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Literature for subfamily S1A

Summary Distribution Literature

(Topics flags: S Structure, I Inhibitor, P Specificity, V Review. To select only the references relevant to a single topic, click the link above. See explanation.)

    2025
  1. Cheng,Y., Su,J., Jiao,Q., Jia,T. and Hu,X.
    Recent advance on the physiological functions of proteases in chloroplast
    Biochem Biophys Res Commun765, 151813-151813. PubMed  Europe PubMed DOI  V
    2. 2024
  2. Aubert,A., Jung,K., Hiroyasu,S., Pardo,J. and Granville,D.J.
    Granzyme serine proteases in inflammation and rheumatic diseases
    Nat Rev Rheumatol20, 361-376. PubMed  Europe PubMed DOI
  3. Cigalotto,L. and Martinvalet,D.
    Granzymes in health and diseases: the good, the bad and the ugly
    Front Immunol15, 1371743-1371743. PubMed  Europe PubMed DOI
  4. Daneva,G.N., Tsiakanikas,P., Adamopoulos,P.G. and Scorilas,A.
    Kallikrein-related peptidases: mechanistic understanding for potential therapeutic targeting in cancer
    Expert Opin Ther Targets1-20. PubMed  Europe PubMed DOI  V
  5. Lin,H., Xu,M., Jiang,L., Yuan,C., Jiang,C., Huang,M., Li,J. and Xu,P.
    Water-medicated specifically targeting the S1 pockets among serine proteases using an arginine analogue
    Bioorg Chem152, 107734-107734. PubMed  Europe PubMed DOI
  6. Morejon,B. and Michel,K.
    The expanded immunoregulatory protease network in mosquitoes is governed by gene co-expression
    bioRxiv PubMed  Europe PubMed DOI
  7. Sun,J., Liu,C., Wang,L. and Song,L.
    The Establishment of Complement System Is from Gene Duplication and Domain Shuffling
    Int J Mol Sci25, PubMed  Europe PubMed DOI
    8. 2023
  8. Gul,I., Abbas,M.N., Kausar,S., Luo,J., Gao,X., Mu,Y., Fan,W. and Cui,H.
    Insight into crustacean cathepsins: Structure-evolutionary relationships and functional roles in physiological processes
    Fish Shellfish Immunol139, 108852-108852. PubMed  Europe PubMed DOI  V
    9. 2022
  9. Coban,A., Bornberg-Bauer,E. and Kemena,C.
    Domain Evolution of Vertebrate Blood Coagulation Cascade Proteins
    J Mol Evol90, 418-428. PubMed  Europe PubMed DOI
  10. Lee,K.Y., Chau,C.H., Price,D.K. and Figg,W.D.
    Drugging the undruggable: activity-based protein profiling offers opportunities for targeting the KLK activome
    Cancer Biol Ther23, 136-138. PubMed  Europe PubMed DOI
  11. Matus,C.E., Ehrenfeld,P. and Figueroa,C.D.
    The family of kallikrein-related peptidases and kinin peptides as modulators of epidermal homeostasis
    Am J Physiol Cell Physiol323, C1070-C1070. PubMed  Europe PubMed DOI  V
  12. Morizane,S., Sunagawa,K., Nomura,H. and Ouchida,M.
    Aberrant serine protease activities in atopic dermatitis
    J Dermatol Sci107, 2-7. PubMed  Europe PubMed DOI
  13. Song,Y., Ke,Y., Kang,M. and Bao,R.
    Function, molecular mechanisms, and therapeutic potential of bacterial HtrA proteins: An evolving view
