Literature for peptidase S01.223: acrosin

(Topics flags: S Structure, I Inhibitor, K Knockout, V Review. To select only the references relevant to a single topic, click the link above. See explanation.)

2024
1. Shibata,T., Bhat,S.A., Cao,D., Saito,S., Bernstein,E.A., Nishi,E., Medenilla,J.D., Wang,E.T., Chan,J.L., Pisarska,M.D., Tourtellotte,W.G., Giani,J.F., Bernstein,K.E. and Khan,Z.
   Testicular ACE regulates sperm metabolism and fertilization through the transcription factor PPARgamma
   J Biol Chem300, 105486-105486. PubMed  Europe PubMed DOI
2020
2. Hirose,M., Honda,A., Fulka,H., Tamura-Nakano,M., Matoba,S., Tomishima,T., Mochida,K., Hasegawa,A., Nagashima,K., Inoue,K., Ohtsuka,M., Baba,T., Yanagimachi,R. and Ogura,A.
   Acrosin is essential for sperm penetration through the zona pellucida in hamsters
   Proc Natl Acad Sci U S A117, 2513-2518. PubMed  Europe PubMed DOI  K
2017
3. Isotani,A., Matsumura,T., Ogawa,M., Tanaka,T., Yamagata,K., Ikawa,M. and Okabe,M.
   A delayed sperm penetration of cumulus layers by disruption of acrosin gene in rats
   Biol Reprod97, 61-68. PubMed  Europe PubMed DOI
2014
4. Zhao,J., Sun,N., Gao,Y., Lv,D., Liu,Y., Jiang,Y., Dong,G., Chen,Q., Li,W., Zhou,Y., Zhu,J., Sheng,C. and Lv,J.
   Discovery of novel guanidinophenylpyrazole human acrosin inhibitors by molecular hybridization
   MedChemComm5, 1520-1527. DOI  I
5. Zhao,J., Tian,W., Qi,J., Lv,D., Liu,Y., Jiang,Y., Dong,G., Chen,Q., Zhou,Y., Zhu,J., Wang,H., Sheng,C. and Lv,J.
   Design and synthesis of phenylisoxazole derivatives as novel human acrosin inhibitors
   Bioorg Med Chem Lett24, 2802-2806. PubMed  Europe PubMed DOI  I
2013
6. Chen,Q., Tian,W., Han,G., Qi,J., Zheng,C., Zhou,Y., Ding,L., Zhao,J., Zhu,J., Lv,J. and Sheng,C.
   Design and synthesis of novel benzoheterocyclic derivatives as human acrosin inhibitors by scaffold hopping
   Eur J Med Chem59, 176-182. PubMed  Europe PubMed DOI  I
7. Mao,H.T. and Yang,W.X.
   Modes of acrosin functioning during fertilization
   Gene526, 75-79. PubMed  Europe PubMed DOI  K
8. Ning,W., Zhu,J., Zheng,C., Liu,X., Song,Y., Zhou,Y., Zhang,X., Zhang,L., Sheng,C. and Lv,J.
   Fragment-based design of novel quinazolinon derivatives as human acrosin inhibitors
   Chem Biol Drug Des81, 437-441. PubMed  Europe PubMed DOI  I
9. Tian,W., Han,G., Zhu,J., Qi,J., Chen,Q., Zhao,J., Zheng,C., Zhang,L., Zhou,Y. and Lv,J.
   Synthesis and acrosin inhibitory activities of 5-phenyl-1H-pyrazole-3-carboxylic acid amide derivatives
   Bioorg Med Chem Lett23, 4177-4184. PubMed  Europe PubMed DOI  I
2012
10. Adham,I.M., Schlosser,M. and Engel,W.
    Acrosin
    [ISSN:978-0-12-407742-3]3, 2731-2735. DOI
11. Liu,X., Chen,Q., Zhu,J., Fan,Y., Ding,L., Zhao,J., Han,G., Tian,W., Qi,J., Zhou,Y. and Lv,J.
    Synthesis and acrosin inhibitory activity of methyl 5-substituted-1H-benzo[d]imidazol-2-yl carbamate derivatives
