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[YEAR:15-2-2001]Pinto,D.J., Orwat,M.J., Wang,S., Fevig,J.M., Quan,M.L., Amparo,E., Cacciola,J., Rossi,K.A., Alexander,R.S., Smallwood,A.M., Luettgen,J.M., Liang,L., Aungst,B.J., Wright,M.R., Knabb,R.M., Wong,P.C., Wexler,R.R. and Lam,P.Y.
Discovery of 1-[3-(aminomethyl)phenyl]-N-3-fluoro-2'-(methylsulfonyl)-[1,1'-biphenyl]-4 -yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide (DPC423), a highly potent, selective, and orally bioavailable inhibitor of blood coagulation factor Xa
J Med Chem44, 566-578. PubMed Europe PubMed DOI I
2001
