Small-molecule inhibitor: LB30057
Name
- Common name
- LB30057
- Other names
- CI-1028; PD 172524
Inhibition
- Peptidases inhibited
- thrombin
- Mechanism
- A potent and reversible, selective inhibitor of thrombin. Ki = 0.38 nM for human thrombin, Ki = 3290 nM for bovine trypsin (Oh et al. 1998).
Chemistry
- CID at PubChem
- 56603774
- Structure
- Formula weight
- 494
![[LB30057 (S01.217 inhibitor) structure ]](http://pubchem.ncbi.nlm.nih.gov/image/imgsrv.fcgi?t=l&cid=56603774)
Properties
- Synthesis
- Kim et al. 2006