    Bioorg Med Chem Lett22, 3554-3559. PubMed  Europe PubMed DOI  I
12. Slowinska,M. and Ciereszko,A.
    Identification of the second form of acrosin in turkey spermatozoa
    Reprod Domest Anim47, 849-855. PubMed  Europe PubMed DOI
2011
13. Ding,L., Zhu,J., Zheng,C., Sheng,C., Qi,J., Liu,X., Han,G., Zhao,J., Lv,J. and Zhou,Y.
    Synthesis and acrosin inhibitory activity of substituted 4-amino-N-(diaminomethylene) benzenesulfonamide derivatives
    Bioorg Med Chem Lett21, 6674-6677. PubMed  Europe PubMed DOI  I
14. Jiang,J.H., Liu,X.F., Zhen,C.H., Zhou,Y.J., Zhu,J., Lv,J.G. and Sheng,C.Q.
    Acrosin structure-based design, synthesis and biological activities of 7-azaindol derivatives as new acrosin inhibitors
    Chin Chem Lett22, 272-275. DOI  I
15. Liu,X., Dong,G., Zhang,J., Qi,J., Zheng,C., Zhou,Y., Zhu,J., Sheng,C. and Lu,J.
    Discovery of novel human acrosin inhibitors by virtual screening
    J Comput Aided Mol Des25, 977-985. PubMed  Europe PubMed DOI  I
16. Moreno,R.D., Laserre,A.A. and Barros,C.
    Protease activity involvement in the passage of mammalian sperm through the zona pellucida
    Biol Res44, 145-150. PubMed  Europe PubMed DOI
17. Qi,J.J., Zhou,Y.J., Liu,X.F., Ding,L.L., Zheng,C.H., Sheng,C.Q., Lv,J.G. and Zhu,J.
    Synthesis and crystal structure of a novel ethyl 5-(4-(2-phenylacetamido) phenyl)-1H-pyrazole-3-carboxylate as an acrosin inhibitor
    Jiegou Huaxue30, 1604-1608.  I
18. Sasanami,T., Yoshizaki,N., Dohra,H. and Kubo,H.
    Sperm acrosin is responsible for the sperm binding to the egg envelope during fertilization in Japanese quail (Coturnix japonica)
    Reproduction142, 267-276. PubMed  Europe PubMed DOI
2010
19. Kawano,N., Kang,W., Yamashita,M., Koga,Y., Yamazaki,T., Hata,T., Miyado,K. and Baba,T.
    Mice lacking two sperm serine proteases, ACR and PRSS21, are subfertile, but the mutant sperm are infertile in vitro
    Biol Reprod83, 359-369. PubMed  Europe PubMed DOI  K
20. Lu,D.Y., Yu,L.M., Yao,J.Z., Sheng,C.Q., Chai,Y.F. and Lou,Z.Y.
    Optimization of the synthesis of human acrosin inhibitor 4'-acetaminophenyl 4-guanidinobenzoate hydrochloride by the orthogonal design
    Chung Kuo Yao Hsueh Tsa Chih45, 231-233.  I
21. Slowinska,M., Olczak,M., Liszewska,E., Watorek,W. and Ciereszko,A.
    Isolation, characterization and cDNA sequencing of acrosin from turkey spermatozoa
    Comp Biochem Physiol B Biochem Mol Biol157, 127-136. PubMed  Europe PubMed DOI
22. Zhang,X.M., Zhu,J., Liu,X.F., Sheng,C.Q., Zheng,C.H., Fu,X.D., Song,Y.L., Zhou,Y.J. and Lu,J.G.
    Design, synthesis and activity evaluation of 9-substituted-2-amino-6-guanidinopurines as acrosin inhibitors
    Gaodeng Xuexiao Huaxue Xuebao/Chemical Journal of Chinese Universities31, 1753-1761.  I
2009
23. Zhang,J., Zheng,C.H., Sheng,C.Q., Zhou,Y.J., Zhu,J. and Lu,J.G.
    Characterization of human acrosin active site and binding modes with its inhibitors
    Gaodeng Xuexiao Huaxue Xuebao/Chemical Journal of Chinese Universities30, 2409-2414.
