine peptidases
dl-3-mercapto-2-benzylpropanoylglycine dl-3-mercapto-2-benzylpropanoylglycine
DMP323 DMP323
DMP450 DMP450
DNA or RNA aptamer effector of aspartic peptidase DNA or RNA aptamer effector of aspartic peptidase
DNA or RNA aptamer inhibitor of cysteine peptidase DNA or RNA aptamer inhibitor of cysteine peptidase
DNA or RNA aptamer inhibitor of metallopeptidase DNA or RNA aptamer inhibitor of metallopeptidase
DNA or RNA aptamer inhibitor of serine peptidase DNA or RNA aptamer inhibitor of serine peptidase
DNA or RNA aptamer inhibitor of threonine peptidase DNA or RNA aptamer inhibitor of threonine peptidase
DON 6-diazo-5-oxo-L-norleucylglycine
doxocycline tetracycline derivatives
doxycycline tetracycline derivatives
DPC 333 DPC 333
DPC 906 razaxaban
DPC-602 DPC-602
DPC423 DPC423
DPLG3 DPLG3
DS-1040 DS-1040
DS-8108b DS-8108b
DS1040 DS-1040
DSB beverimat
DSP-7238 small-molecule serine peptidase inhibitors
DSR-12727 DSR-12727
DTZ small-molecule serine peptidase inhibitors
DU 176b edoxaban
DU-1219 alacepril
DU-176 edoxaban
DU-176b edoxaban
DU176b edoxaban
dual enkephalinase inhibitor PL265
DuP 714 S18326
dutogliptin dutogliptin
DX-9065a DX-9065a
DX600 DX600
E
E-64 E64
E-76 peptide inhibitors of serine peptidases
E2072 E2072
E2609 small-molecule inhibitors of aspartic peptidases
E3024 E3024
E64 E64
E64-R-P-NH(2) E64-R-P-NH(2)
E64c Ep475
E64d E64d
EACA EACA
ebelactone A ebelactone A
ebelactone B ebelactone A
ebselen small-molecule inhibitors of cysteine peptidases
ebselen small-molecule inhibitors of metallopeptidases
EC27 EC27
EC33 EC33
edetic acid EDTA
edoxaban edoxaban
edoxaban tosylate edoxaban
EDTA EDTA
EF6265 EF6265
efegatran arginine- or lysine-based inhibitors of serine peptidases
EGTA EGTA
EH58 EH58
EI-1941-2 EI-1941-2
EL-17 small-molecule serine peptidase inhibitors
elasnin elasnin
Elaspol sivelestat
Elaspor sivelestat
elastatinal elastatinal
Eliquis apixaban
ELN318463 small-molecule inhibitors of aspartic peptidases
ELN475516 small-molecule inhibitors of aspartic peptidases
ELND006 ELND006
ELND007 ELND007
EMD 495235 EMD 495235
EMD 58265 EMD 58265
EMDB-1 EMDB-1
Emricasan PF3491390
EMS-275291 EMS-275291
enalapril enalapril
enalaprilat enalapril
enalkiren enalkiren
Entresto LBQ657
EOAI3402143 small-molecule inhibitors of cysteine peptidases
Ep-457 epoxide inhibitors of cysteine peptidases
Ep-459 epoxide inhibitors of cysteine peptidases
EP1013 Z-VD-FMK
EP217609 EP217609
EP42675 EP42675
Ep475 Ep475
epibestatin small-molecule serine peptidase inhibitors
epicoccalone epicoccalone
epigallocatechin-3-gallate polyphenol inhibitors of metallopeptidases
EPNP EPNP
epostatin epostatin
epoxide inhibitors of aspartic peptidases epoxide inhibitors of aspartic peptidases
epoxide inhibitors of cysteine peptidases epoxide inhibitors of cysteine peptidases
epoxide inhibitors of serine peptidases epoxide inhibitors of serine peptidases
epoxide inhibitors of threonine peptidases epoxide inhibitors of threonine peptidases
epoxomicin epoxomicin
epoxyketone inhibitors of threonine peptidases epoxide inhibitors of threonine peptidases
epoxysuccinate 8c epoxide inhibitors of cysteine peptidases
epsilon-aminocaproic acid (EACA) EACA
epsilon-aminohexanoic acid EACA
equisetin F01-221A
ER-319711 ER-319711
ER143 small-molecule serine peptidase inhibitors
eribaxaban eribaxaban
erythrosin B small-molecule serine peptidase inhibitors
ES-8891 small-molecule inhibitors of aspartic peptidases
esculetin esculetin
EST E64d
estatin A epoxide inhibitors of cysteine peptidases
estatin B epoxide inhibitors of cysteine peptidases
etacrynic acid t-butylamide inhibitor etacrynic acid t-butylamide inhibitor
ethylene glycol tetraacetic acid EGTA
ethylenediaminetetraacetic acid EDTA
N-ethylmaleimide NEM
1-ethylpyrrole-2,5-dione NEM
eurystatin eurystatin
evogliptin evogliptin
exanta melagatran
F
F-9775A small-molecule inhibitors of cysteine peptidases
F-9775B small-molecule inhibitors of cysteine peptidases
F01-221A F01-221A
F04W2166A pullularin C
F3A H3H derivative
F449 small-molecule inhibitors of metallopeptidases
F4H H3H derivative
F573 small-molecule inhibitors of cysteine peptidases
falcitidin falcitidin
faldaprevir faldaprevir
fasidotril fasidotril
fatty acid inhibitor of metallopeptidase fatty acid inhibitor of metallopeptidase
fatty acid inhibitors of aspartic peptidases fatty acid inhibitors of aspartic peptidases
fatty acid inhibitors of serine peptidases fatty acid inhibitors of serine peptidases
FE 999011 FE 999011
FE999024 FE999024
FE999026 FE999026
fellutamide B fellutamide B
fenchylamine sulfonamide fenchylamine sulfonamide
FG-2575 FG-2575
Fidexaban ZK-807834
FII phosphorus-containing inhibitors of metallopeptidases
FK-448 small-molecule serine peptidase inhibitors
FK-706 FK-706
flavone 3,3"-diamino-4"-methoxyflavone polyphenol inhibitors of proteasomes
flovagatran flovagatran
fluoroketone inhibitors of aspartic peptidases fluoroketone inhibitors of aspartic peptidases
fluoromethylketone halomethane inhibitors of serine peptidases
N-(4-fluorophenylsulfonyl)-L-valyl-L-leucinal SJA6017
fluorosalinosporamide fluorosalinosporamide
fluostatin A fluostatin A
fluostatin B fluostatin B
FM 19 FM 19
FMK halomethane inhibitors of serine peptidases
fmk peptidyl halomethane inhibitors of cysteine peptidases
FMK-9a peptidyl halomethane inhibitors of cysteine peptidases
FMPI (Streptomyces rishiriensis) phosphorus-containing inhibitors of metallopeptidases
FN-439 FN-439
fondaparinux fondaparinux
Fortovase saquinavir
Fosamprenavir (prodrug) amprenavir
fosinopril fosinopril
FOY gabexate mesilate
FOY007 gabexate mesilate
FOY305 camostat mesilate
Foypan camostat mesilate
FPRCH2Cl PPACK
fPrt D-Phe-Pro-D-Arg-D-Thr-CONH2
FR136706 FR136706
FR217840 FR217840
FR255031 FR255031
FR901277 FR901277
FR901451 FR901451
FR901533 FR901533
FT-9 small-molecule inhibitors of aspartic peptidases
FT671 FT671
FT827 FT827
fukugetin small-molecule inhibitors of cysteine peptidases
fumagalone fumagillin
fumagillin fumagillin
furin inhibitor 1 furin inhibitor 1
furin inhibitor 2 hexa-D-arginine
furin inhibitor I furin inhibitor 1
furin inhibitor II hexa-D-arginine
furoyl saccharin furoyl saccharin
FUT-175 nafamostat mesilate
FUT-187 sepimostat mesilate
FV-162 epoxide inhibitors of threonine peptidases
FXV673 otamixaban
FY01 FY01
G
G17905 G17905
G5 ubiquitin isopeptidase inhibitor compound 2c
Gabadur leupeptin
gabexate mesilate gabexate mesilate
GACFSIAHECGA peptide inhibitors of metallopeptidase
galardin galardin
gallinamide A gallinamide A
Galvus vildagliptin
gambogic acid gambogic acid
gamma-boroGlu boron-containing inhibitors of threonine peptidases
gamma-pyrone-3-acetic acid gamma-pyrone-3-acetic acid
gamma-secretase inhibitor 1 Z-Leu-Leu-Nle-H
gamma-secretase inhibitor II MW167
gamma-secretase inhibitor IX DAPT
gamma-secretase inhibitor XII gamma-secretase inhibitor XII
gamma-secretase inhibitor XII Z-Ile-Leu-CHO
gamma-secretase inhibitors gamma-secretase inhibitors
GB111-NH2 small-molecule inhibitors of cysteine peptidases
GC373 GC373
GC375 GC375
GC376 GC376
gemigliptin gemigliptin
gemopatrilat gemopatrilat
GEMSA GEMSA
genistein polyphenol inhibitors of serine peptidases
GFG-semicarbazone Gly-Phe-Gly-semicarbazone
GI254023X GI254023X
GL-189 GL-189
GL1001 MLN-4760
Glactiv sitagliptin
GlbA glidobactin A
glecaprevir glecaprevir
glidobactin A glidobactin A
gliotoxin gliotoxin
Gln-Arg-Phe-Ser-Arg opiorphin
globomycin globomycin
Glp-Asn-Pro-Tyr-Trp-Trp-NHMec Glp-Asn-Pro-Tyr-Trp-Trp-NHMec
Glu-boroPro Glu-boroPro
Glu-Gly-Arg-CH(2)Cl Glu-Gly-Arg-CH(2)Cl
Glu-Leu-Asp-Leu*Ala-Val-Glu-Phe OM00-3
Glu-Phe-Arg-CH(2)Cl Glu-Phe-Arg-CH(2)Cl
Glu-thiol Glu-thiol
Glu-Val-Asn-Leu*Ala-Ala-Glu-Phe OM99-2
glutamate phosphonate phosphorus-containing inhibitors of metallopeptidases
glutamate thiol Glu-thiol
Gly-Gly-Tyr(Bzl)-Arg Gly-Gly-Tyr(Bzl)-Arg
Gly-Phe-CHN2 Gly-Phe-diazomethane
Gly-Phe-diazomethane Gly-Phe-diazomethane
Gly-Phe-Gly-semicarbazone Gly-Phe-Gly-semicarbazone
Gly-Pro-Phe-(PO2CH2)-Gly-Pro-Nle phosphorus-containing inhibitors of metallopeptidases
glycolic acid carboxylate-containing inhibitors of metallopeptidases
glycoprilat small-molecule inhibitors of metallopeptidases
glycyrrhetinic acid small-molecule serine peptidase inhibitors
glyoxal, nitrile or semicarbazide inhibitors of serine peptidases glyoxal, nitrile or semicarbazide inhibitors of serine peptidases
GM6001 galardin
GNE-6640 small-molecule inhibitors of cysteine peptidases
GNE-6776 small-molecule inhibitors of cysteine peptidases
GNE-892 GNE-892
GNF6702 GNF6702
gosogliptin gosogliptin
GP205 small-molecule serine peptidase inhibitors
GPI 5693 GPI 5693
GPI5232 phosphorus-containing inhibitors of metallopeptidases
grassypeptolide A small-molecule serine peptidase inhibitors
grassystatin A grassystatin A
grassystatin B grassystatin A
grassystatin C grassystatin A
grassystatin D grassystatin A
grassystatin E grassystatin A
grassystatin F grassystatin A
