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What peptidase is affected by this inhibitor?
Substrate name :
inhibitor name
(1S,2S)-2-amino-1-(4-nitrophenyl) propane-1,3-diol compound 13b
(2-benzyl-3-mercaptopropanoyl)-L-alanylglycinamide
(2R,3S)-AHPB-Pro
(2S,3R)-AHMH-Pro
(2S,3R)-AHMH-Thia
(2S,3R)-AHPB-Pro
(2S,3R)-AHPB-Pro-OMe
(2S,3R)-AHPB-Pro-Phe-OMe
(3S,4S)-3-amino-4-mercapto-6-phenyl-hexane-1-sulfonic acid (aminopeptidase A inhibitor)
(Asp-Arg)9-Leu-Pro-Tyr-CO-NHOH
(Asp-Arg)9-Trp-Leu-et-CO-NHOH
(Asp-Arg)9-Val-Leu-Arg-CO-NHOH
(CYGAK)(2)
(p-amidinophenyl)methanesulfonate
(R)-2-(3-
[amino(imino) methyl]amino
phenyl)-3-sulfanylpropanoic acid
(S)-(+)-5-[1-(2-methoxymethylpyrrolidinyl)sulfonyl]isatin
1,10-phenanthroline
1,3-di-(N-benzyloxycarbonyl-L-leucyl-L-leucyl)aminoacetone
1,3-bis(CBZ Leu-NH)-2-propanone
1-chloro-3-amino-4-phenyl-butanone-2
2,2’-Bipyridine
2,2’-dipyridyldisulfide
2-(3-benzylureido)-Lys-Lys-Arg-H
2-(3-mercaptopropyl)pentanedioic acid (GCP II inhibitor)
2-(5-
[amino(imino)methyl]amino
-2-chlorophenyl)-3-sulfanylpropanoic acid
2-(7-methoxy-naphthyl)-propanoyl-Lys-Lys-Arg-H
2-aminobenzoyl-Lys-Lys-Arg-H
2-benzyl-3,4-epithiobutanoic acid
2-benzyl-3,4-epoxybutanoic acid (BEBA)
2-benzyl-3,4-iminobutanoic acid
2-benzyl-3-iodopropanoic acid
2-benzyl-5-nitro-4-oxopentanoic acid
2-mercaptoacetyl-L-leucyl-L-phenylalanine
2-mercaptoacetyl-L-phenylalanyl-L-leucine
2-mercaptomethyl-3-guanidinoethylthiopropanoic acid (metallocarboxypeptidase/aminopeptidase inhibitor)
2-naphthoyl-Lys-Lys-Arg-H
2-phenylethaneboronic acid
3-(dihydroxyboryl)benzoic acid 1
3-amino-cyclic-imide compound 13a
3-amino-cyclic-imide compound 13b
3-amino-cyclic-imide compound 13d
3-amino-cyclic-imide compound 13e
3-amino-cyclic-imide compound 13f
3-amino-cyclic-imide compound 13g
3-amino-cyclic-imide compound 13h
3-amino-cyclic-imide compound 13i
3-mercaptoisobutyrate
3-mercaptopropionate
3-methoxy-phenacetyl-Lys-Lys-Arg-H
3-phenylpropane-1,2-diamine compound 12i
3-phenylpropane-1,2-diamine compound A6
3-phenylpropane-1,2-diamine compound B6
3-TAPAP
3-thienylalanine-ornithine-proline (ACE inhibitor)
4-(2-aminoethyl)-benzensulfonyl fluoride
4-chloro-3-(3-isothiureidopropoxy)isocoumarin
4-chloro-3-ethoxy-7-guanidinoisocoumarin (trypsin inhibitor)
4-chloro-7-guanidino-3-methoxyisocoumarin
4-hydroxy-2-nonenal (HNE)
4-hydroxymercuribenzoate
4-phenyl-phenacetyl-Lys-Lys-Arg-H
5,5’-dithiobis-2-nitrobenzoic acid (DTNB)
5-oxoprolinal (pyroglutamyl peptidase I inhibitor)
5-S-5-benzamido-4-oxo-6-phenylhexanoyl-L-proline
5-S-5-benzamido-4-oxo-6-phenylhexanoyl-L-tryptophan
5-
[amino(imino)methyl]amino
-2-(sulfanylmethyl)pentanoic acid
5S,6S penem (inhibitor of signal peptidase I)
6-beta-iodopenicillanate
6-diazo-5-oxo-D-norleucine (gamma-glutamyltranspeptidase inhibitor)
6-diazo-5-oxo-L-norleucylglycine (gamma-glutamyl transpeptidase inhibitor)
6-mercaptopurine
6-thioguanine
7-amino-3-(2-bromoethoxy)-4-chloroisocoumarin (pancreatic elastase inhibitor)
8-hydroxyquinoline
A-310840
A-311263
A-357300 (MetAP2 inhibitor)
A-705239 (calpain-1 inhibitor)
A-705253
A-74704 (retropepsin inhibitor)
A-77003 (retropepsin inhibitor)
A-790742 (retropepsin inhibitor)