    Comput Struct Biotechnol J20, 40-49. PubMed  Europe PubMed DOI  V
  14. Sotiropoulou,G., Zingkou,E. and Pampalakis,G.
    Novel specific activity-based probes validate KLK proteases as druggable targets
    Cancer Biol Ther23, 401-403. PubMed  Europe PubMed DOI
  15. Tagirasa,R. and Yoo,E.
    Role of Serine Proteases at the Tumor-Stroma Interface
    Front Immunol13, 832418-832418. PubMed  Europe PubMed DOI  V
  16. Zupanic,N., Pocic,J., Leonardi,A., Sribar,J., Kordis,D. and Krizaj,I.
    Serine pseudoproteases in physiology and disease
    FEBS J PubMed  Europe PubMed DOI  V
    17. 2021
  17. Weiss,S.A.I., Rehm,S.R.T., Perera,N.C., Biniossek,M.L., Schilling,O. and Jenne,D.E.
    Origin and Expansion of the Serine Protease Repertoire in the Myelomonocyte Lineage
    Int J Mol Sci22, PubMed  Europe PubMed DOI
    18. 2019
  18. Goettig,P., Brandstetter,H. and Magdolen,V.
    Surface loops of trypsin-like serine proteases as determinants of function
    Biochimie166, 52-76. PubMed  Europe PubMed DOI  P
    19. 2018
  19. Iqbal,M., Dubey,M., Gudmundsson,M., Viketoft,M., Jensen,D.F. and Karlsson,M.
    Comparative evolutionary histories of fungal proteases reveal gene gains in the mycoparasitic and nematode-parasitic fungus Clonostachys rosea
    BMC Evol Biol18, 171-171. PubMed  Europe PubMed DOI
    20. 2017
  20. Premzl,M.
    Comparative genomic analysis of eutherian kallikrein genes
    Mol Genet Metab Rep10, 96-99. PubMed  Europe PubMed DOI
    21. 2016
  21. Waldner,B.J., Fuchs,J.E., Huber,R.G., von Grafenstein,S., Schauperl,M., Kramer,C. and Liedl,K.R.
    Quantitative correlation of conformational binding enthalpy with substrate specificity of serine proteases
    J Phys Chem B120, 299-308. PubMed  Europe PubMed DOI
    22. 2015
  22. Akula,S., Thorpe,M., Boinapally,V. and Hellman,L.
    Granule associated serine proteases of hematopoietic cells - an analysis of their appearance and diversification during vertebrate evolution
    PLoS ONE10, 0143091- PubMed  Europe PubMed DOI
  23. Cao,X., He,Y., Hu,Y., Zhang,X., Wang,Y., Zou,Z., Chen,Y., Blissard,G.W., Kanost,M.R. and Jiang,H.
    Sequence conservation, phylogenetic relationships, and expression profiles of nondigestive serine proteases and serine protease homologs in Manduca sexta
    Insect Biochem Mol Biol62, 51-63. PubMed  Europe PubMed DOI
  24. Dias,R.O., Via,A., Brandao,M.M., Tramontano,A. and Silva-Filho,M.C.
    Digestive peptidase evolution in holometabolous insects led to a divergent group of enzymes in Lepidoptera
    Insect Biochem Mol Biol58, 1-11. PubMed  Europe PubMed DOI
    25. 2014
  25. Ahmad,J., Bird,P.I. and Kaiserman,D.
    Analysis of the evolution of granule associated serine proteases of immune defence (GASPIDs) suggests a revised nomenclature
    Biol Chem395, 1253-1262. PubMed  Europe PubMed DOI
  26. Douaiher,J., Succar,J., Lancerotto,L., Gurish,M.F., Orgill,D.P., Hamilton,M.J., Krilis,S.A. and Stevens,R.L.
    Development of mast cells and importance of their tryptase and chymase serine proteases in inflammation and wound healing
    Adv Immunol122, 211-252. PubMed  Europe PubMed DOI  V
  27. Pustelny,K., Zdzalik,M., Stach,N., Stec-Niemczyk,J., Cichon,P., Czarna,A., Popowicz,G., Mak,P., Drag,M., Salvesen,G.S., Wladyka,B., Potempa,J., Dubin,A. and Dubin,G.
    Staphylococcal SplB serine protease utilizes a novel molecular mechanism of activation
    J Biol Chem289, 15544-15553. PubMed  Europe PubMed DOI
    28. 2013
  28. Koumandou,V.L. and Scorilas,A.
    Evolution of the plasma and tissue kallikreins, and their alternative splicing isoforms