grazoprevir grazoprevir
GRL-001 small-molecule inhibitors of cysteine peptidases
GRL-02031 GRL-02031
GRL-04810 GRL-04810
GRL-05010 GRL-05010
GRL-0519 GRL-0519
GRL-06579A GRL-06579A
GRL-0739 small-molecule inhibitors of aspartic peptidases
GRL-10413 small-molecule inhibitors of aspartic peptidases
GRL-1388 small-molecule inhibitors of aspartic peptidases
GRL-1398 small-molecule inhibitors of aspartic peptidases
GRL-142 GRL-142
GRL-216 small-molecule inhibitors of aspartic peptidases
GRL-286 small-molecule inhibitors of aspartic peptidases
GRL-4410A small-molecule inhibitors of aspartic peptidases
GRL-5010A small-molecule inhibitors of aspartic peptidases
GRL-8234 GRL-8234
GRL-98065 GRL-98065
GRL007 small-molecule inhibitors of aspartic peptidases
GRL008 GRL008
GS-8374 GS-8374
GS-9256 GS-9256
GS-9450 small-molecule inhibitors of cysteine peptidases
GS-9451 vedroprevir
GS-9857 voxilaprevir
GSI-953 begacestat
GSI-I Z-Leu-Leu-Nle-H
GSI-IX DAPT
GSI-XII gamma-secretase inhibitor XII
GSI1 Z-Leu-Leu-Nle-H
GSK188909 GSK188909
GSK2793660 GSK2793660
guanidinoethylmercaptosuccinic acid GEMSA
guanosine triphosphate SB 331750
GW-311616 GW-311616
GW0385 GW0385
GW280264X GW280264X
GW311616A GW-311616
GW3333 GW3333
GW433908 (prodrug) amprenavir
GW475151 GW475151
GW640385 GW0385
GW7647 GW7647
GW796406 GW796406
GW813893 GW813893
GW813893 small-molecule serine peptidase inhibitors
H
H-142 H-142
H-189 H-189
H-256 H-256
H-261 H-261
H-boronorleucine (pinacol) boron-containing inhibitors of serine peptidases
H.77 H.77
H17 (A02.001 inhbiitor) small-molecule inhibitors of aspartic peptidases
H376/95 melagatran
H3H derivative H3H derivative
HA08 HA08
HA28 DNA or RNA aptamer inhibitor of serine peptidase
haloacetyl amino acid amides haloacetyl amino acid amides
haloacetyl metallopeptidase inhibitor haloketone inhibitor of metallopeptidase
haloketone inhibitor of metallopeptidase haloketone inhibitor of metallopeptidase
halomethane inhibitors of serine peptidases halomethane inhibitors of serine peptidases
HBK001 HBK001
HBX 41,108 HBX 41,108
HBX41108 HBX 41,108
HBY-793 HBY-793
HD1 S01.217-binding aptamer
HD1-22 S01.217-binding aptamer
HD1-22 (S01.217 exosite ligand) small-molecule serine peptidase inhibitors
HD22 S01.217-binding aptamer
hemin hemin
hepin-13 hepin-13
heterocyclic acylating inhibitors of serine peptidases heterocyclic acylating inhibitors of serine peptidases
hexa-Arg hexa-D-arginine
hexa-arginine hexa-D-arginine
hexa-D-arginine hexa-D-arginine
hexa-D-arginine amide hexa-D-arginine
HFI419 HFI419
hinokiflavone polyphenol inhibitors of metallopeptidases
hispidin unclassified small-molecule inhibitors of peptidases
histargin histargin
HIV-Nmu HIV-Nmu
HMBA PCMB
HMBSA PCMB
HMR-3840 HMR-3840
HNSA HNSA
Hoe 498 ramipril
homocysteine homocysteine
HONHCOCH(iBu)CO-L-Ala-Gly-NH2 hydroxamate-containing inhibitors of metallopeptidases
HPI HPI
HWH-10d HWH-10d
Hxm-Phe-Arg-Gln (M12.217) hydroxamate-containing inhibitors of metallopeptidases
Hxm-Phe-Ser-Asn (M12.217 inhibitor hydroxamate-containing inhibitors of metallopeptidases
HY023016 (prodrug) dabigatran
hydroxamate-containing inhibitors of aspartic peptidases hydroxamate-containing inhibitors of aspartic peptidases
hydroxamate-containing inhibitors of cysteine peptidases hydroxamate-containing inhibitors of cysteine peptidases
hydroxamate-containing inhibitors of metallopeptidases hydroxamate-containing inhibitors of metallopeptidases
[(R)-3-(N-hydroxy)-carboxamido-2-benzylpropanoyl]-L-alanine kelatorphan
4-hydroxy-5,6-dihydro-2-pyrone derivative tipranavir
hydroxyethylene sulfone pseudo-peptide bond inhibitors of aspartic peptidases
p-hydroxymercuribenzenesulfonate PCMB
p-hydroxymercuribenzoate PCMB
I
I-432 MI-432
I5B2 phosphorus-containing inhibitors of metallopeptidases
IC260 small-molecule inhibitors of aspartic peptidases
icariin icariin
IcatC aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
ICI 186,756 ICI 186,756
ICI-200,880 ICI-200,880
ICI200355 halomethane inhibitors of serine peptidases
IDE inhibitor 1 IDE inhibitor 1
IDN-6556 PF3491390
IDN-8050 IDN-8050
IDN5370/CGP82630 small-molecule inhibitors of caspases
IDR-803 IDR-803
IDR-804 IDR-804
IDR-805 IDR-805
idrabiotaparinux idrabiotaparinux
idraparinux idraparinux
IDX316 small-molecule serine peptidase inhibitors
IDX320 IDX320
Ii1 hydroxamate-containing inhibitors of metallopeptidases
Ile-Pro-Ile diprotin
Ile-Pro-Pro bradykinin-potentiating peptides
ilepatril ilepatril
ilomastat galardin
imarikiren imarikiren
imidapril imidapril
imidaprilat imidapril
imigliptin imigliptin
IN973 small-molecule inhibitors of aspartic peptidases
INCB003619 INCB003619
INCB3619 INCB3619
Incivek telaprevir
indinavir indinavir
indolo-phakellin compound small-molecule inhibitors of threonine peptidases
inhibitor 24 inhibitor 24
inogatran arginine- or lysine-based inhibitors of serine peptidases
insulapeptolide small-molecule serine peptidase inhibitors
insulysin inhibitors insulysin inhibitors
invirase saquinavir
iodoacetamide iodoacetamide
2-iodoacetate iodoacetate
iodoacetate iodoacetate
iodotyrostatin tyrostatin
IPR19 small-molecule serine peptidase inhibitors
IPSI-001 IPSI-001
irreversible metallopeptidase inhibitors irreversible metallopeptidase inhibitors
isatin sulfonamide-based inhibitor of caspase isatin sulfonamide-based inhibitor of caspase
isatin-based inhibitors of cysteine peptidases isatin-based inhibitors of cysteine peptidases
isatoic anhydride isatin-based inhibitors of cysteine peptidases
isatoic anhydride heterocyclic acylating inhibitors of serine peptidases
isoleucyl-thiazolidide isoleucyl-thiazolidide
isosyringolin A syringolin A
isovaleric acid-D-His-L-Ile-L-Val-L-Pro-NH(2) falcitidin
isovaleryl-L-tyrosyl-L-valyl-DL-tyrosinal tyropeptin A
N-isovaleryl-tyrosyl-leucyl-tyrosinal tyrostatin
ITMN-191 danoprevir
ITMN-8187 ITMN-8187
IU1 IU1
IVA-His-Pro-Phe-His-CHS-Leu-Phe-NH2 L-364,099
IVDE77 small-molecule inhibitors of metallopeptidases
IVF N-iodoacetyl-valine-phenylalanine-amide
IW449 small-molecule inhibitors of metallopeptidases
ixazomib ixazomib
izenamide A pseudo-peptide bond inhibitors of aspartic peptidases
J
J94 small-molecule serine peptidase inhibitors
JA-2 JA-2
Januvia sitagliptin
JCP104 small-molecule serine peptidase inhibitors
JE-2147 KNI-764
JG-365 JG-365
JH3 small-molecule serine peptidase inhibitors
jizanpeptin small-molecule serine peptidase inhibitors
JJ1 small-molecule serine peptidase inhibitors
JK043 small-molecule inhibitors of cysteine peptidases
JLK isocoumarin JLK isocoumarin
JLK-6 JLK-6
JLK2 JLK isocoumarin
JMC08-4 small-molecule inhibitors of metallopeptidases
JMV 390-1 JMV 390-1
JMV1195 JMV1195
JMV2764 JMV2764
JMV4463 JMV4463
JNJ 10329670 JNJ 10329670
JNJ 27265732 JNJ 27265732
JNJ 40929837 JNJ 40929837
JNJ-10311795 RWJ-355871
JNJ-26993135 JNJ-26993135
JNJ-27390467 JNJ-27390467
JNJ-54861911 JNJ-54861911
JNJ-853346 small-molecule serine peptidase inhibitors
JNJ-9375 small-molecule serine peptidase inhibitors
JNJ0966 small-molecule inhibitors of metallopeptidases
JO146 JO146
JPM-OEt JPM-OEt
JS-1 JS-1
JTP-4819 JTP-4819
JTV-803 JTV-803
JW33 small-molecule inhibitors of aspartic peptidases
JW41 (A02.001 inhbiitor) small-molecule inhibitors of aspartic peptidases
JW46 (A02.001 inhbiitor) small-molecule inhibitors of aspartic peptidases
K
K-26 K-26
K-7174 K-7174
K11002 K11002
K11017 K11017
K11777 K777
K18v2 S01.232-binding aptamer
K32v2 S01.232-binding aptamer
K579 K579
K77111 K777
K777 K777
kalata B1 small-molecule serine peptidase inhibitors
Kall1-T4 r S01.212-binding aptamer
Kamei compound 18 hydroxamate-containing inhibitors of metallopeptidases
KB-R7785 KB-R7785
KBE009 small-molecule inhibitors of aspartic peptidases
kelatorphan kelatorphan
kempopeptin A ;kempopeptin B cyclic peptide inhibitors of serine peptidases
kempopeptin C cyclic peptide inhibitors of serine peptidases
kendomycin kendomycin
keto-ACE 5-S-5-benzamido-4-oxo-6-phenylhexanoyl-L-proline
keto-glutamine analogue keto-glutamine analogue
ketomethylene metallopeptidase inhibitors ketomethylene metallopeptidase inhibitors
ketomethylene peptide inhibitors ketomethylene peptide inhibitors
KF33955 belactosin A
KGP94 KGP94
KK1-300 ONO-KK1-300-01
KM(O(2))YR-H Lys-Met(sulfone)-Tyr-Arg-H
KMI-008 KMI-008
KMI-260 KMI-260
KMI-358 KMI-358
KMI-360 KMI-360
KMI-370 KMI-370
KMI-420 KMI-420
KMI-429 KMI-429
KMI-570 KMI-570
KMI-684 KMI-684
KNI-10006 KNI-10006
KNI-10033 KNI-10033
KNI-10075 KNI-10075
KNI-10127 KNI-10127
KNI-10161 KNI-10161
KNI-10166 KNI-10166
KNI-10333 pseudo-peptide bond inhibitors of aspartic peptidases
KNI-10343 pseudo-peptide bond inhibitors of aspartic peptidases
KNI-10395 pseudo-peptide bond inhibitors of aspartic peptidases
KNI-10516 KNI-10516
KNI-10740 pseudo-peptide bond inhibitors of aspartic peptidases
KNI-10742 pseudo-peptide bond inhibitors of aspartic peptidases
KNI-10743 pseudo-peptide bond inhibitors of aspartic peptidases
KNI-10774a KNI-10774a
