Literature for peptidase C01.075: cruzipain

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2019
1. Barbosa da Silva,E., Dall,E., Briza,P., Brandstetter,H. and Ferreira,R.S.
   Cruzain structures: apocruzain and cruzain bound to S-methyl thiomethanesulfonate and implications for drug design
   Acta Crystallogr F Struct Biol Commun (2019) 75, 419-427. PubMed  Europe PubMed DOI  S
2018
2. Giroud,M., Dietzel,U., Anselm,L., Banner,D., Kuglstatter,A., Benz,J., Blanc,J.B., Gaufreteau,D., Liu,H., Lin,X., Stich,A., Kuhn,B., Schuler,F., Kaiser,M., Brun,R., Schirmeister,T., Kisker,C., Diederich,F. and Haap,W.
   Repurposing a library of human cathepsin L ligands: identification of macrocyclic lactams as potent rhodesain and Trypanosoma brucei inhibitors
   J Med Chem (2018) 61, 3350-3369. PubMed  Europe PubMed DOI  S  I
2013
3. Assis,D.M., Gontijo,V.S., de Oliveira Pereira,I., Santos,J.A., Camps,I., Nagem,T.J., Ellena,J., Izidoro,M.A., Dos Santos Tersariol,I.L., de Barros,N.M., Doriguetto,A.C., Dos Santos,M.H. and Juliano,M.A.
   Inhibition of cysteine proteases by a natural biflavone: behavioral evaluation of fukugetin as papain and cruzain inhibitor
   J Enzyme Inhib Med Chem (2013) 28, 661-670. PubMed  Europe PubMed DOI  S  I
2012
4. Lee,G.M., Balouch,E., Goetz,D.H., Lazic,A., McKerrow,J.H. and Craik,C.S.
   Mapping inhibitor binding modes on an active cysteine protease via nuclear magnetic resonance spectroscopy
   Biochemistry (2012) 51, 10087-10098. PubMed  Europe PubMed DOI  E  S  I
2010
5. Mott,B.T., Ferreira,R.S., Simeonov,A., Jadhav,A., Ang,K.K., Leister,W., Shen,M., Silveira,J.T., Doyle,P.S., Arkin,M.R., McKerrow,J.H., Inglese,J., Austin,C.P., Thomas,C.J., Shoichet,B.K. and Maloney,D.J.
   Identification and optimization of inhibitors of trypanosomal cysteine proteases: cruzain, rhodesain, and TbCatB
   J Med Chem (2010) 53, 52-60. PubMed  Europe PubMed DOI  S  I
2009
6. Bryant,C., Kerr,I.D., Debnath,M., Ang,K.K., Ratnam,J., Ferreira,R.S., Jaishankar,P., Zhao,D., Arkin,M.R., McKerrow,J.H., Brinen,L.S. and Renslo,A.R.
   Novel non-peptidic vinylsulfones targeting the S2 and S3 subsites of parasite cysteine proteases
   Bioorg Med Chem Lett (2009) 19, 6218-6221. PubMed  Europe PubMed DOI  S  I
7. Kerr,I.D., Lee,J.H., Farady,C.J., Marion,R., Rickert,M., Sajid,M., Pandey,K.C., Caffrey,C.R., Legac,J., Hansell,E., McKerrow,J.H., Craik,C.S., Rosenthal,P.J. and Brinen,L.S.
   Vinyl sulfones as antiparasitic agents and a structural basis for drug design
   J Biol Chem (2009) 284, 25697-25703. PubMed  Europe PubMed DOI  PMC  EPMC  S  I
2005
8. [YEAR:15-3-2005]Choe,Y., Brinen,L.S., Price,M.S., Engel,J.C., Lange,M., Grisostomi,C., Weston,S.G., Pallai,P.V., Cheng,H., Hardy,L.W., Hartsough,D.S., McMakin,M., Tilton,R.F., Baldino,C.M. and Craik,C.S.
   Development of alpha-keto-based inhibitors of cruzain, a cysteine protease implicated in Chagas disease
   Bioorg Med Chem (15-3-2005) 13, 2141-2156. PubMed  Europe PubMed DOI  S  I
2003
9. Huang,L., Brinen,L.S. and Ellman,J.A.
   Crystal structures of reversible ketone-based inhibitors of the cysteine protease cruzain
   Bioorg Med Chem (2003) 11, 21-29. PubMed  Europe PubMed DOI  S  I
1997
10. Gillmor,S.A., Craik,C.S. and Fletterick,R.J.
    Structural determinants of specificity in the cysteine protease cruzain
    Protein Sci (1997) 6, 1603-1611. PubMed  Europe PubMed DOI  PMC  EPMC  S  I
1995
11. McGrath,M.E., Eakin,A.E., Engel,J.C., McKerrow,J.H., Craik,C.S. and Fletterick,R.J.
    The crystal structure of cruzain: A therapeutic target for Chagas' disease
    J Mol Biol (1995) 247, 251-259. PubMed  Europe PubMed DOI  S