    PLoS ONE8, e68074-e68074. PubMed  Europe PubMed DOI
    29. 2011
  29. Gohara,D.W. and Di Cera,E.
    Allostery in trypsin-like proteases suggests new therapeutic strategies
    Trends Biotechnol29, 577-585. PubMed  Europe PubMed DOI
  30. Wahlgren,W.Y., Pal,G., Kardos,J., Porrogi,P., Szenthe,B., Patthy,A., Graf,L. and Katona,G.
    The catalytic aspartate is protonated in the Michaelis complex formed between trypsin and an in vitro evolved substrate-like inhibitor: a refined mechanism of serine protease action
    J Biol Chem286, 3587-3596. PubMed  Europe PubMed DOI  S
    31. 2010
  31. Antalis,T.M., Buzza,M.S., Hodge,K.M., Hooper,J.D. and Netzel-Arnett,S.
    The cutting edge: membrane-anchored serine protease activities in the pericellular microenvironment
    Biochem J428, 325-346. PubMed  Europe PubMed DOI  V
  32. Anthony,D.A., Andrews,D.M., Watt,S.V., Trapani,J.A. and Smyth,M.J.
    Functional dissection of the granzyme family: cell death and inflammation
    Immunol Rev235, 73-92. PubMed  Europe PubMed DOI  V
  33. Trivedi,N.N. and Caughey,G.H.
    Mast cell peptidases: chameleons of innate immunity and host defense
    Am J Respir Cell Mol Biol42, 257-267. PubMed  Europe PubMed DOI
    34. 2009
  34. Bugge,T.H., Antalis,T.M. and Wu,Q.
    Type II transmembrane serine proteases
    J Biol Chem284, 23177-23181. PubMed  Europe PubMed DOI  V
    35. 2008
  35. Jang,I.H., Nam,H.J. and Lee,W.J.
    CLIP-domain serine proteases in Drosophila innate immunity
    BMB Rep41, 102-107. PubMed  Europe PubMed
  36. Lundwall,A. and Brattsand,M.
    Kallikrein-related peptidases
    Cell Mol Life Sci65, 2019-2038. PubMed  Europe PubMed DOI
  37. Schmidt,A.E., Sun,M.F., Ogawa,T., Bajaj,S.P. and Gailani,D.
    Functional role of residue 193 (chymotrypsin numbering) in serine proteases: influence of side chain length and beta-branching on the catalytic activity of blood coagulation factor XIa
    Biochemistry47, 1326-1335. PubMed  Europe PubMed DOI
  38. Shah,P.K., Tripathi,L.P., Jensen,L.J., Gahnim,M., Mason,C., Furlong,E.E., Rodrigues,V., White,K.P., Bork,P. and Sowdhamini,R.
    Enhanced function annotations for Drosophila serine proteases: a case study for systematic annotation of multi-member gene families
    Gene407, 199-215. PubMed  Europe PubMed DOI
    39. 2007
  39. [YEAR:1-2-2007]Xu,H., Shan,J., Jurukovski,V., Yuan,L., Li,J. and Tian,K.
    TSP50 encodes a testis-specific protease and is negatively regulated by p53
    Cancer Res67, 1239-1245. PubMed  Europe PubMed DOI
    40. 2006
  40. Srinivasan,A., Giri,A.P. and Gupta,V.S.
    Structural and functional diversities in lepidopteran serine proteases
    Cell Mol Biol Lett11, 132-154. PubMed  Europe PubMed DOI
    41. 2005
  41. Page,M.J., MacGillivray,R.T. and Di Cera,E.
    Determinants of specificity in coagulation proteases
    J Thromb Haemost3, 2401-2408. PubMed  Europe PubMed DOI
  42. Zamolodchikova,T.S., Smirnova,E.V., Andrianov,A.N., Kashparov,I.V., Kotsareva,O.D., Sokolova,E.A., Ignatov,K.B. and Pemberton,A.D.
    Cloning and molecular modeling of duodenase with respect to evolution of substrate specificity within mammalian serine proteases that have lost a conserved active-site disulfide bond
    Biochemistry (Mosc)70, 672-684. PubMed  Europe PubMed DOI
    43. 2004
  43. Castro,H.C., Zingali,R.B., Albuquerque,M.G., Pujol-Luz,M. and Rodrigues,C.R.
    Snake venom thrombin-like enzymes: from reptilase to now
    Cell Mol Life Sci61, 843-856. PubMed  Europe PubMed DOI
  44. Clements,J.A., Willemsen,N.M., Myers,S.A. and Dong,Y.
    The tissue kallikrein family of serine proteases: functional roles in human disease and potential as clinical biomarkers
    Crit Rev Clin Lab Sci41, 265-312. PubMed  Europe PubMed DOI
  45. Olsson,A.Y., Lilja,H. and Lundwall,A.
    Taxon-specific evolution of glandular kallikrein genes and identification of a progenitor of prostate-specific antigen
    Genomics84, 147-156. PubMed  Europe PubMed DOI
    46. 2003
  46. [YEAR:13-5-2003]Bergstrom,R.C., Coombs,G.S., Ye,S., Madison,E.L., Goldsmith,E.J. and Corey,D.R.