KNI-10823 pseudo-peptide bond inhibitors of aspartic peptidases
KNI-1657 pseudo-peptide bond inhibitors of aspartic peptidases
KNI-272 kynostatin-272
KNI-577 KNI-577
KNI-764 KNI-764
kojistatin A kojistatin A
KR-62436 glyoxal, nitrile or semicarbazide inhibitors of serine peptidases
KR66222 KR66222
KR66223 KR66223
KRI-1314 KRI-1314
KRP-109 KRP-109
kunitzin-OS peptide inhibitors of serine peptidases
kunitzin-RE peptide inhibitors of serine peptidases
kushennol small-molecule inhibitors of cysteine peptidases
kynapcin small-molecule serine peptidase inhibitors
kynostatin-272 kynostatin-272
KYP-2047 KYP-2047
Kyprolis carfilzomib
KYT-1 KYT-1
KYT-36 KYT-36
KZ7088 vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases
KZR-504 epoxide inhibitors of threonine peptidases
KZR-616 epoxide inhibitors of threonine peptidases
L
L-006235 L-235
L-1037536 odanacatib
L-2,4-diaminobutyryl-piperidinamide Dab-Pip
L-2-amino-4-boronobutanoic acid ABBA
L-235 L-235
L-363,564 L-363,564
L-364,099 small-molecule inhibitors of aspartic peptidases
L-364,099 pseudo-peptide bond inhibitors of aspartic peptidases
L-364,099 L-364,099
L-375,378 L-375,378
L-658,758 L-658,758
L-659,286 L-659,286
L-659,286 elastase inhibitor beta-lactam inhibitors of serine peptidases
L-680,833 L-680,833
L-681,176 L-681,176
L-682,679 L-682,679
L-683,845 L-683,845
L-685,434 L-685,434
L-685,458 L-685,458
L-694,458 L-694,458
L-709,049 aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
L-709049 Ac-Tyr-Val-Ala-Asp-H
L-735,524 indinavir
L-833905 peptide isostere cysteine peptidase inhibitors
L-873724 L-873724
L-butaneboronic acid boron-containing inhibitors of metallopeptidases
L505 small-molecule inhibitors of aspartic peptidases
L646 small-molecule inhibitors of aspartic peptidases
L655,240 small-molecule inhibitors of aspartic peptidases
L659286 small-molecule serine peptidase inhibitors
lactacystin clasto-lactacystin beta-lactone
lactam inhibitors of proteasomes lactam inhibitors of proteasomes
lactam or lactone inhibitors of cysteine peptidases lactam or lactone inhibitors of cysteine peptidases
LAF237 vildagliptin
LAF389 bengamide
lanabecestat lanabecestat
lapstatin lapstatin
LB-30870 small-molecule serine peptidase inhibitors
LB-4b small-molecule inhibitors of metallopeptidases
LB30057 LB30057
LB30870 LB30870
LBQ657 LBQ657
LC15-0133 LC15-0133
LC15-0444 gemigliptin
LC53-0110 LC53-0110
LC53-0151 LC53-0110
LCZ696 LBQ657
LDD-1588 small-molecule inhibitors of cysteine peptidases
LDN-0021835 LDN-0021835
LDN-57444 LDN-57444
cyclo(-L-Leu-D-Phe-L-Pro-L-Phe-D-Leu-L-Val-) phepropeptin B
Leu-Leu-PheCH2Cl peptidyl halomethane inhibitors of cysteine peptidases
Leu-Phe-VS-CH3 vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases
Leu-Val-Val-Tyr-Pro-Trp-Thr spinorphin
leucinal leucinal
leucinethiol leucinethiol
leuhistin leuhistin
leupeptazin small-molecule inhibitors of cysteine peptidases
leupeptin leupeptin
leupyrrin B1 small-molecule serine peptidase inhibitors
LHVS LHVS
linagliptin linagliptin
lipopeptide peptide inhibitors of serine peptidases
lisinopril lisinopril
Lixiana edoxaban
LJNK small-molecule inhibitors of metallopeptidases
LK-732 arginine- or lysine-based inhibitors of serine peptidases
LK-733 LK-733
LL11 S01.217-binding aptamer
LLLLRVKR multi-Leu peptide
loggerpeptin peptide inhibitors of serine peptidases
lomofungin small-molecule inhibitors of metallopeptidases
lopinavir lopinavir
Lotensin benazeprilat
loxistatin E64d
LP-130 pseudo-peptide bond inhibitors of aspartic peptidases
LP-149 LP-149
LSEAL peptide LSEAL peptide
LTI-1 small-molecule inhibitors of metallopeptidases
LU-001 small-molecule inhibitors of threonine peptidases
LU-005i LU-005i
LU-015 small-molecule inhibitors of threonine peptidases
LU-102 LU-102
luteolin luteolin
LVLQTM LVLQTM
LVV-haemorphin 7 peptide inhibitors of metallopeptidase
LVV-hemorphin 7 LVV-hemorphin 7
LY-411,575 LY411575
LY-411575 LY411575
LY-570310 telaprevir
LY178550 LY178550
LY2434074 LY2434074
LY2811376 LY2811376
LY2886721 LY2886721
LY3000328 LY3000328
LY312340 LY312340
LY3314814 lanabecestat
LY411575 LY411575
LY450139 semagacestat
LY514962 alpha-ketoamide inhibitors of serine peptidases
LY517717 LY517717
LY52 LY52
lyngbyastatin lyngbyastatin
LYP LYP
LYP2 bestatin derivative bestatin
LYP3 LYP3
Lys-Ala chloromethyl ketone halomethane inhibitors of serine peptidases
Lys-Ala-Phe-Arg peptide inhibitors of metallopeptidase
Lys-Met(sulfone)-Tyr-Arg-H Lys-Met(sulfone)-Tyr-Arg-H
Lys[Z(NO2)]-pyrrolidide Lys[Z(NO2)]-pyrrolidide
Lys[Z(NO2)]-thiazolidide Lys[Z(NO2)]-thiazolidide
lysianadioic acid lysianadioic acid
lysinethiol lysinethiol
LZNP Lys[Z(NO2)]-pyrrolidide
LZNT Lys[Z(NO2)]-thiazolidide
M
M826 M826
M83 small-molecule serine peptidase inhibitors
M867 M867
MA-LF 2-mercaptoacetyl-L-leucyl-L-phenylalanine
macrocyclic inhibitor of aspartic peptidase macrocyclic inhibitor of aspartic peptidase
macrocyclic inhibitor of cysteine peptidase macrocyclic inhibitor of cysteine peptidase
macrocyclic inhibitor of serine peptidase macrocyclic inhibitor of serine peptidase
macrocyclic peptidomimetic macrocyclic inhibitor of aspartic peptidase
macyranone A small-molecule inhibitors of threonine peptidases
MALT-inhibitor 2 MALT-inhibitor 2
MAPI microbial alkaline proteinase inhibitor MAPI microbial alkaline proteinase inhibitor
marchantin M marchantin M
marimastat marimastat
Marizev omarigliptin
marizomib salinosporamide A
matlystatin A matlystatin A
matlystatin B matlystatin B
maturation inhibitor beverimat
MB21 small-molecule serine peptidase inhibitors
MBi-4 small-molecule inhibitors of aspartic peptidases
MCB3937 MCB3937
MCI-9038 argatroban
MD1 MD1
MD2 MD2
MD3 MD3
MD805 argatroban
MDCO-2010 small-molecule serine peptidase inhibitors
mdivi-1 small-molecule inhibitors of metallopeptidases
MDL 100173 MDL 100173
MDL 100240 (proinhibitor) MDL 100173
MDL 27,088 small-molecule inhibitors of metallopeptidases
MDL 27,788 small-molecule inhibitors of metallopeptidases
MDL104903 MDL104903
MDL201053 Z-FA-FMK
MDL28170 MDL28170
MDL73347 MDL73347
melagatran melagatran
melatonin melatonin
memapsin-2 inhibitors memapsin-2 inhibitors
MeOSuc-Ala-Ala-Ala-Pro-PheCH(2)Cl halomethane inhibitors of serine peptidases
MeOSuc-Ala-Ala-Pro-boroVal boron-containing inhibitors of serine peptidases
MeOSuc-Ala-Ala-Pro-Val-CH(2)Cl MeOSuc-Ala-Ala-Pro-Val-CH(2)Cl
mepazine mepazine
Mepentil thymopentin
mercaptoacyl amino acids mercaptoacyl amino acids
mercaptoacyldipeptides mercaptoacyldipeptides
Merck 662086 LDN-57444
Merck C gamma-secretase inhibitors
Merck L915 small-molecule inhibitors of metallopeptidases
Mesupron (prodrug) WX-UK1
metal ejectors metal ejectors
metal-abstraction peptide peptide inhibitors of metallopeptidase
metal-binding inhibitor of metallopeptidase chelating inhibitors of metallopeptidases
metal-containing inhibitor of aspartic peptidase (general) metal-containing inhibitor of aspartic peptidase (general)
metal-containing inhibitor of cysteine peptidase (general) metal-containing inhibitor of cysteine peptidase (general)
metal-containing inhibitor of metallopeptidase (general) metal-containing inhibitor of metallopeptidase (general)
metal-containing inhibitor of serine peptidase (general) metal-containing inhibitor of serine peptidase (general)
metal-containing inhibitor of threonine peptidase (general) metal-containing inhibitor of threonine peptidase (general)
metastat COL-3
methionine thiol PC18
4-methylumbelliferyl p-(NNN-trimethylammonium)cinnamate MUTMAC
4-methylumbelliferyl p-guanidinobenzoate MUGB
MF-480 aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
MG-101 ALLN
MG-262 MG-262
MG115 MG115
MG132 MG132
MGPA 2-mercaptomethyl-3-guanidinoethylthiopropanoic acid
MGTA 2-mercaptomethyl-3-guanidinoethylthiopropanoic acid
MI-1148 MI-1148
MI-2 MALT-inhibitor 2
MI-432 MI-432
MI-460 small-molecule serine peptidase inhibitors
Michael acceptor vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases
microcystin-LR small-molecule inhibitors of threonine peptidases
micropeptin micropeptin
microviridin microviridin
microviridin J microviridin
microviridin K microviridin
minocycline tetracycline derivatives
MIP-1232 small-molecule serine peptidase inhibitors
miraziridine A miraziridine A
mitoxantrone small-molecule inhibitors of cysteine peptidases
MIV-0711 small-molecule inhibitors of cysteine peptidases
MIV-247 small-molecule inhibitors of cysteine peptidases
MIV-711 MIV-711
MJ-24 small-molecule inhibitors of metallopeptidases
MK-0431 sitagliptin
MK-0626 MK-0626
MK-0674 MK-0674
MK-0752 MK-0752
MK-0822 odanacatib
MK-1220 MK-1220
MK-1256 MK-1256
MK-1597 MK-1597
MK-2748 MK-2748
MK-3102 omarigliptin
MK-421 enalapril
MK-422 enalapril
MK-431 sitagliptin
MK-4519 MK-4519
MK-5172 grazoprevir
MK-521 lisinopril
MK-626 MK-0626
MK-6325 MK-6325
MK-639 indinavir
MK-7009 vaniprevir
MK-8141 MK-8141
MK-822 odanacatib
MK-8718 small-molecule inhibitors of aspartic peptidases
MK-8831 small-molecule serine peptidase inhibitors
