Literature for peptidase M16.011: falcilysin

(Topics flags: I Inhibitor, V Review. To select only the references relevant to a single topic, click the link above. See explanation.)

2025
1. Dalal,A., Malik,J., Singh,P. and Rathi,B.
   Plasmodium falciparum falcilysin as an emerging potential drug target for antimalarial drug discovery
   Drug Discov Today (2025) 31, 104582-104582. PubMed  Europe PubMed DOI
2024
2. Lin,J., Yan,X., Chung,Z., Liew,C.W., El Sahili,A., Pechnikova,E.V., Preiser,P.R., Bozdech,Z., Gao,Y.G. and Lescar,J.
   Inhibition of falcilysin from Plasmodium falciparum by interference with its closed-to-open dynamic transition
   Commun Biol (2024) 7, 1070-1070. PubMed  Europe PubMed DOI  PMC  EPMC  I
2021
3. Kahlon,G., Lira,R., Masvlov,N., Pompa,E., Brar,N., Eagon,S., Anderson,M.O., Andaya,A., Chance,J.P., Fejzic,H., Keniston,A., Huynh,N., Celis,N., Vidal,B., Trieu,N., Rodriguez,P. and Mallari,J.P.
   Corrigendum to "Structure guided development of potent piperazine-derived hydroxamic acid inhibitors targeting falcilysin" [Bioorg. Med. Chem. Lett. 32 (2021) 127683]
   Bioorg Med Chem Lett (2021) 37, 127836-127836. PubMed  Europe PubMed DOI
2020
4. Kahlon,G., Lira,R., Masvlov,N., Pompa,E., Brar,N., Eagon,S., Anderson,M.O., Andaya,A., Chance,J.P., Fejzic,H., Keniston,A., Vidal,B., Trieu,N., Rodriguez,P. and Mallari,J.P.
   Structure Guided Development of Potent Piperazine-Derived Hydroxamic Acid Inhibitors Targeting Falcilysin
   Bioorg Med Chem Lett (2020) 32, 127683-127683. PubMed  Europe PubMed DOI
2018
5. Chance,J.P., Fejzic,H., Hernandez,O., Istvan,E.S., Andaya,A., Maslov,N., Aispuro,R., Crisanto,T., Nguyen,H., Vidal,B., Serrano,W., Kuwahara,B., Pugne Andanado,C., Goldberg,D.E. and Mallari,J.P.
   Development of piperazine-based hydroxamic acid inhibitors against falcilysin, an essential malarial protease
   Bioorg Med Chem Lett (2018) 28, 1846-1848. PubMed  Europe PubMed DOI  I
2012
6. Mallari,J.P. and Goldberg,D.E.
   Falcilysin
   [ISSN:978-0-12-407744-7] (2012) 3, 1459-1461. DOI
2007
7. Ponpuak,M., Klemba,M., Park,M., Gluzman,I.Y., Lamppa,G.K. and Goldberg,D.E.
   A role for falcilysin in transit peptide degradation in the Plasmodium falciparum apicoplast
   Mol Microbiol (2007) 63, 314-334. PubMed  Europe PubMed DOI
8. Ralph,S.A.
   Subcellular multitasking - multiple destinations and roles for the Plasmodium falcilysin protease
   Mol Microbiol (2007) 63, 309-313. PubMed  Europe PubMed DOI
2004
9. Goldberg,D.E. and Murata,C.
   Falcilysin
   [ISSN:0-12-079610-4] (2004) 2, 892-893.  V
2003
10. [YEAR:26-9-2003]Murata,C.E. and Goldberg,D.E.
    Plasmodium falciparum falcilysin: a metalloprotease with dual specificity
    J Biol Chem (26-9-2003) 278, 38022-38028. PubMed  Europe PubMed DOI
11. Murata,C.E. and Goldberg,D.E.
    Plasmodium falciparum falcilysin: an unprocessed food vacuole enzyme
    Mol Biochem Parasitol (2003) 129, 123-126. PubMed  Europe PubMed DOI
1999
12. [YEAR:5-11-1999]Eggleson,K.K., Duffin,K.L. and Goldberg,D.E.
    Identification and characterization of falcilysin, a metallopeptidase involved in hemoglobin catabolism within the malaria parasite Plasmodium falciparum
    J Biol Chem (5-11-1999) 274, 32411-32417. PubMed  Europe PubMed DOI