A-792611 (retropepsin inhibitor)
A-80987 (retropepsin inhibitor)
A-84538 (retropepsin inhibitor)
A70450 (candidapepsin inhibitor)
AAE581 (cathepsin K inhibitor)
AaTI (
Aedes aegypti
)
AB192 (DPP4 inhibitor)
ABBA (gamma-glutamyl transpeptidase inhibitor)
ABT-279 (DPP4 inhibitor)
ABT-341 (DPP4 inhibitor)
ABZ-Arg-Gln-Asp-Arg-H
ABZ-Arg-Gln-Asp-Lys-H
Abz-Gly-Phe-Ser-Ile-Phe-Arg-Gln-EDDnp
Abz-Gly-Phe-Ser-Pro-Pro-Arg-Gln-EDDnp
Ac-APnLD-al (acetyl-Ala-Pro-norLeu-Asp-aldehyde)
Ac-Asp-Glu-Val-Asp-H
Ac-Asp-Val-Ala-Asp-CH(2)F
ac-Gly-Val-Arg-chloromethyltrifluoroacetate
Ac-His-Pro? (PO2-CH2)Isoxa(Phe)a -OH
Ac-Ile-Glu-Thr-Asp-CHO
Ac-Ile-Glu-Thr-Asp-H
Ac-KPI-1 I (
Ancylostoma caninum
) inhibitor unit 5, 6, or 8
Ac-Leu-Ala-Ala-Gln(Me2)-FMK
Ac-Leu-Ala-Ala-Gln(Me2)-pMK
Ac-Leu-Leu-Met-H
Ac-Leu-Leu-Nle-H
Ac-Leu-Phe-Phe-Glu-FMK
Ac-Lys-Thr-Glu-Glu-Ile-Ser-Val-Val-Sta-Val-Ala-Glu-Phe
Ac-Phe-Ala-Ser-Gly-Lys-Arg-H
Ac-Phe-Glu-Lys-Ala-cmk
Ac-Pro-Arg-Leu-AsnVS
Ac-Trp-Glu-His-Asp-H
Ac-Tyr-Val-Ala-Asp-H
Ac-Val-Glu-Ile-Asp-CHO
Ac-YVAD-CMK
Ac-YVKD-CMK
acetamidoacetonitrile
acetyl-Leu-Val-Lys-CHO
acivicin
aclacinomycin A
Acp62F protein (
Drosophila melanogaster
)
actinonin
Ada-Ahx3-L3VS
AE-3763 (neutrophil elastase inhibitor)
AEBSF
aeropin
aeruginosin EI461
AG-1776 (retropepsin inhibitor)
agaricoglyceride A
agaricoglyceride monoacetate
Agariogylceride A
ageladine A (MMP-12 inhibitor)
AK275 (calpain inhibitor)
Ala-Ala-Phe-CH(2)Cl
Ala-Ala-Phe-chloromethyl ketone
alaserpin (Lepidoptera)
aliskiren
ALLM
ALLN
alocasin
alogliptin
alpha-1-antichymotrypsin
alpha-1-peptidase inhibitor
alpha-2-HS-glycoprotein
alpha-2-HS-glycoprotein inhibitor unit 2
alpha-2-macroglobulin
alpha-2-macroglobulin-like 1 protein
alpha-amylase/subtilisin inhibitor (
Hordeum
-type)
alpha-benzyl-2-oxo-1,3-oxazolidine-4-acetic acid (BOOA)
alpha-diazo-p-bromoacetophenone
ALS 1-0635 (MMP13 inhibitor)
AMAC
amastatin
amblin inhibitor unit 1 (
Amblyomma hebraeum
)
AmFPI-1 (
Antheraea mylitta
)
AMG-126737 (tryptase inhibitor)
amoebiasin-1
amoebiasin-2
ampicillin
amprenavir
amyloid precursor-like protein 2
anabaenopeptin G (carboxypeptidase A inhibitor)
anabaenopeptin H
ancovenin
angiotensin IV
anilide inhibitor (SARS-CoV 3CL peptidase inhibitor)
anophelin
antihemorrhagic factor (
Gloydius blomhoffi
)
antipain
antistasin
antistasin inhibitor unit 1
antithrombin
APC 2059
APC-366 (tryptase inhibitor)
APC2848
APC3328
apixaban
APMSF
apratastat (TACE/MMP inhibitor)
aprin
aprotinin
apstatin
Arg-Thr-Ser-Lys-Lys-Arg
argatroban
argyrin A
ARH067637
arphamenine A
arphamenine B
Artemisinin-dipeptidyl vinyl sulfone compound 6a
Artemisinin-dipeptidyl vinyl sulfone compound 6b
Artemisinin-dipeptidyl vinyl sulfone compound 6c
Artemisinin-dipeptidyl vinyl sulfone compound 6d
arylomycin A2
AS-101 compound
AS111793 (MMP-12 inhibitor)
Ascaris trypsin inhibitor
ascidian trypsin inhibitor
Asp-?[PO2CH2]-LeuOH
ASP4000 (DPP IV inhibitor)
ASP8497 (DPP4 inhibitor)
aspartate thiol
aspartic protease inhibitor (
Bacillus licheniformis
)
Aspergillus elastase inhibitor
aspin
aspin-2
assemblin dimerization inhibitor
atazanavir
AtSerpin1 (
Arabidopsis thaliana
)
auranofin
aurintricarboxylic acid (ATA) (calpain inhibitor)
AVR2 protein (
Passalora
sp.)