MK-8931 verubecestat
MK0791 cilastatin
MK351A MK351A
MKI talopeptin
ML132 ML132
ML188 ML188
ML300 small-molecule inhibitors of cysteine peptidases
ML323 ML323
ML345 small-molecule inhibitors of metallopeptidases
ML364 small-molecule inhibitors of cysteine peptidases
ML5 ML5
ML604440 small-molecule inhibitors of threonine peptidases
MLN-341 bortezomib
MLN-4760 MLN-4760
MLN-4924 small-molecule inhibitors of threonine peptidases
MLN2238 (pro-inhibitor) ixazomib
MLN273 (XT01.001 inibitor) MLN273 (XT01.001 inibitor)
MLN519 MLN519
MLN9708 ixazomib
MLT-827 MLT-827
MMI-166 MMI-166
MMI270 CGS27023A
MMP-8 inhibitor I MMP-8 inhibitor I
MMP-9i peptide inhibitors of metallopeptidase
MMP13i-A small-molecule inhibitors of metallopeptidases
MMP2/MMP9 inhibitor I small-molecule inhibitors of metallopeptidases
MMP2/MMP9 inhibitor II small-molecule inhibitors of metallopeptidases
MMP408 MMP408
MMPSI MMPSI
MNRC-5 MNRC-5
moexipril moexipril
moexiprilat moexipril
molassamide peptide inhibitors of serine peptidases
momordin Ic small-molecule inhibitors of cysteine peptidases
Mor-Phe-Nle-CHF-NME CP-81,282
morpholine-4-carboxylic acid (S)-1-[4-cyano-1-(3-morpholin-4-yl-propyl)-piperidin-4-ylcarbamoyl]-4,4-dimethyl-hexyl-amide small-molecule inhibitors of cysteine peptidases
morpholinurea-leucine-homophenylalanine-vinyl phenyl sulfone LHVS
MQPA argatroban
MR-889 MR-889
MRK-003 MRK-003
MRK-560 MRK-560
MRK003 MRK-003
MRT12113 small-molecule serine peptidase inhibitors
MS-560 small-molecule inhibitors of metallopeptidases
MTSET small-molecule inhibitors of cysteine peptidases
MUGB MUGB
multi-Leu peptide multi-Leu peptide
mupain-1 mupain-1
MUTMAC MUTMAC
MV026031 small-molecule inhibitors of cysteine peptidases
MV026630 MV026630
MV151 Ada-Ahx3-L3VS
MV201 epoxide inhibitors of cysteine peptidases
MVT-101 MVT-101
MW167 MW167
myricetin myricetin
myricetin polyphenol inhibitors of metallopeptidases
myxovirescin myxovirescin
N
N-(1-benzyl-2-carbamoyl-2-oxoethyl)-2-[E-2-(4-diethylaminomethylphenyl)ethen-1-yl]benzamide A-705253
N-(1-carbamoyl-1-oxohex-1-yl)-2-[E-2-(4-dimethylaminomethylphenyl)-ethen-1-yl]benzamide A-705239
N-(1-carboxy-3-phenylpropyl)-phenylalanyl-alpha-aspargine HPI
N-(2-chloroethyl)-N-methylphenylalanine haloketone inhibitor of metallopeptidase
N-(3-chloropropionyl)-L-phenylalanine N-(3-chloropropionyl)-L-phenylalanine
N-(3-Mercapto-5-methyl-1-oxohexyl)-l-phenylalanine C20
N-(4-morpholine)carbonyl-beta-(1-naphthyl)-l-alanine-l-leucine boronic acid MLN273 (XT01.001 inibitor)
N-(N-(1-carboxyl-3-phenylpropyl)-phe)-iso-ser, N-(N-(1-carboxyl-3-phenylpropyl)phenylalanyl)isoserine SCH39370
N-(pyridine-3-carbonyl)-Val-boroPro ARI-3531
N-(pyridine-4-carbonyl)-D-Ala-boroPro ARI-3099
N-[(R)-2-benzyl-5-cyano-4-oxopentanoyl]-L-phenylalanine irreversible metallopeptidase inhibitors
N-[2-(1-formyl-2-methyl-propyl)-1-(4-piperidin-1-ylbut-2-enoyl)-pyrrolidin-3-yl]-methane sulfonoamide GW-311616
N-[2-(2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethylamino)-2-methylpropyl]-2-methylpyrazolo[1,5-a]pyrimidine-6-carboxamide hydrochloride anagliptin
N-[N-(3,5-difluorophenylacetyl)-L-alanyl]-S-phenylglycine tbutyl ester DAPT
N-acetyl-isoleucyl-prolyl-phenylalaninal aldehyde- or ketone-related inhibitors of serine peptidases
N-acetyl-L-alanyl-L-alanyl-alpha-azaalanine p-nitrophenyl ester N-acetyl-L-alanyl-L-alanyl-alpha-azaalanine p-nitrophenyl ester
N-alkoxy-arylsulfonamide N-alkoxy-arylsulfonamide
N-benzyloxycarbonyl-prolyl-3-fluoropyrrolidine proline-based inhibitors of serine peptidases
N-benzyloxycarbonyl-prolyl-prolinal Z-Pro-Pro-H and similar inhibitors of prolyl oligopeptidase
N-benzyloxycarbonyl-thioprolyl-thioprolinal-dimethylacetal (ZTTA) Z-Pro-Pro-H and similar inhibitors of prolyl oligopeptidase
N-benzyloxycarbonyl-Val-Leu-leucinal Z-Val-Leu-Leu-H
N-bromoacetyl-D-leucylglycine N-bromoacetyl-D-leucylglycine
N-bromoacetyl-N-methyl-L-phenylalanine N-bromoacetyl-N-methyl-L-phenylalanine
N-bromosuccinimide small-molecule serine peptidase inhibitors
N-chloroacetyl-N-hydroxy-alpha-Phe-OMe haloketone inhibitor of metallopeptidase
N-chloroacetyl-N-hydroxy-beta-L-phenylalanine N-methylamide irreversible metallopeptidase inhibitors
N-chloroacetyl-N-hydroxy-beta-Phe-NHMe haloketone inhibitor of metallopeptidase
N-chloroacetyl-N-hydroxyleucine methyl ester haloketone inhibitor of metallopeptidase
N-ethoxycarbonyl-D-phenylalanyl-L-prolyl-alpha-azalysine p-nitrophenyl ester azapeptide inhibitors of serine peptidases
N-hydroxy-2-(naphthalene-2-ylsulfanyl)-acetamide HNSA
N-iodoacetyl-valine-phenylalanine-amide N-iodoacetyl-valine-phenylalanine-amide
N-isobutyl-N-[4-methoxyphenylsulfonyl]glycyl hydroxamic acid N-isobutyl-N-[4-methoxyphenylsulfonyl]glycyl hydroxamic acid
N-isovaleryl-tyrosyl-valyl-argininal strepin P-1
N-mercaptoacetyl-Phe-Tyr-amide N-mercaptoacetyl-Phe-Tyr-amide
N-methyl peptide reduced peptide bond inhibitors
N-phenethylphosphonyl-L-leucyl-L-tryptophane phosphoramidon
N-phenylmaleimide N-phenylmaleimide
N-piperazinyl-CO-Leu-Hph-VS-Ph APC3328
N-sulfamoyl-L-phenylalanine thiol inhibitors of metallopeptidases
N-l-(2(R,S)-carboxy-4-phenylbutyl)-cyclopentylcarbonyl-(S)-tryptophan CCT
N3 N3
NA101 small-molecule inhibitors of cysteine peptidases
nafamostat mesilate nafamostat mesilate
NAM-105 syrbactin analogue
NAM-93 syrbactin analogue
NAM-95 syrbactin analogue
namalide small-molecule inhibitors of metallopeptidases
NAPAP NAPAP
Naph-KKR-H Naph-KKR-H
napsagatran napsagatran
NapSul-Ile-Trp-CHO NapSul-Ile-Trp-CHO
narlaprevir narlaprevir
nazumamide A nazumamide A
nazumazole small-molecule serine peptidase inhibitors
NB-360 NB-360
NBS small-molecule serine peptidase inhibitors
NC-001 small-molecule inhibitors of threonine peptidases
NC-005 NC-005
NC-022 small-molecule inhibitors of threonine peptidases
NC-2300 NC-2300
NC002 epoxide inhibitors of threonine peptidases
NC002 epoxide inhibitors of threonine peptidases
NC2213 NC2213
NCO-700 NCO-700
ND-322 ND-322
ND-336 small-molecule inhibitors of metallopeptidases
ND-364 (metabolite of NS322) ND-322
ND-378 thiirane inhibitors of metallopeptidases
ND-478 (prodrug of ND-322) ND-322
nelfinavir nelfinavir
NEM NEM
NESS002ie NESS002ie
Neurodur leupeptin
NF arphamenine A
NF arphamenine B
NH(2)-(D-Arg)(9)-Val-Leu-Arg-CO-NHOH R9LF-1
NH(2)-CH-Ph-P(O)(OH)CH(2)-CH-CH(2)Ph(p-Ph)-CONH-CH-CH(3)-COOH(-) P8B
nickel pyrithione complex metal-containing inhibitor of cysteine peptidase (general)
Ninlaro ixazomib
Nip-Leu-Leu-LeuVS-Me Nip-Leu-Leu-LeuVS-Me
NITD679 small-molecule inhibitors of aspartic peptidases
NITD731 small-molecule inhibitors of aspartic peptidases
nitrile inhibitors of cysteine peptidases nitrile inhibitors of cysteine peptidases
nitrobenzyloxycarbonyl arginine chloromethylketone peptidyl halomethane inhibitors of cysteine peptidases
nitrobestatin bestatin
nitrogen mustard chlorambucil
nitroxoline nitroxoline
NK-1.8k NK-1.8k
NK-1.9k NK-1.9k
NK3201 NK3201
NLVS Nip-Leu-Leu-LeuVS-Me
NNGH N-isobutyl-N-[4-methoxyphenylsulfonyl]glycyl hydroxamic acid
nona-d-arginine amide nona-d-arginine amide
nona-L-arginine nona-L-arginine
norleucine1-angiotensin IV angiotensin IV
Norvir ritonavir
nostodione A nostodione A
nostopeptin BN920 peptide inhibitors of serine peptidases
nostosin A (Nostoc sp.) aldehyde- or ketone-related inhibitors of serine peptidases
nostosin B (Nostoc sp.) aldehyde- or ketone-related inhibitors of serine peptidases
NPGB NPGB
NPI-0047 salinosporamide B
NPI-0052 salinosporamide A
NPI52 NPI52
NPI64 aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
NPLT phosphoramidon
NS-134 NS-134
NS-629 NS-134
NSC 163501 acivicin
NSC 18508 small-molecule inhibitors of cysteine peptidases
NSC 251810 small-molecule inhibitors of cysteine peptidases
NSC 632839 NSC 632839
NSC 89167 small-molecule inhibitors of cysteine peptidases
NSC D750499 BU-32
NSC1011 small-molecule inhibitors of metallopeptidases
NSC13345 small-molecule inhibitors of cysteine peptidases
NSC185058 NSC185058
NSC48300 NSC48300
NSC635393 small-molecule serine peptidase inhibitors
NSITC NapSul-Ile-Trp-CHO
NTE-1 small-molecule inhibitors of metallopeptidases
NTE-2 small-molecule inhibitors of metallopeptidases
NU655 small-molecule inhibitors of aspartic peptidases
NVP-AHW700-NX NVP-AHW700-NX
NVP-DPP728 NVP-DPP728
NVP-LAF237 vildagliptin
NWL-117 vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases
NWL-154 vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases
O
OA-Hy small-molecule inhibitors of metallopeptidases
odanacatib odanacatib
OF4949 OF4949
Olysio simeprevir
OM00-3 OM00-3
OM99-2 OM99-2
Omapatrilat omapatrilat
omapatrilat omapatrilat
omarigliptin omarigliptin
omuralide clasto-lactacystin beta-lactone
Ondero linagliptin
Onglyza saxagliptin
ONO 3403 arginine- or lysine-based inhibitors of serine peptidases
ONO-4817 ONO-4817
ONO-5046 sivelestat
ONO-5334 ONO-5334
Ono-5435 sitagliptin
ONO-6818 ONO-6818
Ono-EI-600 Ono-EI-600
ONO-KK1-300-01 ONO-KK1-300-01
