$VAR1 = undef;

Summary for peptidase C01.077: falcipain-1

Summary Alignment Tree Sequences Sequence features Distribution Literature Substrates

 

Names
MEROPS Namefalcipain-1
Other namesberghepain-1 (Plasmodium berghei), chabaupain-1 (Plasmodium chabaudi), vinckepain-1 (Plasmodium vinvkei), vivapain-1 (Plasmodium vivax)
Domain architecture
MEROPS Classification
Classification Clan CA >> Subclan (none) >> Family C1 >> Subfamily A >> C01.077
Holotypefalcipain-1 (Plasmodium falciparum), Uniprot accession P25805 (peptidase unit: 337-569), MERNUM MER0000675
History Identifier created: Handbook of Proteolytic Enzymes (1998) Academic Press, London.
Activity
Catalytic typeCysteine
NC-IUBMBNot yet included in IUBMB recommendations.
PhysiologyMalarial parasite development and nutrition.
Pharmaceutical relevanceSpecific inhibitors blocked parasite invasion of host erythrocytes (Greenbaum et al., 2002), and falcipain-1 is therefore a potential drug target for malaria.
Other databases PANTHERhttp://www.pantherdb.org/panther/familyList.do?searchType=basic&fieldName=all&listType=6&fieldValue=PTHR12411:SF414