2008
24. Bajou,K., Peng,H., Laug,W.E., Maillard,C., Noel,A., Foidart,J.M., Martial,J.A. and DeClerck,Y.A.
    Plasminogen activator inhibitor-1 protects endothelial cells from FasL-mediated apoptosis
    Cancer Cell14, 324-334. PubMed  Europe PubMed DOI
25. Raterman,D. and Springer,M.S.
    The molecular evolution of acrosin in placental mammals
    Mol Reprod Dev75, 1196-1207. PubMed  Europe PubMed DOI
2007
26. Gaboriau,D., Howes,E.A., Clark,J. and Jones,R.
    Binding of sperm proacrosin/beta-acrosin to zona pellucida glycoproteins is sulfate and stereodependent. Synthesis of a novel fertilization inhibitor
    Dev Biol306, 646-657. PubMed  Europe PubMed DOI
27. Gatesy,J. and Swanson,W.J.
    Adaptive evolution and phylogenetic utility of Acr (acrosin), a rapidly evolving mammalian fertilization gene
    J Mammal88, 32-42. DOI
2006
28. Lu,J.G., Sheng,C.Q., Zhang,M., Ji,H.T., Zhang,W.N., Zhou,Y.J., Zhu,J. and Jiang,J.H.
    Homology modeling of human acrosin and its molecular docking study with KF950
    Acta Chimica Sinica64, 1073-1078.
2005
29. Furlong,L.I., Veaute,C. and Vazquez-Levin,M.H.
    Binding of recombinant human proacrosin/acrosin to zona pellucida glycoproteins. II. Participation of mannose residues in the interaction
    Fertil Steril83, 1791-1796. PubMed  Europe PubMed DOI
30. Furlong,L.I., Harris,J.D. and Vazquez-Levin,M.H.
    Binding of recombinant human proacrosin/acrosin to zona pellucida (ZP) glycoproteins. I. Studies with recombinant human ZPA, ZPB, and ZPC
    Fertil Steril83, 1780-1790. PubMed  Europe PubMed DOI
31. Langlois,M.R., Oorlynck,L., Vandekerckhove,F., Criel,A., Bernard,D. and Blaton,V.
    Discrepancy between sperm acrosin activity and sperm morphology: significance for fertilization in vitro
    Clin Chim Acta351, 121-129. PubMed  Europe PubMed DOI
2004
32. Rosatti,M.I., Beconi,M.T. and Cordoba,M.
    Proacrosin-acrosin activity in capacitated and acrosome reacted sperm from cryopreserved bovine semen
    Biocell28, 311-316. PubMed  Europe PubMed
2002
33. Moreno,R.D., Bustamante,E., Schatten,G. and Barros,C.
    Inhibition of mouse in vitro fertilization by an antibody against a unique 18-amino acid domain in the polysulfate-binding domain of proacrosin/acrosin
    Fertil Steril77, 812-817. PubMed  Europe PubMed DOI
2001
34. Schulten,H.J., Nayernia,K., Reim,K., Engel,W. and Burfeind,P.
    Assessment of promoter elements of the germ cell-specific proacrosin gene
    J Cell Biochem83, 155-162. PubMed  Europe PubMed DOI
2000
35. Moreno,R.D. and Barros,C.
    A basic 18-amino acid peptide contains the polysulfate-binding domain responsible for activation of the boar proacrosin/acrosin system
    Biol Reprod62, 1536-1542. PubMed  Europe PubMed
36. [YEAR:15-11-2000]Tranter,R., Read,J.A., Jones,R. and Brady,R.L.
    Effector sites in the three-dimensional structure of mammalian sperm beta-acrosin
    Structure8, 1179-1188. PubMed  Europe PubMed DOI  S  I
1999
37. Crosby,J.A. and Barros,C.
    Effect of recombinant boar beta-acrosin on sperm binding to intact zona pellucida during in vitro fertilization
    Biol Reprod61, 1535-1540. PubMed  Europe PubMed
1998
38. Crosby,J.A., Jones,R., Barros,C. and Carvallo,P.
    Characterization of the functional domains of boar acrosin involved in nonenzymatic binding to homologous zona pellucida glycoproteins
    Mol Reprod Dev49, 426-434. PubMed  Europe PubMed DOI
39. Jansen,S., Jones,R., Jenneckens,I., Marschall,B., Kriegesmann,B., Coadwell,J. and Brenig,B.
    Site-directed mutagenesis of boar proacrosin reveals residues involved in binding of zona pellucida glycoproteins
    Mol Reprod Dev51, 184-192. PubMed  Europe PubMed DOI
40. Suter,L. and Habenicht,U.F.
    Characterization of mouse epididymal acrosin: comparative studies with acrosin from boar and human ejaculated spermatozoa
    Int J Androl21, 95-104. PubMed  Europe PubMed DOI
41. [YEAR:24-4-1998]Yamagata,K., Murayama,K., Okabe,M., Toshimori,K., Nakanishi,T., Kashiwabara,S. and Baba,T.
