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Literature for peptidase T01.005: bacterial proteasome, beta component

Summary Alignment Tree Sequences Sequence features Distribution Structure Literature Substrates

(Topics flags: A Assay, S Structure, T Target, K Knockout, P Specificity, I Inhibitor, V Review. To select only the references relevant to a single topic, click the link above. See explanation.)

    2020
  1. Rozman,K., Alexander,E.M., Ogorevc,E., Bozovicar,K., Sosic,I., Aldrich,C.C. and Gobec,S.
    Psoralen derivatives as inhibitors of Mycobacterium tuberculosis proteasome
    Molecules25, PubMed  Europe PubMed DOI  I
  2. Vimer,S., Ben-Nissan,G., Morgenstern,D., Kumar-Deshmukh,F., Polkinghorn,C., Quintyn,R.S., Vasil'ev,Y.V., Beckman,J.S., Elad,N., Wysocki,V.H. and Sharon,M.
    Comparative structural analysis of 20S proteasome ortholog protein complexes by native mass spectrometry
    ACS Cent Sci6, 573-588. PubMed  Europe PubMed DOI  S
    3. 2019
  3. Becker,S.H., Jastrab,J.B., Dhabaria,A., Chaton,C.T., Rush,J.S., Korotkov,K.V., Ueberheide,B. and Darwin,K.H.
    The Mycobacterium tuberculosis Pup-proteasome system regulates nitrate metabolism through an essential protein quality control pathway
    Proc Natl Acad Sci U S A116, 3202-3210. PubMed  Europe PubMed DOI
  4. Becker,S.H., Li,H. and Heran Darwin,K.
    Biology and Biochemistry of Bacterial Proteasomes
    Subcell Biochem93, 339-358. PubMed  Europe PubMed DOI
  5. Muller,A.U. and Weber-Ban,E.
    The bacterial proteasome at the core of diverse degradation pathways
    Front Mol Biosci6, 23-23. PubMed  Europe PubMed DOI
    6. 2017
  6. Hsu,H.C., Singh,P.K., Fan,H., Wang,R., Sukenick,G., Nathan,C., Lin,G. and Li,H.
    Structural basis for the species-selective binding of N,C-capped dipeptides to the Mycobacterium tuberculosis proteasome
    Biochemistry56, 324-333. PubMed  Europe PubMed DOI
  7. Jastrab,J.B., Samanovic,M.I., Copin,R., Shopsin,B. and Darwin,K.H.
    Loss-of-function mutations in HspR rescue the growth defect of a Mycobacterium tuberculosis proteasome activator E (pafE) mutant
    J Bacteriol199, e00850-16-e00850-16. PubMed  Europe PubMed DOI
  8. Moreira,W., Santhanakrishnan,S., Dymock,B.W. and Dick,T.
    Bortezomib warhead-switch confers dual activity against mycobacterial caseinolytic protease and proteasome and selectivity against human proteasome
    Front Microbiol8, 746-746. PubMed  Europe PubMed DOI  I
  9. Totaro,K.A., Barthelme,D., Simpson,P.T., Jiang,X., Lin,G., Nathan,C.F., Sauer,R.T. and Sello,J.K.
    Rational design of selective and bioactive inhibitors of the Mycobacterium tuberculosis proteasome
    ACS Infect Dis3, 176-181. PubMed  Europe PubMed DOI  I
  10. Wu,Y., Hu,K., Li,D., Bai,L., Yang,S., Jastrab,J.B., Xiao,S., Hu,Y., Zhang,S., Darwin,K.H., Wang,T. and Li,H.
    Mycobacterium tuberculosis proteasomal ATPase Mpa has a beta-grasp domain that hinders docking with the proteasome core protease
    Mol Microbiol105, 227-241. PubMed  Europe PubMed DOI
    11. 2016
  11. Bai,L., Hu,K., Wang,T., Jastrab,J.B., Darwin,K.H. and Li,H.
    Structural analysis of the dodecameric proteasome activator PafE in Mycobacterium tuberculosis
    Proc Natl Acad Sci U S A113, E1983-E1992. PubMed  Europe PubMed DOI
  12. Bolten,M., Delley,C.L., Leibundgut,M., Boehringer,D., Ban,N. and Weber-Ban,E.
    Structural analysis of the bacterial proteasome activator Bpa in complex with the 20S proteasome
    Structure24, 2138-2151. PubMed  Europe PubMed DOI  S
  13. dela Pena,A.H. and Lander,G.C.
    What's the key to unlocking the proteasome's gate?
    Structure24, 2037-2038. PubMed  Europe PubMed DOI
    14. 2015
  14. Jastrab,J.B., Wang,T., Murphy,J.P., Bai,L., Hu,K., Merkx,R., Huang,J., Chatterjee,C., Ovaa,H., Gygi,S.P., Li,H. and Darwin,K.H.
