Literature for peptidase C01.040: cathepsin H

Summary Gene structure Alignment Tree Sequences Sequence features Distribution Structure Literature Substrates Inhibitors Pharma

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    2024
  1. Jangra,S., Raghav,N., Wadhwa,D., Kumar,A., Bhattacharyya,S., Kumar,V. and Sheokand,J.
    Biological evaluation of trans-2,3-dihydrofuro[3,2-c]coumarins as potential cathepsin inhibitors and anticancer agents
    J Biomater Sci Polym Ed (2024) , 1-19. PubMed  Europe PubMed DOI  I
  2. 2016
  3. Raghav,N., Jangra,S., Kumar,A., Bhattacharyya,S., Wadhwa,D. and Sindhu,J.
    Cathepsin B, H and L inhibitors as cell proliferating agents: design, synthesis, computational and pharmacological studies of some novel 2-(2-naphthoyl)-6,6-dimethyl-3-aryl-2,3,6,7-tetrahydrobenzofuran-4(5H)-ones
    RSC Adv (2016) 6, 34588-34599. DOI  I
  4. 2015
  5. Singh,M. and Raghav,N.
    2,3-Dihydroquinazolin-4(1H)-one derivatives as potential non-peptidyl inhibitors of cathepsins B and H
    Bioorg Chem (2015) 59C, 12-22. PubMed  Europe PubMed DOI  I
  6. 2014
  7. Raghav,N. and Singh,M.
    Design, synthesis and docking studies of bischalcones based quinazoline-2(1H)-ones and quinazoline-2(1H)-thiones derivatives as novel inhibitors of cathepsin B and cathepsin H
    Eur J Pharm Sci (2014) 54, 28-39. PubMed  Europe PubMed DOI  I
  8. Raghav,N. and Singh,M.
    Acyl hydrazides and triazoles as novel inhibitors of mammalian cathepsin B and cathepsin H
    Eur J Med Chem (2014) 77, 231-242. PubMed  Europe PubMed DOI  I
  9. Raghav,N. and Garg,S.
    SAR studies of o-hydroxychalcones and their cyclized analogs and study them as novel inhibitors of cathepsin B and cathepsin H
    Eur J Pharm Sci (2014) 60, 55-63. PubMed  Europe PubMed DOI  I
  10. Raghav,N. and Singh,M.
    SAR studies of differently functionalized chalcones based hydrazones and their cyclized derivatives as inhibitors of mammalian cathepsin B and cathepsin H
    Bioorg Med Chem (2014) 22, 4233-4245. PubMed  Europe PubMed DOI  I
  11. Ravish,I. and Raghav,N.
    Curcumin as inhibitor of mammalian cathepsin B, cathepsin H, acid phosphatase and alkaline phosphatase: a correlation with pharmacological activities
    Med Chem Res (2014) 23, 2847-2855. DOI  I
  12. 1989
  13. [YEAR:15-8-1989]Angliker,H., Wikstrom,P., Kirschke,H. and Shaw,E.
    The inactivation of the cysteinyl exopeptidases cathepsin H and C by affinity-labelling reagents
    Biochem J (15-8-1989) 262, 63-68. PubMed  Europe PubMed  PMC  EPMC  I
  14. 1982
  15. Barrett,A.J., Kembhavi,A.A., Brown,M.A., Kirschke,H., Knight,C.G., Tamai,M. and Hanada,K.
    L-trans-Epoxysuccinyl-leucylamido(4-guanidino)butane (E-64) and its analogues as inhibitors of cysteine proteinases including cathepsins B, H and L
    Biochem J (1982) 201, 189-198. PubMed  Europe PubMed  PMC  EPMC  I