    Acrosin accelerates the dispersal of sperm acrosomal proteins during acrosome reaction
    J Biol Chem273, 10470-10474. PubMed  Europe PubMed DOI
1997
42. Adham,I.M., Nayernia,K. and Engel,W.
    Spermatozoa lacking acrosin protein show delayed fertilization
    Mol Reprod Dev46, 370-376. PubMed  Europe PubMed DOI  K
1996
43. Adham,I.M., Kremling,H., Nieter,S., Zimmermann,S., Hummel,M., Schroeter,U. and Engel,W.
    The structures of the bovine and porcine proacrosin genes and their conservation among mammals
    Biol Chem Hoppe Seyler377, 261-265. PubMed  Europe PubMed
1995
44. Adeniran,A.J., Shoshani,I., Minuth,M., Awad,J.A., Elce,J.S. and Johnson,R.A.
    Purification, characterization, and N-terminal amino acid sequence of the adenylyl cyclase-activating protease from bovine sperm
    Biol Reprod52, 490-499. PubMed  Europe PubMed DOI
1994
45. [YEAR:16-12-1994]Baba,T., Azuma,S., Kashiwabara,S. and Toyoda,Y.
    Sperm from mice carrying a targeted mutation of the acrosin gene can penetrate the oocyte zona pellucida and effect fertilization
    J Biol Chem269, 31845-31849. PubMed  Europe PubMed  K
46. Friedl,R., Adham,I.M. and Rottmann,O.J.
    Mapping of the gene encoding bovine preproacrosin (ACR) to chromosome BTA 5 region q35
    Mamm Genome5, 830-831. PubMed  Europe PubMed DOI
47. Hermans,J.M., Jones,R. and Stone,S.R.
    Rapid inhibition of the sperm protease acrosin by protein C inhibitor
    Biochemistry33, 5440-5444. PubMed  Europe PubMed DOI
48. [YEAR:13-9-1994]Richardson,R.T. and O'Rand,M.G.
    Cloning and sequencing of cDNAs for rabbit preproacrosin and a novel preproacrosin-related cDNA
    Biochim Biophys Acta1219, 215-218. PubMed  Europe PubMed DOI
1991
49. Klemm,U., Flake,A. and Engel,W.
    Rat sperm acrosin: cDNA sequence, derived primary structure and phylogenetic origin
    Biochim Biophys Acta1090, 270-272. PubMed  Europe PubMed DOI
50. Kobayashi,T., Matsuda,Y., Oshio,S., Kaneko,S., Nozawa,S., Mhori,H., Akihama,S. and Fujimoto,Y.
    Human acrosin: purification and some properties
    Syst Biology Reprod Med27, 9-16. DOI
51. Kremling,H., Keime,S., Wilhelm,K., Adham,I.M., Hameister,H. and Engel,W.
    Mouse proacrosin gene: Nucleotide sequence, diploid expression, and chromosomal localization
    Genomics11, 828-834. PubMed  Europe PubMed
52. Kremling,H., Flake,A., Adham,I.M., Radtke,J. and Engel,W.
    Exon-intron structure and nucleotide sequence of the rat proacrosin gene
    DNA Seq2, 57-60. PubMed  Europe PubMed
1990
53. [YEAR:30-11-1990]Kashiwabara,S., Arai,Y., Kodaira,K. and Baba,T.
