Literature for peptidase S08.063: site-1 peptidase

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2025
1. Bullington,A.V., Micallo,I., Bajaj,B., Kumar,P., Schlamowitz,N., Silva,A., Hendrix,S., Zelcer,N. and Kober,D.L.
   Structural basis for substrate selectivity by site-one protease revealed by studies with a small-molecule inhibitor
   Proc Natl Acad Sci U S A122, e2426931122-e2426931122. PubMed  Europe PubMed DOI  I
2019
2. Olaposi,O.I., Oyekanmi,N., Ojo,A.A. and Eniafe,G.O.
   Membrane-bound transcription factor site-1 protease in PF429242 bound state: computational kinetics and dynamics of reversible binding
   Drug Res (Stuttg)69, 643-649. PubMed  Europe PubMed DOI  I
2018
3. Al-Maskari,M., Care,M.A., Robinson,E., Cocco,M., Tooze,R.M. and Doody,G.M.
   Site-1 protease function is essential for the generation of antibody secreting cells and reprogramming for secretory activity
   Sci Rep8, 14338-14338. PubMed  Europe PubMed DOI  I
4. Urata,S., Uno,Y., Kurosaki,Y. and Yasuda,J.
   The cholesterol, fatty acid and triglyceride synthesis pathways regulated by site 1 protease (S1P) are required for efficient replication of severe fever with thrombocytopenia syndrome virus
   Biochem Biophys Res Commun503, 631-636. PubMed  Europe PubMed DOI  I
2017
5. Caruana,B.T., Skoric,A., Brown,A.J. and Lutze-Mann,L.H.
   Site-1 protease, a novel metabolic target for glioblastoma
   Biochem Biophys Res Commun490, 760-766. PubMed  Europe PubMed DOI  I
6. Hyrina,A., Meng,F., McArthur,S.J., Eivemark,S., Nabi,I.R. and Jean,F.
   Human subtilisin kexin isozyme-1 (SKI-1)/site-1 protease (S1P) regulates cytoplasmic lipid droplet abundance: a potential target for indirect-acting anti-dengue virus agents
   PLoS ONE12, e0174483-e0174483. PubMed  Europe PubMed DOI  I
7. Nakagawa,T., Suzuki-Nakagawa,C., Watanabe,A., Asami,E., Matsumoto,M., Nakano,M., Ebihara,A., Uddin,M.N. and Suzuki,F.
   Site-1 protease is required for the generation of soluble (pro)renin receptor
   J Biochem161, 369-379. PubMed  Europe PubMed DOI  I
8. Verhelst,S.H.L.
   Intramembrane proteases as drug targets
   FEBS J284, 1489-1502. PubMed  Europe PubMed DOI  I
2011
9. Majumdar,S., Chen,A., Palmer-Smith,H. and Basak,A.
   Novel circular, cyclic and acyclic psi(CH(2)O) containing peptide inhibitors of SKI-1/S1P: synthesis, kinetic and biochemical evaluations
   Curr Med Chem18, 2770-2782. PubMed  Europe PubMed DOI  I
10. Urata,S., Yun,N., Pasquato,A., Paessler,S., Kunz,S. and de la Torre,J.C.
    Antiviral activity of a small-molecule inhibitor of arenavirus glycoprotein processing by the cellular site 1 protease
    J Virol85, 795-803. PubMed  Europe PubMed DOI  I
2010
11. Basak,A., Mitra,D., Das,A.K., Mohottalage,D. and Basak,A.
    C(2)-Symmetric azobenzene-amino acid conjugates and their inhibition of subtilisin kexin isozyme-1
    Bioorg Med Chem Lett20, 3977-3981. PubMed  Europe PubMed DOI  I
12. Rojek,J.M., Pasqual,G., Sanchez,A.B., Nguyen,N.T., de la Torre,J.C. and Kunz,S.
    Targeting the proteolytic processing of the viral glycoprotein precursor is a promising novel antiviral strategy against arenaviruses
    J Virol84, 573-584. PubMed  Europe PubMed DOI  T  I
2008
13. Hawkins,J.L., Robbins,M.D., Warren,L.C., Xia,D., Petras,S.F., Valentine,J.J., Varghese,A.H., Wang,I.K., Subashi,T.A., Shelly,L.D., Hay,B.A., Landschulz,K.T., Geoghegan,K.F. and Harwood,H.J., Jr.
    Pharmacologic inhibition of site 1 protease activity inhibits sterol regulatory element-binding protein processing and reduces lipogenic enzyme gene expression and lipid synthesis in cultured cells and experimental animals
    J Pharmacol Exp Ther326, 801-808. PubMed  Europe PubMed DOI  I
2007
14. Hay,B.A., Abrams,B., Zumbrunn,A.Y., Valentine,J.J., Warren,L.C., Petras,S.F., Shelly,L.D., Xia,A., Varghese,A.H., Hawkins,J.L., Van Camp,J.A., Robbins,M.D., Landschulz,K. and Harwood,H.J., Jr.
    Aminopyrrolidineamide inhibitors of site-1 protease
    Bioorg Med Chem Lett17, 4411-4414. PubMed  Europe PubMed DOI  I
2006
15. Basak,S., Mohottalage,D. and Basak,A.
    Multibranch and pseudopeptide approach for design of novel inhibitors of subtilisin kexin isozyme-1
    Protein Pept Lett13, 863-876. PubMed  Europe PubMed DOI  I
16. [YEAR:21-6-2006]Pasquato,A., Pullikotil,P., Asselin,M.C., Vacatello,M., Paolillo,L., Ghezzo,F., Basso,F., Di Bello,C., Dettin,M. and Seidah,N.G.
    The proprotein convertase SKI-1/S1P. In vitro analysis of Lassa virus glycoprotein-derived substrates and ex vivo validation of irreversible peptide inhibitors
    J Biol Chem281, 23471-23481. PubMed  Europe PubMed DOI  I
2004
17. [YEAR:27-8-2004]Basak,S., Stewart,N.A., Chretien,M. and Basak,A.
    Aminoethyl benzenesulfonyl fluoride and its hexapeptide (Ac-VFRSLK) conjugate are both in vitro inhibitors of subtilisin kexin isozyme-1
    FEBS Lett573, 186-194. PubMed  Europe PubMed DOI  I
2003
18. Okada,T., Haze,K., Nadanaka,S., Yoshida,H., Seidah,N.G., Hirano,Y., Sato,R., Negishi,M. and Mori,K.
    A serine protease inhibitor prevents endoplasmic reticulum stress-induced cleavage but not transport of the membrane-bound transcription factor ATF6
    J Biol Chem278, 31024-31032. PubMed  Europe PubMed DOI  I
2001
19. Caron,M., Auclair,R., Vigouroux,C., Glorian,M., Forest,C. and Capeau,J.
    The HIV protease inhibitor indinavir impairs sterol regulatory element-binding protein-1 intranuclear localization, inhibits preadipocyte differentiation, and induces insulin resistance
    Diabetes50, 1378-1388. PubMed  Europe PubMed  I