2010
  1. Meng,W., Brigance,R.P., Chao,H.J., Fura,A., Harrity,T., Marcinkeviciene,J., O'Connor,S.P., Tamura,J.K., Xie,D., Zhang,Y., Klei,H.E., Kish,K., Weigelt,C.A., Turdi,H., Wang,A., Zahler,R., Kirby,M.S. and Hamann,L.G.
    Discovery of 6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methylimidazo[1,2-a]pyrimidine-2-carboxamides as potent, selective dipeptidyl peptidase-4 (DPP4) inhibitors
    J Med Chem53, 5620-5628. PubMed  Europe PubMed DOI  I