    Acrosin biosynthesis in meiotic and postmeiotic spermatogenic cells
    Biochem Biophys Res Commun173, 240-245. PubMed  Europe PubMed DOI
54. Kashiwabara,S., Baba,T., Takada,M., Watanabe,K., Yano,Y. and Arai,Y.
    Primary structure of mouse proacrosin deduced from the cDNA sequence and its gene expression during spermatogenesis
    J Biochem108, 785-791. PubMed  Europe PubMed
55. Keime,S., Adham,I.M. and Engel,W.
    Nucleotide sequence and exon-intron organization of the human proacrosin gene
    Eur J Biochem190, 195-200. PubMed  Europe PubMed DOI
56. Klemm,U., Maier,W.M., Tsaousidou,S., Adham,I.M., Willison,K. and Engel,W.
    Mouse preproacrosin: cDNA sequence, primary structure and postmeiotic expression in spermatogenesis
    Differentiation42, 160-166. PubMed  Europe PubMed
1989
57. [YEAR:1-7-1989]Adham,I.M., Klemm,U., Maier,W.M., Hoyer-Fender,S., Tsaousidou,S. and Engel,W.
    Molecular cloning of preproacrosin and analysis of its expression pattern in spermatogenesis
    Eur J Biochem182, 563-568. PubMed  Europe PubMed
58. Baba,T., Kashiwabara,S., Watanabe,K., Itoh,H., Michikawa,Y., Kimura,K., Takada,M., Fukamizu,A. and Arai,Y.
    Activation and maturation mechanisms of boar acrosin zymogen based on the deduced primary structure
    J Biol Chem264, 11920-11927. PubMed  Europe PubMed
59. Baba,T., Michikawa,Y., Kawakura,K. and Arai,Y.
    Activation of boar proacrosin is effected by processing at both N- and C-terminal portions of the zymogen molecule
    FEBS Lett244, 132-136. PubMed  Europe PubMed
60. Baba,T., Michikawa,Y., Kashiwabara,S. and Arai,Y.
    Proacrosin activation in the presence of a 32-kDa protein from boar spermatozoa
    Biochem Biophys Res Commun160, 1026-1032. PubMed  Europe PubMed
1987
61. Hardy,D.M., Wild,G.C. and Tung,K.S.
    Purification and initial characterization of proacrosins from guinea pig testes and epididymal spermatozoa
    Biol Reprod37, 189-199. PubMed  Europe PubMed
1984
62. Fock-Nuzel,R., Lottspeich,F., Henschen,A. and Muller-Esterl,W.
    Boar acrosin is a two-chain molecule. Isolation and primary structure of the light chain; homology with the pro-part of other serine proteinases
    Eur J Biochem141, 441-446. PubMed  Europe PubMed
1983
63. Brown,C.R.
    Purification of mouse sperm acrosin, its activation from proacrosin and effect on homologous egg investments
    J Reprod Fertil69, 289-295. PubMed  Europe PubMed
64. Florke-Gerloff,S., Topfer-Petersen,E., Muller-Esterl,W., Schill,W.B. and Engel,W.
    Acrosin and the acrosome in human spermatogenesis
    Hum Genet65, 61-67. PubMed  Europe PubMed
1981
65. Muller-Esterl,W. and Fritz,H.
    Sperm acrosin
    Methods Enzymol80, 621-632. PubMed  Europe PubMed DOI  V
1980
66. Muller-Esterl,W. and Fritz,H.
    Interactions of boar acrosin with detergents
    Hoppe Seylers Z Physiol Chem361, 1673-1682. PubMed  Europe PubMed  I
67. [YEAR:15-9-1980]Sumi,H. and Toki,N.
    Inhibitors of the acrosomal proteinase acrosin: human urinary trypsin inhibitor (UTI) and 4-(2-carboxyethyl) phenyl trans 4-aminomethylcyclohexanecarboxylate hydrochloride (DV-1006)
    Experientia36, 1103-1104. PubMed  Europe PubMed
1978
68. Fink,E. and Wendt,V.
    Demonstration of acrosin in mouse spermatozoa
    J Reprod Fertil53, 75-76. PubMed  Europe PubMed
69. Kettner,C., Springhorn,S., Shaw,E., Muller,W. and Fritz,H.
    Inactivation of boar acrosin by peptidyl-arginyl-chloromethanes. Comparison of the reactivity of acrosin, trypsin and thrombin