    Binding of nonphysiological protein and peptide substrates to proteases: differences between urokinase-type plasminogen activator and trypsin and contributions to the evolution of regulated proteolysis
    Biochemistry42, 5395-5402. PubMed  Europe PubMed DOI
  47. Grossman,W.J., Revell,P.A., Lu,Z.H., Johnson,H., Bredemeyer,A.J. and Ley,T.J.
    The orphan granzymes of humans and mice
    Curr Opin Immunol15, 544-552. PubMed  Europe PubMed DOI  V
  48. Netzel-Arnett,S., Hooper,J.D., Szabo,R., Madison,E.L., Quigley,J.P., Bugge,T.H. and Antalis,T.M.
    Membrane anchored serine proteases: a rapidly expanding group of cell surface proteolytic enzymes with potential roles in cancer
    Cancer Metastasis Rev22, 237-258. PubMed  Europe PubMed DOI  V
  49. Szabo,R., Wu,Q., Dickson,R.B., Netzel-Arnett,S., Antalis,T.M. and Bugge,T.H.
    Type II transmembrane serine proteases
    Thromb Haemost90, 185-193. PubMed  Europe PubMed DOI  V
    50. 2002
  50. [YEAR:25-10-2002]Krem,M.M., Prasad,S. and Di Cera,E.
    Ser(214) is crucial for substrate binding to serine proteases
    J Biol Chem277, 40260-40264. PubMed  Europe PubMed DOI
    51. 2001
  51. Nakao,M., Osaka,K., Kato,Y., Fujiki,K. and Yano,T.
    Molecular cloning of the complement C1r/C1s/MASP2-like serine proteases from the common carp (Cyprinus carpio)
    Immunogenetics52, 255-263. PubMed  Europe PubMed DOI
    52. 2000
  52. [YEAR:17-10-2000]Gan,L., Lee,I., Smith,R., Argonza-Barrett,R., Lei,H., McCuaig,J., Moss,P., Paeper,B. and Wang,K.
    Sequencing and expression analysis of the serine protease gene cluster located in chromosome 19q13 region
    Gene257, 119-130. PubMed  Europe PubMed DOI
  53. [YEAR:1-12-2000]Harvey,T.J., Hooper,J.D., Myers,S.A., Stephenson,S.A., Ashworth,L.K. and Clements,J.A.
    Tissue-specific expression patterns and fine mapping of the human kallikrein (KLK) locus on proximal 19q13.4
    J Biol Chem275, 37397-37406. PubMed  Europe PubMed DOI
  54. Jiang,H. and Kanost,M.R.
    The clip-domain family of serine proteinases in arthropods
    Insect Biochem Mol Biol30, 95-105. PubMed  Europe PubMed DOI
  55. [YEAR:7-3-2000]Kam,C.M., Hudig,D. and Powers,J.C.
    Granzymes (lymphocyte serine proteases): characterization with natural and synthetic substrates and inhibitors
    Biochim Biophys Acta1477, 307-323. PubMed  Europe PubMed DOI  V
  56. Krem,M.M., Rose,T. and Di Cera,E.
    Sequence determinants of function and evolution in serine proteases
    Trends Cardiovasc Med10, 171-176. PubMed  Europe PubMed DOI
  57. [YEAR:7-3-2000]Matsui,T., Fujimura,Y. and Titani,K.
    Snake venom proteases affecting hemostasis and thrombosis
    Biochim Biophys Acta1477, 146-156. PubMed  Europe PubMed DOI
  58. Poorafshar,M., Aveskogh,M., Munday,B. and Hellman,L.
    Identification and structural analysis of four serine proteases in a monotreme, the platypus, Ornithorhynchus anatinus
    Immunogenetics52, 19-28. PubMed  Europe PubMed DOI
  59. [YEAR:16-9-2000]Yousef,G.M., Chang,A., Scorilas,A. and Diamandis,E.P.