ONO-MI1-514 small-molecule inhibitors of metallopeptidases
ONO-MI1-570 small-molecule inhibitors of metallopeptidases
ONO-WH-236 small-molecule serine peptidase inhibitors
ONO3307 ONO3307
ONX 0914 ONX 0914
ONX0912 ONX0912
OP 1,10-phenanthroline
opiorphin opiorphin
oprozomib oprozomib
ortho-dihydrotanshinone small-molecule inhibitors of cysteine peptidases
oscillapeptin oscillapeptin
oscillarin oscillarin
OST-4077 OST-4077
otamixaban otamixaban
ovalicin fumagillin
ovalicin ovalicin
oxirane inhibitor epoxide inhibitors of cysteine peptidases
6-oxo-6-deoxyfumagillol fumagillin
P
p-(amidinophenyl)methanesulfonyl fluoride (p-APMSF) APMSF
P-1946 P-1946
p-aminobenzoate (PAMBA) PAMBA
p-bromophenacyl bromide p-bromophenacyl bromide
p-iodo-D-phenylalanine hydroxamate hydroxamate-containing inhibitors of metallopeptidases
P-Leu-Phe P-Leu-Phe
p-NH2-Bz-Gly-Pro-D-Leu-D-Ala-NHOH FN-439
p-nitrophenyl N2-acetyl-N1-benzylcarbazate p-nitrophenyl N2-acetyl-N1-benzylcarbazate
p-nitrophenyl-p"-guanidinobenzoate NPGB
P005091 P5091
P0217564 P5091
P045204 small-molecule inhibitors of cysteine peptidases
P12-3A peptide inhibitors of metallopeptidase
P217564 P217564
P22077 P22077
P32/98 isoleucyl-thiazolidide
P5091 P5091
P8B P8B
P9941 P9941
PA-457 beverimat
PAC-22 PAQ-22
paecilopeptin paecilopeptin
palmatine small-molecule serine peptidase inhibitors
PAMBA PAMBA
pancaspase inhibitor peptidyl halomethane inhibitors of cysteine peptidases
PAQ-22 PAQ-22
paritaprevir ABT-450
PC18 PC18
PCMB PCMB
PD 163594 PD 163594
PD 172524 LB30057
PD-129,541 cyclic peptide peptide inhibitors of aspartic peptidases
PD-130,328 PD-130,328
PD-135,040 (A01.017 inhbitor) PD-135,040 (A01.017 inhbitor)
PD-198961 PD-198961
PD0348292 eribaxaban
PD125967 PD125967
PD150606 PD150606
PD151746 PD151746
PD166793 hydroxamate-containing inhibitors of metallopeptidases
Pefabloc AEBSF
pentenocin B pentenocin B
pepstatin pepstatin
pepstatin A pepstatin
peptide fluoromethylketone peptidyl halomethane inhibitors of cysteine peptidases
peptide inhibitors of aspartic peptidases peptide inhibitors of aspartic peptidases
peptide inhibitors of cysteine peptidases peptide inhibitors of cysteine peptidases
peptide inhibitors of metallopeptidase peptide inhibitors of metallopeptidase
peptide inhibitors of serine peptidases peptide inhibitors of serine peptidases
peptide inhibitors of threonine peptidases peptide inhibitors of threonine peptidases
peptide isostere cysteine peptidase inhibitors peptide isostere cysteine peptidase inhibitors
peptide isostere inhibitors of serine peptidases peptide isostere inhibitors of serine peptidases
peptide IVYPW peptide IVYPW
peptide leucine arginine cyclic peptide inhibitors of serine peptidases
peptidyl cyclopropenone inhibitor of cysteine peptidase peptidyl cyclopropenone inhibitor of cysteine peptidase
peptidyl diazoethane diazo inhibitors of cysteine peptidases
peptidyl diazomethane diazo inhibitors of cysteine peptidases
peptidyl halomethane inhibitors of cysteine peptidases peptidyl halomethane inhibitors of cysteine peptidases
peptidyl halomethane inhibitors of threonine peptidases peptidyl halomethane inhibitors of threonine peptidases
peptidyl sulfonium salt peptidyl sulfonium salt
peptidyl-chloromethane halomethane inhibitors of serine peptidases
peptidyl-fluoromethane halomethane inhibitors of serine peptidases
perindopril perindopril
perindoprilat (proinhibitor) perindopril
PES_103 hydroxamate-containing inhibitors of metallopeptidases
PETIR-001 PETIR-001
PF-00356231 PF-00356231
PF-00734200 gosogliptin
PF-03084014 PF-3084014
PF-03491390 PF3491390
PF-04886847 PF-04886847
PF-3084014 PF-3084014
PF-429242 PF-429242
PF-5480090 small-molecule inhibitors of metallopeptidases
PF-734200 gosogliptin
PF152 PF152
PF3491390 PF3491390
PG-116800 PG-116800
PG394 small-molecule inhibitors of aspartic peptidases
PG418 small-molecule inhibitors of aspartic peptidases
PGI-02776 (prodrug of ZJ-43) ZJ-43
pGlu-Trp-Pro-Arg-Pro-Gln-Ile-Pro-Pro teprotide
Phe-Gly-H phenylalanylglycinal
phebestin phebestin
phenacein phenacein
o-phenanthroline 1,10-phenanthroline
1,10-phenanthroline 1,10-phenanthroline
1,10-phenanthroline-5,6-dione 1,10-phenanthroline
Phendione 1,10-phenanthroline
phenyl vinyl sulfone phenyl vinyl sulfone
phenylacetyl-Arg-Val-Arg-4-amidinobenzylamide phenylacetyl-Arg-Val-Arg-4-amidinobenzylamide
phenylalanylglycinal phenylalanylglycinal
phenylboronic acid boron-containing inhibitors of serine peptidases
phenylmethane sulfonylfluoride PMSF
phenylnorstatine inhibitor pseudo-peptide bond inhibitors of aspartic peptidases
phepropeptin cyclic peptide inhibitors of threonine peptidases
phepropeptin B phepropeptin B
phevalin phevalin
PhN 1,10-phenanthroline
phosphinate phosphorus-containing inhibitors of metallopeptidases
phosphinic acid phosphorus-containing inhibitors of metallopeptidases
phosphonate phosphorus-containing inhibitors of metallopeptidases
phosphonic acid phosphorus-containing inhibitors of metallopeptidases
2-(phosphonomethyl)pentanedioic acid PMPA
phosphoramidon phosphoramidon
phosphorus-containing inhibitors of aspartic peptidases phosphorus-containing inhibitors of aspartic peptidases
phosphorus-containing inhibitors of cysteine peptidases phosphorus-containing inhibitors of cysteine peptidases
phosphorus-containing inhibitors of metallopeptidases phosphorus-containing inhibitors of metallopeptidases
phosphorus-containing inhibitors of serine peptidases phosphorus-containing inhibitors of serine peptidases
phosphorus-containing inhibitors of threonine peptidases phosphorus-containing inhibitors of threonine peptidases
phosphoryl-L-leucyl-L-phenylalanine P-Leu-Phe
photoreactive inhibitors photoreactive inhibitors
PHX-1149T dutogliptin
PHX1149 PHX1149
PHX1766 PHX1766
PI-083 PI-083
PI-1840 PI-1840
pimozide pimozide
piperastatin piperastatin A
piperastatin A piperastatin A
piperlongumine small-molecule inhibitors of threonine peptidases
PIQ-22 PIQ-22
Piv-His-Pro-Phe-His-Leu-OH-Leu-Tyr-Tyr-Ser-NH2 CH-66
PK101 PK101
PKF241-466 small-molecule inhibitors of metallopeptidases
PKF242-484 small-molecule inhibitors of metallopeptidases
PKF275-055 PKF275-055
PKS21025 small-molecule inhibitors of threonine peptidases
PKS2104 small-molecule inhibitors of threonine peptidases
PKS21221 small-molecule inhibitors of threonine peptidases
PKS3080 small-molecule inhibitors of threonine peptidases
PKSI-527 PKSI-527
PL-100 PL-100
PL250 PL250
PL265 PL265
PL302 PL302
planktopeptin cyclic peptide inhibitors of serine peptidases
plasma kallikrein-binding aptamer S01.212-binding aptamer
plectasin plectasin
plectasin small-molecule serine peptidase inhibitors
Plummer"s inhibitor 2-mercaptomethyl-3-guanidinoethylthiopropanoic acid
PMPA PMPA
PMSF PMSF
PNASN-1 small-molecule serine peptidase inhibitors
PNU-140690 tipranavir
Pol 647 Pol 647
Pol 656 Pol 656
Poly R nona-L-arginine
polycresulen small-molecule serine peptidase inhibitors
polyhedral metallacarborane polyhedral metallacarborane
polyozellin small-molecule serine peptidase inhibitors
polyphenol inhibitors of aspartic peptidases polyphenol inhibitors of aspartic peptidases
polyphenol inhibitors of cysteine peptidases polyphenol inhibitors of cysteine peptidases
polyphenol inhibitors of metallopeptidases polyphenol inhibitors of metallopeptidases
polyphenol inhibitors of proteasomes polyphenol inhibitors of proteasomes
polyphenol inhibitors of serine peptidases polyphenol inhibitors of serine peptidases
poststatin poststatin
PPACK PPACK
PPI-2458 PPI-2458
PPNDS small-molecule inhibitors of metallopeptidases
PR-047 PR-047
PR-171 carfilzomib
PR-619 PR-619
PR-825 small-molecule inhibitors of threonine peptidases
PR-924 PR-924
PR-957 ONX 0914
PR3 epoxide inhibitors of threonine peptidases
PR39 peptide PR39 peptide
Pradaxa dabigatran
pralnacasan pralnacasan
prezista darunavir
Primaxin cilastatin
Prinivil lisinopril
Prinomastat Prinomastat
Pro-boroPro boron-containing inhibitors of serine peptidases
Pro-His-Pro-Phe-His-Sta-Val-Ile-His-Lys H-189
Pro-Leu-Gly-hydroxamate Pro-Leu-Gly-hydroxamate
Pro-Leu-Gly-NHOH Pro-Leu-Gly-hydroxamate
Pro-Phe-psi(PO2CH2)-Leu-Pro-NH2 phosphorus-containing inhibitors of metallopeptidases
Pro-Pro-diphenylphosphonate prodipine
Pro-Thr-Glu-Phe-R-Phe-Arg-Glu (R = -CH2NH-) H-256
probestin probestin
prodipine prodipine
proflavin proflavin
prohisin prohisin
proline-based inhibitor of metallopeptidase proline-based inhibitor of metallopeptidase
proline-based inhibitors of cysteine peptidases proline-based inhibitors of cysteine peptidases
proline-based inhibitors of serine peptidases proline-based inhibitors of serine peptidases
promazine small-molecule inhibitors of cysteine peptidases
propargyl-based cysteine peptidase inhibitors propargyl-based cysteine peptidase inhibitors
propeptin propeptin
propioxatin hydroxamate-containing inhibitors of metallopeptidases
propioxatin A propioxatin A
proprotein convertase propeptide-like peptide peptide inhibitors of serine peptidases
