Literature for peptidase C48.002: SENP1 peptidase

Summary Gene structure Alignment Tree Sequences Sequence features Distribution Structure Literature Substrates

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    2022
  1. Bailly,C.
    Anti-inflammatory and anticancer p-terphenyl derivatives from fungi of the genus Thelephora
    Bioorg Med Chem70, 116935-116935. PubMed  Europe PubMed DOI  V  I
  2. Brand,M., Bommeli,E.B., Rutimann,M., Lindenmann,U. and Riedl,R.
    Discovery of a Dual SENP1 and SENP2 Inhibitor
    Int J Mol Sci23, PubMed  Europe PubMed DOI  I
  3. Wei,H., Guo,J., Sun,X., Gou,W., Ning,H., Shang,H., Liu,Q., Hou,W. and Li,Y.
    Discovery of Natural Ursane-type SENP1 Inhibitors and the Platinum Resistance Reversal Activity Against Human Ovarian Cancer Cells: A Structure-Activity Relationship Study
    J Nat Prod85, 1248-1255. PubMed  Europe PubMed DOI  I
  4. 2021
  5. Goossens,J.F., Goossens,L. and Bailly,C.
    Hinokiflavone and Related C-O-C-Type Biflavonoids as Anti-cancer Compounds: Properties and Mechanism of Action
    Nat Prod Bioprospect PubMed  Europe PubMed DOI  V  I
  6. 2020
  7. Lindenmann,U., Brand,M., Gall,F., Frasson,D., Hunziker,L., Kroslakova,I., Sievers,M. and Riedl,R.
    Discovery of a class of potent and selective non-competitive sentrin-specific protease 1 inhibitors
    ChemMedChem15, 675-679. PubMed  Europe PubMed DOI  I
  8. 2018
  9. Ambaye,N., Chen,C.H., Khanna,S., Li,Y.J. and Chen,Y.
    Streptonigrin inhibits SENP1 and reduces the protein level of hypoxia-inducible factor 1alpha (HIF1alpha) in cells
    Biochemistry57, 1807-1813. PubMed  Europe PubMed DOI  I
  10. 2016
  11. Chen,Y.-Y., Sun,J.-L., Li,S., Zhang,J. and Wu,Y.-L.
    Preliminary study on the synthesis and biological activity of small molecule inhibitor JK043 of SUMO-specific protease 1
    J Shanghai Jiaotong Univ Med Sci36, 224-228. DOI  I
  12. Wu,J., Lei,H., Zhang,J., Chen,X., Tang,C., Wang,W., Xu,H., Xiao,W., Gu,W. and Wu,Y.
    Momordin Ic, a new natural SENP1 inhibitor, inhibits prostate cancer cell proliferation
    Oncotarget7, 58995-59005. PubMed  Europe PubMed DOI  I
  13. Yoshioka,Y., Namiki,D., Makiuchi,M., Sugaya,K., Onose,J., Ashida,H. and Abe,N.
    Vialinin A and thelephantin G, potent inhibitors of tumor necrosis factor-alpha production, inhibit sentrin/SUMO-specific protease 1 enzymatic activity
    Bioorg Med Chem Lett26, 4237-4240. PubMed  Europe PubMed DOI  I
  14. 2013
  15. Sommer,S., Weikart,N.D., Linne,U. and Mootz,H.D.
    Covalent inhibition of SUMO and ubiquitin-specific cysteine proteases by an in situ thiol-alkyne addition
    Bioorg Med Chem21, 2511-2517. PubMed  Europe PubMed DOI  I
  16. 2012
  17. Chen,Y., Wen,D., Huang,Z., Huang,M., Luo,Y., Liu,B., Lu,H., Wu,Y., Peng,Y. and Zhang,J.
    2-(4-Chlorophenyl)-2-oxoethyl 4-benzamidobenzoate derivatives, a novel class of SENP1 inhibitors: virtual screening, synthesis and biological evaluation
    Bioorg Med Chem Lett22, 6867-6870. PubMed  Europe PubMed DOI  I
  18. Uno,M., Koma,Y., Ban,H.S. and Nakamura,H.
    Discovery of 1-[4-(N-benzylamino)phenyl]-3-phenylurea derivatives as non-peptidic selective SUMO-sentrin specific protease (SENP)1 inhibitors
    Bioorg Med Chem Lett22, 5169-5173. PubMed  Europe PubMed DOI  I
  19. 2011
  20. Albrow,V.E., Ponder,E.L., Fasci,D., Bekes,M., Deu,E., Salvesen,G.S. and Bogyo,M.
    Development of small molecule inhibitors and probes of human SUMO deconjugating proteases
    Chem Biol18, 722-732. PubMed  Europe PubMed DOI  I
  21. 2004
  22. Hemelaar,J., Borodovsky,A., Kessler,B.M., Reverter,D., Cook,J., Kolli,N., Gan-Erdene,T., Wilkinson,K.D., Gill,G., Lima,C.D., Ploegh,H.L. and Ovaa,H.
    Specific and covalent targeting of conjugating and deconjugating enzymes of ubiquitin-like proteins
    Mol Cell Biol24, 84-95. PubMed  Europe PubMed DOI  I