    Hoppe Seylers Z Physiol Chem359, 1183-1191. PubMed  Europe PubMed  I
1977
70. Zahler,W.L. and Polakoski,K.L.
    Benzamidine as an inhibitor of proacrosin activation in bull sperm
    Biochim Biophys Acta480, 461-468. PubMed  Europe PubMed  I
1976
71. Borhan,G.S., Schleuning,W.D., Tschesche,H. and Fritz,H.
    Occurrence of multiple forms of bull and ram acrosin during proenzyme activation and inhibition of activation by p-nitrophenyl-p'-guanidino-benzoate
    Hoppe Seylers Z Physiol Chem357, 667-671. PubMed  Europe PubMed  I
72. Brown,C.R. and Hartree,E.F.
    Identification of acrosin in mouse spermatozoa
    J Reprod Fertil46, 249-251. PubMed  Europe PubMed
73. Polakoski,K.L. and Zaneveld,L.J.
    Proacrosin
    Methods Enzymol45, 325-329. PubMed  Europe PubMed DOI  V
74. Schleuning,W.D. and Fritz,H.
    Sperm acrosin
    Methods Enzymol45, 330-342. PubMed  Europe PubMed DOI  V
1975
75. Brown,C.R., Andani,Z. and Hartree,E.F.
    Studies on ram acrosin. Fluorimetric titration of operational molarity with 4-methylumbelliferyl p-guanidinobenzoate
    Biochem J149, 147-154. PubMed  Europe PubMed  I
76. Schiessler,H., Schleuning,W.D. and Fritz,H.
    Cleavage specificity of boar acrosin on polypeptide substrates, ribonuclease and insulin B-chain
    Hoppe Seylers Z Physiol Chem356, 1931-1936. PubMed  Europe PubMed
77. Schill,W.B., Schleuning,W.D., Fritz,H., Wendt,V. and Heimburger,N.
    Immunofluorescent localization of acrosin in spermatozoa by boar acrosin antibodies
    Naturwissenschaften62, 540-541. PubMed  Europe PubMed
1973
78. Schleuning,W.D., Schiessler,H. and Fritz,H.
    Highly purified acrosomal proteinase (boar acrosin): isolation by affinity chromatography using benzamidine-cellulose and stabilization
    Hoppe Seylers Z Physiol Chem354, 550-554. PubMed  Europe PubMed  I
1972
79. Fink,E., Schiessler,H., Arnhold,M. and Fritz,H.
    [Isolation of a trypsin-like enzyme (acrosin) from boar spermatozoa]
    Hoppe Seylers Z Physiol Chem353, 1633-1637. PubMed  Europe PubMed
80. Fritz,H., Forg-Brey,B., Schiessler,H., Arnhold,M. and Fink,E.
    [Characterization of a trypsin-like proteinase (acrosin) from boar spermatozoa by inhibition with different protein proteinase inhibitors, II. Inhibitors from leeches, soybeans, peanuts, bovine colostrum and sea anemones]
    Hoppe Seylers Z Physiol Chem353, 1010-1012. PubMed  Europe PubMed
81. Fritz,H., Heimburger,N., Meier,M., Arnhold,M., Zaneveld,L.J. and Schumacher,G.F.
    [Human acrosin: kinetics of the inhibition by inhibitors from human sera]
    Hoppe Seylers Z Physiol Chem353, 1953-1956. PubMed  Europe PubMed
82. Fritz,H., Forg-Brey,B., Fink,E., Meier,M., Schiessler,H. and Schirren,C.
    [Human acrosin: isolation and properties]
    Hoppe Seylers Z Physiol Chem353, 1943-1949. PubMed  Europe PubMed
83. Fritz,H., Forg-Brey,B., Fink,E., Schiessler,H., Jaumann,E. and Arnhold,M.
    [Characterization of a trypsin-like proteinase (acrosin) from boar spermatozoa by inhibition with different protein proteinase inbibitors. I. Seminal trypsin inhibitors and the trypsin- kallikrein inhibitor from bovine organs]
    Hoppe Seylers Z Physiol Chem353, 1007-1009. PubMed  Europe PubMed
1968
84. [YEAR:9-8-1968]Stambaugh,R. and Buckley,J.
    Zona pellucida dissolution enzymes of the rabbit sperm head
    Science161, 585-586. PubMed  Europe PubMed
1965
85. Srivastava,P.N., Adams,C.E. and Hartree,E.F.
    Enzymic action of acrosomal preparations on the rabbit ovum in vitro
    J Reprod Fertil10, 61-67. PubMed  Europe PubMed