    An adenosine triphosphate-independent proteasome activator contributes to the virulence of Mycobacterium tuberculosis
    Proc Natl Acad Sci U S A112, E1763-E1772. PubMed  Europe PubMed DOI
  15. Mehra,R., Chib,R., Munagala,G., Yempalla,K.R., Khan,I.A., Singh,P.P., Khan,F.G. and Nargotra,A.
    Discovery of new Mycobacterium tuberculosis proteasome inhibitors using a knowledge-based computational screening approach
    Mol Divers19, 1003-1019. PubMed  Europe PubMed DOI  I
  16. Russo,F., Gising,J., Akerbladh,L., Roos,A.K., Naworyta,A., Mowbray,S.L., Sokolowski,A., Henderson,I., Alling,T., Bailey,M.A., Files,M., Parish,T., Karlen,A. and Larhed,M.
    Optimization and evaluation of 5-styryl-oxathiazol-2-one Mycobacterium tuberculosis proteasome inhibitors as potential antitubercular agents
    ChemistryOpen4, 342-362. PubMed  Europe PubMed DOI  I
    17. 2014
  17. Anandan,T., Han,J., Baun,H., Nyayapathy,S., Brown,J.T., Dial,R.L., Moltalvo,J.A., Kim,M.S., Yang,S.H., Ronning,D.R., Husson,R.N., Suh,J. and Kang,C.M.
    Phosphorylation regulates mycobacterial proteasome
    J Microbiol52, 743-754. PubMed  Europe PubMed DOI
  18. Delley,C.L., Laederach,J., Ziemski,M., Bolten,M., Boehringer,D. and Weber-Ban,E.
    Bacterial proteasome activator Bpa (rv3780) is a novel ring-shaped interactor of the mycobacterial proteasome
    PLoS ONE9, e114348-e114348. PubMed  Europe PubMed DOI
    19. 2013
  19. Lin,G., Chidawanyika,T., Tsu,C., Warrier,T., Vaubourgeix,J., Blackburn,C., Gigstad,K., Sintchak,M., Dick,L. and Nathan,C.
    N,C-Capped dipeptides with selectivity for mycobacterial proteasome over human proteasomes: role of S3 and S1 binding pockets
    J Am Chem Soc135, 9968-9971. PubMed  Europe PubMed DOI  I
  20. Maldonado,A.Y., Burz,D.S., Reverdatto,S. and Shekhtman,A.
    Fate of Pup inside the Mycobacterium proteasome studied by in-cell NMR
    PLoS ONE8, e74576-e74576. PubMed  Europe PubMed DOI
  21. Samanovic,M.I., Li,H. and Darwin,K.H.
    The Pup-proteasome system of Mycobacterium tuberculosis
    Subcell Biochem66, 267-295. PubMed  Europe PubMed DOI
  22. Song,J.X. and Jiang,X.
    [Establishment of a Mycobacterium tuberculosis proteasome inhibitor model in vitro]
    Zhonghua Jie He He Hu Xi Za Zhi36, 363-366. PubMed  Europe PubMed  A  I
    23. 2012
  23. Burns,K.E., McAllister,F.E., Schwerdtfeger,C., Mintseris,J., Cerda-Maira,F., Noens,E.E., Wilmanns,M., Hubbard,S.R., Melandri,F., Ovaa,H., Gygi,S.P. and Darwin,K.H.
    Mycobacterium tuberculosis prokaryotic ubiquitin-like protein-deconjugating enzyme is an unusual aspartate amidase
    J Biol Chem287, 37522-37529. PubMed  Europe PubMed DOI
  24. Lin,G., Li,H. and Nathan,C.F.
    Bacterial proteasome
    [ISSN:978-0-12-407742-3]3, 3671-3677. DOI
    25. 2011
  25. Kale,A.J., McGlinchey,R.P., Lechner,A. and Moore,B.S.
    Bacterial self-resistance to the natural proteasome inhibitor salinosporamide A
    ACS Chem Biol6, 1257-1264. PubMed  Europe PubMed DOI  I
    26. 2010
  26. Burns,K.E., Cerda-Maira,F.A., Wang,T., Li,H., Bishai,W.R. and Darwin,K.H.
    "Depupylation" of prokaryotic ubiquitin-like protein from mycobacterial proteasome substrates
    Mol Cell39, 821-827. PubMed  Europe PubMed DOI
  27. Cerda-Maira,F.A., Pearce,M.J., Fuortes,M., Bishai,W.R., Hubbard,S.R. and Darwin,K.H.
    Molecular analysis of the prokaryotic ubiquitin-like protein (Pup) conjugation pathway in Mycobacterium tuberculosis