proteasome inhibitor 3 MG-262
proteasome inhibitor aldehydes proteasome inhibitor aldehydes
proteasome inhibitor I Z-Ile-Glu(OtBu)-Ala-Leu-H
proteasome inhibitor II Z-Leu-Leu-Phe-H
proteasome inhibitor III MG-262
PS-273 MLN273 (XT01.001 inibitor)
PS-519 MLN519
PS1 Z-Ile-Glu(OtBu)-Ala-Leu-H
PS341 bortezomib
pseudo-iodotyrostatin tyrostatin
pseudo-peptide bond inhibitors of aspartic peptidases pseudo-peptide bond inhibitors of aspartic peptidases
pseudo-tyrostatin tyrostatin
pseudoaeruginosin pseudoaeruginosin
pseudoaeruginosin NS1 pseudoaeruginosin
pseudoaeruginosin NS2 pseudoaeruginosin
pseudopeptide reduced peptide bond inhibitors
pseudopeptide threonine peptidase inhibitor pseudopeptide threonine peptidase inhibitor
PSI Z-Ile-Glu(OtBu)-Ala-Leu-H
PSI-3 MG-262
PSI-III MG-262
psysol 2 small-molecule serine peptidase inhibitors
PT-100 PT-100
PT-630 Glu-boroPro
PTL11028 PTL11028
pullularin C pullularin C
puromycin puromycin
purpurin small-molecule inhibitors of metallopeptidases
PW28 sulfonyl fluoride inhibitor of threonine peptidase
pyrizinostatin pyrizinostatin
pyroGlu-Lys-Trp-Ala-Pro Bj-PRO-5a
pyrrolidine inhibitor of metallopeptidase proline-based inhibitor of metallopeptidase
Q
Q-VD-OPh Q-VD-OPh
Q448 small-molecule serine peptidase inhibitors
QCBT7 small-molecule inhibitors of threonine peptidases
QGC001 (prodrug of EC33) EC33
Quadropril spirapril
QUB-F1 phosphorus-containing inhibitors of serine peptidases
QUB-TL1 small-molecule serine peptidase inhibitors
quercetin quercetin
quinapril quinapril
quinaprilat (proinhibitor) quinapril
quinoline-Val-Asp(OMe)-CH2-OPh Q-VD-OPh
quinolyl-valyl-O-methylaspartyl-[-2,6-difluorophenoxy]-methyl ketone Q-VD-OPh
quisqualic acid quisqualic acid
R
R-3032 R-3032
R-569 R-569
R-94138 R-94138
R7227 danoprevir
R9D-14 S01.217-binding aptamer
R9LF-1 R9LF-1
RA-14 small-molecule inhibitors of cysteine peptidases
RA-9 RA-9
RA190 small-molecule inhibitors of cysteine peptidases
RA36 S01.217-binding aptamer
racecadotril (prodrug) thiorphan
ramipril ramipril
ramiprilat ramipril
Rasilez aliskiren
razaxaban razaxaban
RB 101(S) RB 101(S)
RB 105 RB 105
RB 106 2-mercaptoacyl-dipeptides
RB006 S01.217-binding aptamer
RB104 RB104
RB150 (prodrug of EC33) EC33
RB25 RB25
RB3007 RB3007
RB3014 RB3014
RBx-0128 small-molecule serine peptidase inhibitors
RBx-0597 small-molecule serine peptidase inhibitors
RE31 S01.217-binding aptamer
RE31TBA S01.217-binding aptamer
Rebimastat BMS-275291
recursterol recursterol
reduced peptide bond inhibitor of aspartic peptidase pseudo-peptide bond inhibitors of aspartic peptidases
reduced peptide bond inhibitors reduced peptide bond inhibitors
regasepin1 small-molecule inhibitors of metallopeptidases
regasepin2 small-molecule inhibitors of metallopeptidases
relacatib relacatib
remikiren remikiren
Rendix dabigatran
Renormax spirapril
resveratrol resveratrol
retagliptin retagliptin
retropepsin dimerization inhibitors retropepsin dimerization inhibitors
retropepsin inhibitors retropepsin inhibitors
Revlimid small-molecule inhibitors of threonine peptidases
Reyataz atazanavir
RG7227 danoprevir
RID-F small-molecule inhibitors of threonine peptidases
ridaifen-F small-molecule inhibitors of threonine peptidases
Ridaura metal-containing inhibitor of cysteine peptidase (general)
ritonavir ritonavir
rivaroxaban rivaroxaban
RK-805 fumagillin
RK-805 RK-805
Ro 28-2653 Ro 28-2653
Ro 31-8472 Ro 31-8472
Ro 31-8959 saquinavir
Ro 32-7315 Ro 32-7315
Ro 42-5892 remikiren
Ro-1130830 RS-130830
RO-206-0222 small-molecule inhibitors of metallopeptidases
RO1 RO1
RO200-1770 RO200-1770
Ro31-9790 Ro31-9790
Ro32-3555 Ro32-3555
RO4929097 RO4929097
RO5444101 RO5444101
RO5459072 RO5459072
RO5461111 small-molecule inhibitors of cysteine peptidases
Roche 28-2653 Ro 28-2653
ronastat nafamostat mesilate
RPR120844 RPR120844
RPR209685 RPR209685
RR-11a RR-11a
RRGF peptide inhibitors of metallopeptidase
RS-10085 moexipril
RS-130830 RS-130830
RS-5139 temocapril
RSV resveratrol
RTD-1 peptide inhibitors of metallopeptidase
RTS-V5 small-molecule inhibitors of threonine peptidases
rugosin B polyphenol inhibitors of serine peptidases
rugosin E polyphenol inhibitors of serine peptidases
rupintrivir rupintrivir
ruprintrivir rupintrivir
ruthenium compound metal-containing inhibitor of cysteine peptidase (general)
ruviprase peptide inhibitors of serine peptidases
RWJ-355871 RWJ-355871
RWJ-445167 RWJ-445167
RWJ-51084 RWJ-51084
RWJ-51438 RWJ-51438
RWJ-56423 RWJ-56423
RWJ-671818 RWJ-671818
RXP-470.1 RXP-470.1
RXP03 RXP03
RXP401 phosphorus-containing inhibitors of metallopeptidases
RXP401 RXP401
RXP407 RXP407
RXPA380 RXPA380
RYM1 hydroxamate-containing inhibitors of metallopeptidases
S
S-2209 S-2209
S-3304 S-3304
S-allyl-L-cysteine small-molecule inhibitors of cysteine peptidases
S-nitrosothiol compounds S-nitrosothiol compounds
S-PI pepstatin
S01.140-binding aptamer DNA or RNA aptamer inhibitor of serine peptidase
S01.212-binding aptamer S01.212-binding aptamer
S01.213-binding aptamer DNA or RNA aptamer inhibitor of serine peptidase
S01.217-binding aptamer S01.217-binding aptamer
S01.232-binding aptamer S01.232-binding aptamer
S136492 small-molecule inhibitors of metallopeptidases
S17092 S17092
S18326 S18326
S19825 Z-Pro-Pro-H and similar inhibitors of prolyl oligopeptidase
S21402 RB 105
S35972 small-molecule serine peptidase inhibitors
SA898 SA898
sacubitril (prodrug of M13.001 inhibitor LBQ657) LBQ657
SAK-1 SAK-1
SAK1 SAK-1
salinosporamide A salinosporamide A
salinosporamide B salinosporamide B
salinosporamides D-J (proteasome inhibitors) lactam inhibitors of proteasomes
salsolinol small-molecule inhibitors of threonine peptidases
salvianolic acid B small-molecule inhibitors of metallopeptidases
SAN9812 carnostatine
saquinavir saquinavir
SAR1 small-molecule serine peptidase inhibitors
SAR107375 small-molecule serine peptidase inhibitors
SAR114137 small-molecule inhibitors of cysteine peptidases
SAR164653 small-molecule serine peptidase inhibitors
Savaysa edoxaban
saxagliptin saxagliptin
SB 331750 SB 331750
SB-3CT SB-3CT
SB-462795 relacatib
SB-553484 SB-553484
SB203238 SB203238
SB216357 (inhibitor of signal peptidase I) beta-lactam inhibitors of serine peptidases
SC-22716 SC-22716
SC-39026 fatty acid inhibitors of serine peptidases
SC-57461A SC-57461A
SC-78080 small-molecule inhibitors of metallopeptidases
SC080 small-molecule inhibitors of metallopeptidases
SC68896 SC68896
SC81956 SC81956
SCH 32615 SCH 32615
SCH 33844 spirapril
SCH 34826 SCH 34826
SCH 39370 SCH39370
SCH 42354 SCH 42354
SCH 42495 (prodrug of SCH 42354) SCH 42354
SCH 503034 boceprevir
SCH 697466 SCH 697466
SCH 900229 SCH 900229
SCH 900518 narlaprevir
SCH 900567 small-molecule inhibitors of metallopeptidases
SCH-39370 SCH39370
SCH1682496 small-molecule inhibitors of aspartic peptidases
SCH212986 aldehyde- or ketone-related inhibitors of serine peptidases
SCH215426 aldehyde- or ketone-related inhibitors of serine peptidases
SCH39370 SCH39370
SCH446211 SCH6
SCH47896 SCH47896
SCH48446 SCH48446
SCH567312 alpha-ketoamide inhibitors of serine peptidases
SCH6 SCH6
SCO-272 imarikiren
scutellarin scutellarin
scyptolin scyptolin
scytonemide A scytonemide A
SD-2590 small-molecule inhibitors of metallopeptidases
SD-7300 small-molecule inhibitors of metallopeptidases
SD146 SD146
SDMI-1 peptide inhibitors of serine peptidases
SDMI-2 peptide inhibitors of serine peptidases
SDZ 224-015 SDZ 224-015
SDZ283-910 SDZ283-910
secapin peptide inhibitors of serine peptidases
SEL2711 SEL2711
SEL2770 SEL2770
selenium-containing inhibitors of metallopeptidases selenium-containing inhibitors of metallopeptidases
semagacestat semagacestat
sepimostat mesilate sepimostat mesilate
sepin-1 sepin-1
sepinostat mesilate sepimostat mesilate
Ser-Trp-Phe-Pro Ser-Trp-Phe-Pro
SF-1902 A5 SF-1902 A5
SF2809 VI SF2809E
SF2809E SF2809E
SG85 SG85
shishicrellastatin A small-molecule inhibitors of cysteine peptidases
shishicrellastatin B small-molecule inhibitors of cysteine peptidases
SHR117887 SHR117887
SI-591 small-molecule inhibitors of cysteine peptidases
sialorphin sialorphin
silanediol inhibitors of aspartic peptidases silanediol inhibitors of aspartic peptidases
silanediol inhibitors of metallopeptidases silanediol inhibitors of metallopeptidases
silanediol inhibitors of serine peptidases silanediol inhibitors of serine peptidases
silicaptopril captopril (XM02.001)
silybin silybin
simeprevir simeprevir
Sintomodulina thymopentin
siomycin A siomycin A
sirtinol small-molecule serine peptidase inhibitors
sitagliptin sitagliptin
sitagliptun sitagliptin
Sivelestat Ono-EI-600
sivelestat sivelestat
SJA6017 SJA6017
SJB3-019A small-molecule inhibitors of cysteine peptidases
SKF 107457 SKF 107457
SKF 108738 SKF 108738
SLV-306 SLV306
SLV306 SLV306
SLV338 SLV338
SM-19712 SM-19712
SM-25453 hydroxamate-containing inhibitors of metallopeptidases
SM-319777 KNI-764
