Literature for peptidase C01.098: CPC peptidase

(References are filtered for relevance to Inhibitor. To remove the filter click here. See explanation.)

2016
1. Ettari,R., Previti,S., Tamborini,L., Cullia,G., Grasso,S. and Zappala,M.
   The inhibition of cysteine proteases rhodesain and TbCatB: a valuable approach to treat human African trypanosomiasis
   Mini Rev Med Chem (2016) 16, 1374-1391. PubMed  Europe PubMed DOI  V  I
2. Schad,C., Baum,U., Frank,B., Dietzel,U., Mattern,F., Gomes,C., Ponte-Sucre,A., Moll,H., Schurigt,U. and Schirmeister,T.
   Development of a new antileishmanial aziridine-2,3-dicarboxylate-based inhibitor with high selectivity for parasite cysteine proteases
   Antimicrob Agents Chemother (2016) 60, 797-805. PubMed  Europe PubMed DOI  I
2010
3. Mallari,J.P., Zhu,F., Lemoff,A., Kaiser,M., Lu,M., Brun,R. and Guy,R.K.
   Optimization of purine-nitrile TbcatB inhibitors for use in vivo and evaluation of efficacy in murine models
   Bioorg Med Chem (2010) 18, 8302-8309. PubMed  Europe PubMed DOI  I
4. Mott,B.T., Ferreira,R.S., Simeonov,A., Jadhav,A., Ang,K.K., Leister,W., Shen,M., Silveira,J.T., Doyle,P.S., Arkin,M.R., McKerrow,J.H., Inglese,J., Austin,C.P., Thomas,C.J., Shoichet,B.K. and Maloney,D.J.
   Identification and optimization of inhibitors of trypanosomal cysteine proteases: cruzain, rhodesain, and TbCatB
   J Med Chem (2010) 53, 52-60. PubMed  Europe PubMed DOI  S  I
2009
5. Caffrey,C.R. and Steverding,D.
   Kinetoplastid papain-like cysteine peptidases
   Mol Biochem Parasitol (2009) 167, 12-19. PubMed  Europe PubMed DOI  I
6. Mallari,J.P., Shelat,A.A., Kosinski,A., Caffrey,C.R., Connelly,M., Zhu,F., McKerrow,J.H. and Guy,R.K.
   Structure-guided development of selective TbcatB inhibitors
   J Med Chem (2009) 52, 6489-6493. PubMed  Europe PubMed DOI  PMC  EPMC  I
2008
7. Mallari,J.P., Shelat,A.A., Obrien,T., Caffrey,C.R., Kosinski,A., Connelly,M., Harbut,M., Greenbaum,D., McKerrow,J.H. and Guy,R.K.
   Development of potent purine-derived nitrile inhibitors of the trypanosomal protease TbcatB
   J Med Chem (2008) 51, 545-552. PubMed  Europe PubMed DOI  I
8. Mallari,J.P., Shelat,A., Kosinski,A., Caffrey,C.R., Connelly,M., Zhu,F., McKerrow,J.H. and Guy,R.K.
   Discovery of trypanocidal thiosemicarbazone inhibitors of rhodesain and TbcatB
   Bioorg Med Chem Lett (2008) 18, 2883-2885. PubMed  Europe PubMed DOI  PMC  EPMC  I
2003
9. Chibale,K. and Musonda,C.C.
   The synthesis of parasitic cysteine protease and trypanothione reductase inhibitors
   Curr Med Chem (2003) 10, 1863-1889. PubMed  Europe PubMed DOI  I
10. Gantt,K.R., Schultz-Cherry,S., Rodriguez,N., Jeronimo,S.M., Nascimento,E.T., Goldman,T.L., Recker,T.J., Miller,M.A. and Wilson,M.E.
    Activation of TGF-beta by Leishmania chagasi: importance for parasite survival in macrophages
    J Immunol (2003) 170, 2613-2620. PubMed  Europe PubMed  I
1999
11. [YEAR:15-5-1999]Chan,V.J., Selzer,P.M., McKerrow,J.H. and Sakanari,J.A.
    Expression and alteration of the S2 subsite of the Leishmania major cathepsin B-like cysteine protease
    Biochem J (15-5-1999) 340, 113-117. PubMed  Europe PubMed  PMC  EPMC  I