    Mol Microbiol77, 1123-1135. PubMed  Europe PubMed DOI
  28. Cheng,Y. and Pieters,J.
    Novel proteasome inhibitors as potential drugs to combat tuberculosis
    J Mol Cell Biol2, 173-175. PubMed  Europe PubMed DOI  I
  29. Gandotra,S., Lebron,M.B. and Ehrt,S.
    The Mycobacterium tuberculosis proteasome active site threonine is essential for persistence yet dispensable for replication and resistance to nitric oxide
    PLoS Pathog6, e1001040-e1001040. PubMed  Europe PubMed DOI
  30. Imkamp,F., Striebel,F., Sutter,M., Ozcelik,D., Zimmermann,N., Sander,P. and Weber-Ban,E.
    Dop functions as a depupylase in the prokaryotic ubiquitin-like modification pathway
    EMBO Rep11, 791-797. PubMed  Europe PubMed DOI
  31. Li,D., Li,H., Wang,T., Pan,H., Lin,G. and Li,H.
    Structural basis for the assembly and gate closure mechanisms of the Mycobacterium tuberculosis 20S proteasome
    EMBO J29, 2037-2047. PubMed  Europe PubMed DOI  S
  32. Lin,G., Li,D., Chidawanyika,T., Nathan,C. and Li,H.
    Fellutamide B is a potent inhibitor of the Mycobacterium tuberculosis proteasome
    Arch Biochem Biophys501, 214-220. PubMed  Europe PubMed DOI  I
  33. Striebel,F., Hunkeler,M., Summer,H. and Weber-Ban,E.
    The mycobacterial Mpa-proteasome unfolds and degrades pupylated substrates by engaging Pup's N-terminus
    EMBO J29, 1262-1271. PubMed  Europe PubMed DOI
  34. Wang,T., Darwin,K.H. and Li,H.
    Binding-induced folding of prokaryotic ubiquitin-like protein on the Mycobacterium proteasomal ATPase targets substrates for degradation
    Nat Struct Mol Biol17, 1352-1357. PubMed  Europe PubMed DOI
    35. 2009
  35. Cerda-Maira,F. and Darwin,K.H.
    The Mycobacterium tuberculosis proteasome: more than just a barrel-shaped protease
    Microbes Infect11, 1150-1155. PubMed  Europe PubMed DOI
  36. Lin,G., Li,D., de Carvalho,L.P., Deng,H., Tao,H., Vogt,G., Wu,K., Schneider,J., Chidawanyika,T., Warren,J.D., Li,H. and Nathan,C.
    Inhibitors selective for mycobacterial versus human proteasomes
    Nature461, 621-626. PubMed  Europe PubMed DOI  I
  37. Striebel,F., Imkamp,F., Sutter,M., Steiner,M., Mamedov,A. and Weber-Ban,E.
    Bacterial ubiquitin-like modifier Pup is deamidated and conjugated to substrates by distinct but homologous enzymes
    Nat Struct Mol Biol16, 647-651. PubMed  Europe PubMed DOI
    38. 2008
  38. Lin,G., Tsu,C., Dick,L., Zhou,X.K. and Nathan,C.
    Distinct specificities of Mycobacterium tuberculosis and mammalian proteasomes for N-acetyl tripeptide substrates
    J Biol Chem283, 34423-34431. PubMed  Europe PubMed DOI  P
    39. 2007
  39. De Mot,R.
    Actinomycete-like proteasomes in a Gram-negative bacterium
    Trends Microbiol15, 335-338. PubMed  Europe PubMed DOI
  40. Gandotra,S., Schnappinger,D., Monteleone,M., Hillen,W. and Ehrt,S.
    In vivo gene silencing identifies the Mycobacterium tuberculosis proteasome as essential for the bacteria to persist in mice
    Nat Med13, 1515-1520. PubMed  Europe PubMed DOI  T
  41. Kaganman,I.
    The dynamic proteasome
    Nat Methods4, 202-203. DOI
  42. Sharon,M., Witt,S., Glasmacher,E., Baumeister,W. and Robinson,C.V.
    Mass spectrometry reveals the missing links in the assembly pathway of the bacterial 20S proteasome
    J Biol Chem282, 18448-18457. PubMed  Europe PubMed DOI
    43. 2006
  43. Hu,G., Lin,G., Wang,M., Dick,L., Xu,R.M., Nathan,C. and Li,H.
    Structure of the Mycobacterium tuberculosis proteasome and mechanism of inhibition by a peptidyl boronate
    Mol Microbiol59, 1417-1428. PubMed  Europe PubMed DOI  S  I
  44. Lin,G., Hu,G., Tsu,C., Kunes,Y.Z., Li,H., Dick,L., Parsons,T., Li,P., Chen,Z., Zwickl,P., Weich,N. and Nathan,C.
    Mycobacterium tuberculosis prcBA genes encode a gated proteasome with broad oligopeptide specificity
    Mol Microbiol59, 1405-1416. PubMed  Europe PubMed DOI  P
  45. [YEAR:2-11-2006]Pearce,M.J., Arora,P., Festa,R.A., Butler-Wu,S.M., Gokhale,R.S. and Darwin,K.H.
