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Miyamoto,Y., Banno,Y., Yamashita,T., Fujimoto,T., Oi,S., Moritoh,Y., Asakawa,T., Kataoka,O., Yashiro,H., Takeuchi,K., Suzuki,N., Ikedo,K., Kosaka,T., Tsubotani,S., Tani,A., Sasaki,M., Funami,M., Amano,M., Yamamoto,Y., Aertgeerts,K., Yano,J. and Maezaki,H.
Discovery of a 3-pyridylacetic acid derivative (TAK-100) as a potent, selective and orally active dipeptidyl peptidase IV (DPP-4) inhibitor
J Med Chem54, 831-850. PubMed Europe PubMed DOI I
2011