    Genomic organization of the human kallikrein gene family on chromosome 19q13.3-q13.4
    Biochem Biophys Res Commun276, 125-133. PubMed  Europe PubMed DOI
    60. 1998
  60. Baptista,A.M., Jonson,P.H., Hough,E. and Petersen,S.B.
    The origin of trypsin: Evidence for multiple gene duplications in trypsins
    J Mol Evol47, 353-362. PubMed  Europe PubMed DOI
  61. Matsushita,M., Endo,Y., Nonaka,M. and Fujita,T.
    Complement-related serine proteases in tunicates and vertebrates
    Curr Opin Immunol10, 29-35. PubMed  Europe PubMed DOI
  62. Takeda-Shitaka,M. and Umeyama,H.
    Effect of exceptional valine replacement for highly conserved alanine-55 on the catalytic site structure of chymotrypsin-like serine protease
    Chem Pharm Bull (Tokyo)46, 1343-1348. PubMed  Europe PubMed
  63. [YEAR:3-4-1998]Takeda-Shitaka,M. and Umeyama,H.
    Elucidation of the cause for reduced activity of abnormal human plasmin containing an Ala55-Thr mutation: Importance of highly conserved Ala55 in serine proteases
    FEBS Lett425, 448-452. PubMed  Europe PubMed DOI
    64. 1997
  64. Chen,L., DeVries,A.L. and Cheng,C.H.
    Evolution of antifreeze glycoprotein gene from a trypsinogen gene in Antarctic notothenioid fish
    Proc Natl Acad Sci U S A94, 3811-3816. PubMed  Europe PubMed DOI
  65. Ji,X., Azumi,K., Sasaki,M. and Nonaka,M.
    Ancient origin of the complement lectin pathway revealed by molecular cloning of mannan binding protein-associated serine protease from a urochordate, the Japanese ascidian, Halocynthia roretzi
    Proc Natl Acad Sci U S A94, 6340-6345. PubMed  Europe PubMed DOI
  66. Roach,J.C., Wang,K., Gan,L. and Hood,L.
    The molecular evolution of the vertebrate trypsinogens
    J Mol Evol45, 640-652. PubMed  Europe PubMed DOI
    67. 1996
  67. [YEAR:1-10-1996]Dang,Q.D. and Di Cera,E.
    Residue 225 determines the Na(+)-induced allosteric regulation of catalytic activity in serine proteases
    Proc Natl Acad Sci U S A93, 10653-10656. PubMed  Europe PubMed DOI
    68. 1995
  68. Male,R., Lorens,J.B., Smalas,A.O. and Torrissen,K.R.
    Molecular cloning and characterization of anionic and cationic variants of trypsin from Atlantic salmon
    Eur J Biochem232, 677-685. PubMed  Europe PubMed DOI
    69. 1994
  69. Huang,R. and Hellman,L.
    Genes for mast-cell serine protease and their molecular evolution
    Immunogenetics40, 397-414. PubMed  Europe PubMed
  70. Rypniewski,W.R., Perrakis,A., Vorgias,C.E. and Wilson,K.S.
    Evolutionary divergence and conservation of trypsin
    Protein Eng7, 57-64. PubMed  Europe PubMed
    71. 1993
  71. Patthy,L.
    Modular design of proteases of coagulation, fibrinolysis, and complement activation: implications for protein engineering and structure-function studies
    Methods Enzymol222, 10-21. PubMed  Europe PubMed DOI  V
  72. [YEAR:1-10-1993]Perkins,S.J. and Smith,K.F.
    Identity of the putative serine-proteinase fold in proteins of the complement system with nine relevant crystal structures
    Biochem J295, 109-114. PubMed  Europe PubMed  S
    73. 1991
  73. Klemm,U., Flake,A. and Engel,W.
    Rat sperm acrosin: cDNA sequence, derived primary structure and phylogenetic origin
    Biochim Biophys Acta1090, 270-272. PubMed  Europe PubMed DOI
  74. Salvesen,G. and Enghild,J.J.
    Zymogen activation specificity and genomic structures of human neutrophil elastase and cathepsin G reveal a new branch of the chymotrypsinogen superfamily of serine proteinases
    Biomed Biochim Acta50, 665-671. PubMed  Europe PubMed
    75. 1960
  75. Sanger,F. and Shaw,D.C.
    Amino-acid sequence about the reactive serine of a proteolytic enzyme from Bacillus subtilis
    Nature187, 872-873. PubMed  Europe PubMed DOI  I

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