    Identification of substrates of the Mycobacterium tuberculosis proteasome
    EMBO J25, 5423-5432. PubMed  Europe PubMed DOI
    46. 2005
  46. Hong,B., Wang,L., Lammertyn,E., Geukens,N., Van Mellaert,L., Li,Y. and Anne,J.
    Inactivation of the 20S proteasome in Streptomyces lividans and its influence on the production of heterologous proteins
    Microbiology (Reading)151, 3137-3145. PubMed  Europe PubMed DOI  K
    47. 2004
  47. [YEAR:2-1-2004]Kwon,Y.D., Nagy,I., Adams,P.D., Baumeister,W. and Jap,B.K.
    Crystal structures of the Rhodococcus proteasome with and without its pro-peptides: implications for the role of the pro-peptide in proteasome assembly
    J Mol Biol335, 233-245. PubMed  Europe PubMed DOI
  48. Lupas,A., Kania,M. and Baumeister,W.
    Bacterial proteasome
    [ISSN:0-12-079610-4]2, 2061-2063.  V
    49. 2003
  49. [YEAR:12-12-2003]Darwin,K.H., Ehrt,S., Gutierrez-Ramos,J.C., Weich,N. and Nathan,C.F.
    The proteasome of Mycobacterium tuberculosis is required for resistance to nitric oxide
    Science302, 1963-1966. PubMed  Europe PubMed DOI
    50. 2000
  50. Pouch,M.N., Cournoyer,B. and Baumeister,W.
    Characterization of the 20S proteasome from the actinomycete Frankia
    Mol Microbiol35, 368-377. PubMed  Europe PubMed DOI
    51. 1999
  51. De Mot,R., Nagy,I., Walz,J. and Baumeister,W.
    Proteasomes and other self-compartmentalizing proteases in prokaryotes
    Trends Microbiol7, 88-92. PubMed  Europe PubMed DOI
    52. 1998
  52. De Mot,R., Nagy,I. and Baumeister,W.
    A self-compartmentalizing protease in Rhodococcus: the 20S proteasome
    Antonie Van Leeuwenhoek74, 83-87. PubMed  Europe PubMed DOI
  53. Mayr,J., Seemuller,E., Muller,S.A., Engel,A. and Baumeister,W.
    Late events in the assembly of 20S proteasomes
    J Struct Biol124, 179-188. PubMed  Europe PubMed DOI
  54. Nagy,I., Tamura,T., Vanderleyden,J., Baumeister,W. and De Mot,R.
    The 20S proteasome of Streptomyces coelicolor
    J Bacteriol180, 5448-5453. PubMed  Europe PubMed
    55. 1997
  55. Knipfer,N. and Shrader,T.E.
    Inactivation of the 20S proteasome in Mycobacterium smegmatis
    Mol Microbiol25, 375-383. PubMed  Europe PubMed  K
  56. [YEAR:17-10-1997]Mc Cormack,T., Baumeister,W., Grenier,L., Moomaw,C., Plamondon,L., Pramanik,B., Slaughter,C., Soucy,F., Stein,R., Zuhl,F. and Dick,L.
    Active site-directed inhibitors of Rhodococcus 20 S proteasome. Kinetics and mechanism
    J Biol Chem272, 26103-26109. PubMed  Europe PubMed DOI  I
  57. [YEAR:2-1-1997]Zuhl,F., Tamura,T., Dolenc,I., Cejka,Z., Nagy,I., De Mot,R. and Baumeister,W.
    Subunit topology of the Rhodococcus proteasome
    FEBS Lett400, 83-90. PubMed  Europe PubMed DOI
    58. 1996
  58. Aoyama,K., Zuhl,F., Tamura,T. and Baumeister,W.
    2-D crystallization of the Rhodococcus 20S proteasome
    J Struct Biol116, 438-442. PubMed  Europe PubMed
    59. 1995
  59. [YEAR:1-7-1995]Tamura,T., Nagy,I., Lupas,A., Lottspeich,F., Cejka,Z., Schoofs,G., Tanaka,K., De Mot,R. and Baumeister,W.
    The first characterization of a eubacterial proteasome: the 20S complex of Rhodococcus
    Curr Biol5, 766-774. PubMed  Europe PubMed
    60. 1992
  60. Benoist,P., Muller,A., Diem,H.G. and Schwencke,J.
    High-molecular-mass multicatalytic proteinase complexes produced by the nitrogen-fixing actinomycete Frankia strain BR
    J Bacteriol174, 1495-1504. PubMed  Europe PubMed

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