small-molecule inhibitors of aspartic peptidases small-molecule inhibitors of aspartic peptidases
small-molecule inhibitors of caspases small-molecule inhibitors of caspases
small-molecule inhibitors of cysteine peptidases small-molecule inhibitors of cysteine peptidases
small-molecule inhibitors of glutamic peptidases small-molecule inhibitors of glutamic peptidases
small-molecule inhibitors of metallopeptidases small-molecule inhibitors of metallopeptidases
small-molecule inhibitors of peptidases of unspecified catalytic type small-molecule inhibitors of peptidases of unspecified catalytic type
small-molecule inhibitors of threonine peptidases small-molecule inhibitors of threonine peptidases
small-molecule serine peptidase inhibitors small-molecule serine peptidase inhibitors
SNJ-1715 SNJ-1715
SNJ-1757 SNJ-1757
SNJ-1945 SNJ-1945
SNJ-2008 aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
SOL1 SOL1
sophoraflavanone G small-molecule inhibitors of cysteine peptidases
sovaprevir small-molecule serine peptidase inhibitors
Sovriad simeprevir
SP2086 retagliptin
spautin-1 small-molecule inhibitors of cysteine peptidases
SPF-32629 SPF-32629
SPF-32629A SPF-32629
SPF-32629B SPF-32629
SPI-15 small-molecule inhibitors of threonine peptidases
spinorphin spinorphin
spirapril spirapril
SPL-707 small-molecule inhibitors of aspartic peptidases
spongiacidin C small-molecule inhibitors of cysteine peptidases
SPP 635 small-molecule inhibitors of aspartic peptidases
SPP100 aliskiren
spumigin E spumigin E
SQ 14,603 SQ 14,603
SQ 14225 captopril (XM02.001)
SQ 20 881 teprotide
SQ 20,881 teprotide
SQ 24,798 SQ 24,798
SQ 28,603 SQ 28,603
SQ-28603 SQ-28603
SQ14225 captopril (XM02.001)
SR 26831 SR 26831
SR173 hydroxamate-containing inhibitors of aspartic peptidases
SRD44 small-molecule inhibitors of metallopeptidases
SRI 31215 SRI 31215
SsCEI 4 SsCEI 4
SSM-1 SSM-1
SSR182289A SSR182289A
SSR69071 SSR69071
staccopin P1 aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
staccopin P2 aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
statine derivative pseudo-peptide bond inhibitors of aspartic peptidases
stigonemapeptin small-molecule serine peptidase inhibitors
strepin P-1 strepin P-1
streptonigrin small-molecule inhibitors of cysteine peptidases
streptopeptolin cyanopeptolin
SUAM 1221 SUAM 1221
SUAM-14746 SUAM-14746
suberanilohydroxamic acid suberone derivative
suberone derivative suberone derivative
suc-AAPF-CMK Suc-Ala-Ala-Pro-Phe-CH(2)Cl
Suc-Ala-Ala-Pro-Phe-CH(2)Cl Suc-Ala-Ala-Pro-Phe-CH(2)Cl
Suc-Val-Pro-PheP(OPh)2 Suc-Val-Pro-PheP(OPh)2
Suganon evogliptin
sulfonamide inhibitors of metallopeptidases sulfonamide inhibitors of metallopeptidases
sulfonyl fluoride sulfonylating inhibitors of serine peptidases
sulfonyl fluoride inhibitor of threonine peptidase sulfonyl fluoride inhibitor of threonine peptidase
sulfonyl hydroxamate inhibitors of metallopeptidases sulfonyl hydroxamate inhibitors of metallopeptidases
sulfonylating inhibitors of serine peptidases sulfonylating inhibitors of serine peptidases
sulfur-containing inhibitors of cysteine peptidases sulfur-containing inhibitors of cysteine peptidases
sulfur-containing inhibitors of serine peptidases sulfur-containing inhibitors of serine peptidases
sulindac sulfide sulindac sulfide
sulphonamide sulfonamide inhibitors of metallopeptidases
sulphostin sulphostin
SUN13834 SUN13834
SWFP Ser-Trp-Phe-Pro
SylA syringolin A
symplocamide A symplocamide A
symplostatin 4 small-molecule inhibitors of cysteine peptidases
symplostatin 5 small-molecule serine peptidase inhibitors
SYR-322 alogliptin
SYR-472 trelagliptin
SYR-472 small-molecule serine peptidase inhibitors
syrbactin analogue syrbactin analogue
syringolin A syringolin A
T
t-Boc-His-Pro-Phe-His-LeuOHVal-Ile-His H-261
t-plasminogen activator-binding aptamer S01.232-binding aptamer
T06 small-molecule inhibitors of cysteine peptidases
TA-6366 imidapril
TAK-070 small-molecule inhibitors of aspartic peptidases
TAK-100 TAK-100
TAK-272 imarikiren
TAK-272 small-molecule inhibitors of aspartic peptidases
TAK442 TAK442
talabostat PT-100
talopeptin talopeptin
Tanatril imidapril
Tanomastat BAY-129566
tanshinone IIA sulfonic sodium small-molecule inhibitors of cysteine peptidases
TAPI TAPI
TAPI-0 TAPI
TAPI-1 TAPI-1
TAPI-2 TAPI-2
tasiamide F small-molecule inhibitors of aspartic peptidases
Tat-microCL peptide HIV-Nmu
Tat2 peptide peptide inhibitors of threonine peptidases
TBL(4)K 1,3-di-(N-benzyloxycarbonyl-L-leucyl-L-leucyl)aminoacetone
TBODA TBODA
TBTIF thiol inhibitors of metallopeptidases
TCH-013 small-molecule inhibitors of threonine peptidases
TCH-13 small-molecule inhibitors of threonine peptidases
TCMDC-134379 small-molecule serine peptidase inhibitors
TD-0212 small-molecule inhibitors of metallopeptidases
TEI-5624 TEI-5624
TEI-6344 TEI-6344
TEI-8362 TEI-8362
TEI-E548 TEI-E548
TEI-F00806 small-molecule serine peptidase inhibitors
teicoplanin small-molecule inhibitors of cysteine peptidases
telaprevir telaprevir
temocapril temocapril
temocaprilat temocapril
teneligliptin teneligliptin
teprotide teprotide
terrein small-molecule inhibitors of threonine peptidases
Tesavel sitagliptin
tetracycline derivatives tetracycline derivatives
tetrandine small-molecule inhibitors of threonine peptidases
tetrathionate sulfur-containing inhibitors of cysteine peptidases
TG-0205221 TG-0205221
TGN-255 flovagatran
thalassospiramide vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases
thiirane gelatinase inhibitor thiirane inhibitors of metallopeptidases
thiirane inhibitors of cysteine peptidases thiirane inhibitors of cysteine peptidases
thiirane inhibitors of metallopeptidases thiirane inhibitors of metallopeptidases
thimerosal metal-containing inhibitor of metallopeptidase (general)
thiol inhibitors of metallopeptidases thiol inhibitors of metallopeptidases
thiolutin chelating inhibitors of metallopeptidases
thioridazine small-molecule inhibitors of cysteine peptidases
thiorphan thiorphan
thiostrepton thiostrepton
thrombin-binding aptamer S01.217-binding aptamer
Thromstop NAPAP
thymopentin thymopentin
thysanone thysanone
TILAEIKNINAD SsCEI 4
tipranavir tipranavir
TIR-199 syrbactin analogue
TIR-203 XT01.001 inhibitor) TIR-203 XT01.001 inhibitor)
TJK002 small-molecule serine peptidase inhibitors
TL-3 TL-3
TLCK TLCK
TM5275 small-molecule serine peptidase inhibitors
TMC-126 TMC-126
TMC-86A epoxide inhibitors of threonine peptidases
TMC-86B epoxide inhibitors of threonine peptidases
TMC-95 TMC-95
TMC-95A TMC-95
TMC-95B TMC-95
TMC-95C TMC-95
TMC-95D TMC-95
TMC-96 epoxide inhibitors of threonine peptidases
TMC114 darunavir
TMC126 TMC-126
TMC240 TMC240
TMC310911 TMC310911
TMC435 simeprevir
TMC435350 simeprevir
TMI-002 small-molecule inhibitors of metallopeptidases
TMI-005 apratastat
TMI-1 TMI-1
TMI-2 TMI-2
TNP-470 fumagillin
TNP-470 TNP-470
TOP 3-thienylalanine-ornithyl-proline
TOP-008 TOP-008
Tos-LysCH(2)Cl TLCK
Tos-PheCH(2)Cl TPCK
tosedostat CHR-79888
TP-110 TP-110
TP5 thymopentin
TPC-806 small-molecule serine peptidase inhibitors
TPCK TPCK
TPI2155 small-molecule inhibitors of metallopeptidases
Tra-Phe-APAA PKSI-527
Tradjenta linagliptin
Trajenta linagliptin
trandolapril trandolapril
trandolaprilat trandolapril
tranexamic acid tranexamic acid
trans-chalcone polyphenol inhibitors of cysteine peptidases
trelagliptin trelagliptin
trichloro(dioxoethylene-O,O") tellurate AS-101 compound
trifluoroacetyl-peptide inhibitors of elastases trifluoroacetyl-peptide inhibitors of elastases
trifluoromethylketone halomethane inhibitors of serine peptidases
triptolide small-molecule inhibitors of metallopeptidases
triterpenoid C-28 methyl ester CDDO-Me
trivaric acid small-molecule serine peptidase inhibitors
tropolone derivative chelating inhibitors of metallopeptidases
Trp-Leu-Trp-vinylsulfone Trp-Leu-Trp-vinylsulfone
TS-021 TS-021
tsukubachelin peptide inhibitors of metallopeptidase
TTP889 TTP889
tumor necrosis factor-alpha protease inhibitor TAPI
tumor necrosis factor-alpha protease inhibitor-1 TAPI-1
tumor necrosis factor-alpha protease inhibitor-2 TAPI-2
TXA tranexamic acid
TY-51076 TY-51076
TY-51184 TY-51184
TY-51469 TY-51469
tynorphin peptide inhibitors of metallopeptidase
tynorphin tynorphin
Tyr-Phe-hydroxamate Tyr-Phe-hydroxamate
Tyr-Phe-NHOH Tyr-Phe-hydroxamate
Tyr-Pro-D-Ala-NH2 peptide inhibitors of serine peptidases
Tyr-Pro-DClPhe-Phe-NH(2) EMDB-1
tyropeptin A tyropeptin A
tyropeptin B proteasome inhibitor aldehydes
tyropeptin B tyropeptin A
tyropeptin-boronic acid tyropeptin-boronic acid
tyropeptin-boronic acid derivative AS-06 tyropeptin-boronic acid
tyropeptin-boronic acid derivative AS-29 tyropeptin-boronic acid
tyrostatin tyropeptin A
tyrostatin tyrostatin
tyrphostin AG 537 small-molecule serine peptidase inhibitors
U
U 71038 U 71038
U-42,126 acivicin
U-81749 U-81749
U-89360E peptide inhibitors of aspartic peptidases
UAMC00039 UAMC00039
Ubal ubiquitin aldehyde
Ubenimex bestatin
ubiquitin aldehyde ubiquitin aldehyde
