Literature for peptidase M01.018: endoplasmic reticulum aminopeptidase 1

(References are filtered for relevance to Inhibitor. To remove the filter click here. See explanation.)

2020
1. Maben,Z., Arya,R., Rane,D., An,W.F., Metkar,S., Hickey,M., Bender,S., Ali,A., Nguyen,T.T., Evnouchidou,I., Schilling,R., Stratikos,E., Golden,J. and Stern,L.J.
   Discovery of selective inhibitors of endoplasmic reticulum aminopeptidase 1
   J Med Chem63, 103-121. PubMed  Europe PubMed DOI  I
2019
2. Georgiadis,D., Mpakali,A., Koumantou,D. and Stratikos,E.
   Inhibitors of ER aminopeptidase 1 and 2: from design to clinical application
   Curr Med Chem26, 2715-2729. PubMed  Europe PubMed DOI  I
3. Giastas,P., Neu,M., Rowland,P. and Stratikos,E.
   High-resolution crystal structure of endoplasmic reticulum aminopeptidase 1 with bound phosphinic transition-state analogue inhibitor
   ACS Med Chem Lett10, 708-713. PubMed  Europe PubMed DOI  S  I
4. Koumantou,D., Barnea,E., Martin-Esteban,A., Maben,Z., Papakyriakou,A., Mpakali,A., Kokkala,P., Pratsinis,H., Georgiadis,D., Stern,L.J., Admon,A. and Stratikos,E.
   Editing the immunopeptidome of melanoma cells using a potent inhibitor of endoplasmic reticulum aminopeptidase 1 (ERAP1)
   Cancer Immunol Immunother68, 1245-1261. PubMed  Europe PubMed DOI  I
2017
5. Stamogiannos,A., Maben,Z., Papakyriakou,A., Mpakali,A., Kokkala,P., Georgiadis,D., Stern,L.J. and Stratikos,E.
   Critical role of interdomain interactions in the conformational change and catalytic mechanism of endoplasmic reticulum aminopeptidase 1
   Biochemistry56, 1546-1558. PubMed  Europe PubMed DOI  I
2016
6. Kokkala,P., Mpakali,A., Mauvais,F.X., Papakyriakou,A., Daskalaki,I., Petropoulou,I., Kavvalou,S., Papathanasopoulou,M., Agrotis,S., Fonsou,T.M., van Endert,P., Stratikos,E. and Georgiadis,D.
   Optimization and structure-activity relationships of phosphinic pseudotripeptide inhibitors of aminopeptidases that generate antigenic peptides
   J Med Chem59, 9107-9123. PubMed  Europe PubMed DOI  I
7. Stamogiannos,A., Papakyriakou,A., Mauvais,F.X., van Endert,P. and Stratikos,E.
   Screening identifies thimerosal as a selective inhibitor of endoplasmic reticulum aminopeptidase 1
   ACS Med Chem Lett7, 681-685. PubMed  Europe PubMed DOI  I
2014
8. Hitzerd,S.M., Verbrugge,S.E., Ossenkoppele,G., Jansen,G. and Peters,G.J.
   Positioning of aminopeptidase inhibitors in next generation cancer therapy
   Amino Acids46, 793-808. PubMed  Europe PubMed DOI  I
9. Park,H., Shim,J.S., Kim,B.S., Jung,H.J., Huh,T.L. and Kwon,H.J.
   Purpurin inhibits adipocyte-derived leucine aminopeptidase and angiogenesis in a zebrafish model
   Biochem Biophys Res Commun450, 561-567. PubMed  Europe PubMed DOI  I
2002
10. Akada,T., Yamazaki,T., Miyashita,H., Niizeki,O., Abe,M., Sato,A., Satomi,S. and Sato,Y.
    Puromycin insensitive leucyl-specific aminopeptidase (PILSAP) is involved in the activation of endothelial integrins
    J Cell Physiol193, 253-262. PubMed  Europe PubMed DOI  I