ubiquitin vinyl sulfone ubiquitin vinyl sulfone
Ucf-101 Ucf-101
UIC-94017 darunavir
UIC-PI UIC-PI
UK 156,406 UK 156,406
UK-101 UK101
UK-356,202 UK-356,202
UK-370106 carboxylate-containing inhibitors of metallopeptidases
UK-383,367 UK-383,367
UK-396082 UK-396082
UK-69,578 candoxatril
UK-73,967 candoxatril
UK-79,300 candoxatril
UK101 UK101
unclassified small-molecule inhibitors of peptidases unclassified small-molecule inhibitors of peptidases
undecadene-dioic acid bis-[2-(3H-imidazol-4-yl)-ethyl]-amide (S 30372) metal ejectors
unsaturated ester vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases
upain-1 upain-1
upain-2 upain-2
upamostat (prodrug) WX-UK1
urea-linkage inhibitor reduced peptide bond inhibitors
ursolic acid small-molecule serine peptidase inhibitors
V
VA999272 small-molecule serine peptidase inhibitors
Val-boro-Pro PT-100
Val-D-Leu-Pro-Phe-Phe-Val-D-Leu peptide inhibitors of aspartic peptidases
Val-Pro-Leu diprotin
Val-Pro-Pro bradykinin-potentiating peptides
Val-Val-Tyr-Pro-Trp tynorphin
valistatin valistatin
valproic acid small-molecule serine peptidase inhibitors
Vanihep vaniprevir
vaniprevir vaniprevir
VBY-825 vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases
vedroprevir vedroprevir
VEL-0230 VEL-0230
Velcade bortezomib
verubecestat verubecestat
VIa small-molecule inhibitors of aspartic peptidases
vialinin A vialinin A
vibralactone vibralactone
Victrelis boceprevir
Vidupiprant small-molecule inhibitors of cysteine peptidases
vildagliptin vildagliptin
vinyl sulfone vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases
vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases
vinyl sulfone or other Michael acceptor inhibitors of serine peptidases vinyl sulfone or other Michael acceptor inhibitors of serine peptidases
vinyl sulfone or other Michael acceptor inhibitors of threonine peptidases vinyl sulfone or other Michael acceptor inhibitors of threonine peptidases
Viracept (nelfinavir mesylate) nelfinavir
VL-01 small-molecule inhibitors of threonine peptidases
VLX1570 VLX1570
VOX voxilaprevir
voxilaprevir voxilaprevir
VR23 small-molecule inhibitors of threonine peptidases
VRT-018858 VRT-018858
VTI-1002 small-molecule serine peptidase inhibitors
VTP-27999 VTP-27999
VX-166 VX-166
VX-740 pralnacasan
VX-765 VX-765
VX478 amprenavir
VX950 telaprevir
W
WAY-151693 WAY-151693
WAY-281418 WAY-281418
wedelolactone small-molecule inhibitors of threonine peptidases
WEHD-fmk vinyl sulfone or other Michael acceptor inhibitors of serine peptidases
WEHI-842 WEHI-842
WEHI-916 small-molecule inhibitors of aspartic peptidases
WF14861 epoxide inhibitors of cysteine peptidases
WF14865 epoxide inhibitors of cysteine peptidases
WIN 67694 acyloxymethane derivatives
withaferin A withaferin A
witharefin small-molecule inhibitors of threonine peptidases
WLW-vs Trp-Leu-Trp-vinylsulfone
WP1130 WP1130
WRR-666 vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases
WRR-669 vinyl sulfone or other Michael acceptor inhibitors of cysteine peptidases
WRR483 WRR483
WS 79089B FR901533
WS75624 A WS75624 A
WS75624 B WS75624 B
WS79089B FR901533
WX-FX4 WX-FX4
WX-UK1 WX-UK1
WXC-340 WXC-340
WYK-1 small-molecule serine peptidase inhibitors
X
Xarelto rivaroxaban
ximelagatran (prodrug of melagatran) melagatran
XK263 XK263
XL081 small-molecule inhibitors of metallopeptidases
XL188 small-molecule inhibitors of cysteine peptidases
XL784 XL784
XM323 XM323
Y
Y-29794 Y-29794
Y-40613 Y-40613
Y-41654 small-molecule inhibitors of metallopeptidases
YD-3 small-molecule serine peptidase inhibitors
YHJ-7-52 YHJ-7-52
YM-60828 YM-60828
YM-96765 YM-96765
YM150 YM150
YO-01027 YO-01027
YO-2 YO-2
YS-980 YS-980
YSY-01A YSY-01A
YU-102 small-molecule inhibitors of threonine peptidases
YU101 YU101
Z
Z-321 Z-321
Z-AEVD-FMK Z-AEVD-FMK
Z-Ala-Ala-AzaAsn epoxycarboxylate ethyl ester Z-Ala-Ala-AzaAsn epoxycarboxylate ethyl ester
Z-Ala-Ala-AzaAsn-chloromethylketone AJN-230
Z-Ala-Ala-Phe-glyoxal glyoxal, nitrile or semicarbazide inhibitors of serine peptidases
Z-Ala-Ala-Phe-glyoxal aldehyde, glyoxal or ketone inhibitors of aspartic peptidases
Z-Ala-Ala-Phe-H Z-Ala-Ala-Phe-H
z-Ala-Ile-boronic acid z-Ala-Ile-boronic acid
Z-Ala-Pro-Phe-glyoxal glyoxal, nitrile or semicarbazide inhibitors of serine peptidases
Z-Ala-Pro-Phe-H aldehyde- or ketone-related inhibitors of serine peptidases
Z-Arg-Leu-Arg-alpha-aza-glycyl-Ile-Val-OMe Z-Arg-Leu-Arg-alpha-aza-glycyl-Ile-Val-OMe
Z-Asp(OMe)-Glu(OMe)-Val-Asp(OMe)-fluoromethyl ketone Z-DEVD-FMK
Z-Asp(OMe)-Ile-Pro-Asp(OMe)-FMK peptidyl halomethane inhibitors of cysteine peptidases
Z-AVLQ-CN aldehyde, ketone, glyoxal, or semicarbazone inhibitors of cysteine peptidases
Z-DEVD-FMK Z-DEVD-FMK
Z-FA-FMK Z-FA-FMK
Z-FKck acyloxymethylketone C25.001 inhibitor
Z-FL-COCHO ZFL
Z-FY(t-Bu)-DMK Z-Phe-Tyr(OBut)-CHN(2)
Z-FY-CHO Z-FY-CHO
Z-GlyP-L-Leu-L-Leu Z-GlyP-L-Leu-L-Leu
Z-IETD-FMK Z-IETD-FMK
Z-IL(OtBu)AL-H Z-Ile-Glu(OtBu)-Ala-Leu-H
Z-IL-CHO gamma-secretase inhibitor XII
Z-Ile-Glu(OtBu)-Ala-Leu-H Z-Ile-Glu(OtBu)-Ala-Leu-H
z-Ile-Leu-CHO gamma-secretase inhibitor XII
Z-Ile-Leu-CHO Z-Ile-Leu-CHO
Z-L-L-Y-CHN2 diazo inhibitors of cysteine peptidases
Z-L-PheP-L-Leu-L-Ala Z-L-PheP-L-Leu-L-Ala
Z-LEHD-FMK Z-LEHD-FMK
Z-Leu-Abu-CONH-CH2-C6H3(3, 5-(OMe)2 C2I
Z-Leu-Leu-CHO Z-Leu-Leu-CHO
Z-Leu-Leu-Leu-B(OH)2 Z-Leu-Leu-Leu-B(OH)2
Z-Leu-Leu-Leu-FMK Z-Leu-Leu-Leu-FMK
Z-Leu-Leu-Leu-ketoaldehyde Z-Leu-Leu-Leu-ketoaldehyde
Z-Leu-Leu-Leu-vinylsulfone Z-Leu-Leu-Leu-vinylsulfone
Z-Leu-Leu-leucinal MG132
Z-Leu-Leu-LeuVS Z-Leu-Leu-Leu-vinylsulfone
z-Leu-Leu-Nle-CHO Z-Leu-Leu-Nle-H
Z-Leu-Leu-Nle-H Z-Leu-Leu-Nle-H
Z-Leu-Leu-norvalinal MG115
Z-Leu-Leu-Phe-H Z-Leu-Leu-Phe-H
Z-Leu-Leu-Tyr-CHN2 diazo inhibitors of cysteine peptidases
Z-Leu-Leu-Tyr-FMK Z-Leu-Leu-Tyr-FMK
Z-Leu-Lys-CHN2 diazo inhibitors of serine peptidases
Z-Leu-Nle-H calpeptin
(Z-LL)(2) ketone 1,3-di-(N-benzyloxycarbonyl-L-leucyl-L-leucyl)aminoacetone
Z-LVG-CHN2 diazo inhibitors of cysteine peptidases
Z-Lys-COCHO aldehyde- or ketone-related inhibitors of serine peptidases
Z-Lys-H aldehyde- or ketone-related inhibitors of serine peptidases
Z-Phe-(PO2CH2)-Ala-Lys-Ser phosphorus-containing inhibitors of metallopeptidases
Z-Phe-Ala-CH(2)F Z-FA-FMK
Z-Phe-Ala-CMK peptidyl halomethane inhibitors of cysteine peptidases
Z-Phe-Ala-diazomethane Z-Phe-Ala-diazomethane
Z-Phe-Ala-FMK Z-FA-FMK
Z-Phe-Arg-diazomethane Z-Phe-Arg-diazomethane
Z-Phe-Lys-2,4,6-trimethylbenzoyloxymethylketone trifluoroacetate acyloxymethylketone C25.001 inhibitor
Z-Phe-Lys-acyloxymethylketone acyloxymethylketone C25.001 inhibitor
Z-Phe-Phe-diazomethane Z-Phe-Phe-diazomethane
Z-Phe-Phe-fluoromethane Z-Phe-Phe-fluoromethane
Z-Phe-Phe-fluoromethyl ketone Z-Phe-Phe-fluoromethane
Z-Phe-Phe-FMK Z-Phe-Phe-fluoromethane
Z-Phe-Tyr (OBut)-COCHO Z-FY-CHO
Z-Phe-Tyr(OBut)-CHN(2) Z-Phe-Tyr(OBut)-CHN(2)
Z-Pro Z-Pro
Z-Pro-Pro-H and similar inhibitors of prolyl oligopeptidase Z-Pro-Pro-H and similar inhibitors of prolyl oligopeptidase
Z-Pro-Prolinal Z-Pro-Pro-H and similar inhibitors of prolyl oligopeptidase
Z-RLVG-CHN2 diazo inhibitors of cysteine peptidases
Z-Ser-Ser-Gln-Nle-(boro)-Leu Z-Ser-Ser-Gln-Nle-(boro)-Leu
Z-Tyr(I)-Ala-CHN2 diazo inhibitors of cysteine peptidases
Z-Val-Ala-Asp(OMe)-fluoromethylketone ZVAD-FMK
Z-Val-Asn-Ser-Thr-Leu-Gln-chloromethane Z-Val-Asn-Ser-Thr-Leu-Gln-chloromethane
Z-Val-Leu-Leu-H Z-Val-Leu-Leu-H
Z-Val-Lys-H aldehyde- or ketone-related inhibitors of serine peptidases
Z-Val-Phe-H MDL28170
Z-VD-FMK Z-VD-FMK
Z-VDVAD-FMK Z-VDVAD-FMK
Z-VRPR-FMK Z-VRPR-FMK
Z-YVAD-fmk peptidyl halomethane inhibitors of cysteine peptidases
Z13752A Z13752A
Zafatek trelagliptin
zafirlukast small-molecule serine peptidase inhibitors
ZAIB z-Ala-Ile-boronic acid
zankiren zankiren
ZBG chelating inhibitors of metallopeptidases
ZD-0892 ZD-0892
ZD-8321 ZD-8321
Zemiglo gemigliptin
Zestril lisinopril
zFFfmk Z-Phe-Phe-fluoromethane
ZFL ZFL
ZFPLA Z-L-PheP-L-Leu-L-Ala
ZGN-440 beloranib
ZGPLL Z-GlyP-L-Leu-L-Leu
ZHAWOC5135 small-molecule inhibitors of metallopeptidases
ZHAWOC5684 small-molecule inhibitors of metallopeptidases
ZI-10 small-molecule inhibitors of aspartic peptidases
zinc-binding inhibitor of metallopeptidase chelating inhibitors of metallopeptidases
Zincov Zincov
ZJ-11 small-molecule inhibitors of metallopeptidases
ZJ-17 small-molecule inhibitors of metallopeptidases
ZJ-43 ZJ-43
ZK-807834 ZK-807834
ZK824859 arginine- or lysine-based inhibitors of serine peptidases
ZL(3)VS Z-Leu-Leu-Leu-vinylsulfone
ZL3B Z-Leu-Leu-Leu-B(OH)2
ZL3VS Z-Leu-Leu-Leu-vinylsulfone
ZLDI-8 small-molecule inhibitors of metallopeptidases
zLLL Z-Leu-Leu-Leu-FMK
zLLY-fmk Z-Leu-Leu-Tyr-FMK
zofenopril zofenopril
ZRLR Z-Arg-Leu-Arg-alpha-aza-glycyl-Ile-Val-OMe
ZVAD-FMK ZVAD-FMK
zVAM.fmk peptidyl halomethane inhibitors of cysteine peptidases
zVLL-CHO Z-Val-Leu-Leu-H
ZY15557 small-molecule serine peptidase inhibitors
ZYDPLA1 small-molecule serine peptidase inhibitors
{
4-[(4-arsonophenyl)methyl]phenylarsonic acid NSC48300