B27-HYD (calpain inhibitor)
bacitracin A
bacterial serpin (
Bifidobacterium longum
)
bacteriophage lambda CIII protein
baculovirus P35 caspase inhibitor
baculovirus P49 caspase inhibitor
BAL0019193 (signal peptidase I inhibitor)
balicatib (cathepsin K inhibitor)
BAPTA (1,2-bis-(O-aminophenoxy)ethane-N,N,N¢,N¢-tetraacetic acid)
barley trypsin/factor XIIa inhibitor
barley-type serpin
batimastat
Bauhinia trypsin/plasma kallikrein inhibitor
BAY-129566
BCEAB
BCH-2763
bdellastasin
bdellin
begacestat (gamma-secretase inhibitor)
belactosin A
benarthin (pyroglutamyl peptidase inhibitor)
benazeprilat
benzamidine
benzamidoacetonitrile
benzothiazolium compound A01652
benzothiazolium compound A05175
benzothiazolium compound A06725
benzothiazolium compound A09853
benzothiazolium compound A10059
benzothiazolium compound A11605
benzothiazolium compound A17394
benzothiazolium compound A33224
benzothiazolium compound A36638
benzothiazolium compound A38120
benzothiazolium compound A39949
benzothiazolium compound A40437
benzothiazolium compound A41369
benzothiazolium compound A41558
benzothiazolium compound A51818
benzothiazolium compound A51828
benzothiazolium compound A51849
benzothiazolium compound A51858
benzothiazolium compound A51894
benzylpenicillin
benzylsuccinic acid
bestatin
beverimat (retropepsin inhibitor)
bifunctional aspartic peptidase inhibitor (
Bacillus
sp.)
bikazin salivary inhibitor inhibitor unit 1
bikazin salivary inhibitor inhibitor unit 2
bikunin
bikunin inhibitor unit 1
bikunin inhibitor unit 2
BIL-DMK diazomethylketone inhibitor of cysteine peptidases
BILN-2061
biotin-Phe-Ala-fluoromethane
biotin-Phe-Pro-Arg-chloromethylketone
BIRC-1 protein
BIRC-2 protein
BIRC-3 protein
BIRC-7 protein
BIRC-8 protein
Bl-Spn1 (
Branchiostoma lanceolatum
)
BmCI chymotrypsin inhibitor (
Rhipicephalus microplus
)
BMS-186282 (thrombin inhibitor)
BMS-189090 (thrombin inhibitor)
BMS-189664 (thrombin inhibitor)
BMS-262084 (beta-lactam tryptase inhibitor)
BMS-289948
BMS-299897
BMS-363131 (tryptase inhibitor)
BMS-561392 (TACE inhibitor)
BMS-740808 (factor Xa inhibitor)
BMS189921
BmSPI inhibitor (
Bombyx mori
)
BN 82204 (calpain inhibitor)
Boc-Val-Val-Phe-P(O)(OH)-CH(R)-Phe-Val-Val-NH2
boceprevir
Bombina trypsin inhibitor
boophilin inhibitor unit 1
boophilin inhibitor unit 2
bortezomib
bothrojaracin
Bowman-Birk inhibitor (Poaceae) inhibitor unit 1
Bowman-Birk inhibitor (Poaceae) inhibitor unit 2
Bowman-Birk inhibitor (
Glycine
-type) unit 1
Bowman-Birk inhibitor (
Glycine
-type) unit 2
Bowman-Birk trypsin inhibitor (
Medicago
-type) unit 1
Bowman-Birk trypsin/chymotrypsin inhibitor (
Arachis hypogaea
) unit 1
bradykinin
bromein
bromoacetyl, difluoroketone inhibitor of gamma-secretase
bromoacetyl-D-arginine
bromosuccinimide
BSF 409425 (calpain inhibitor)
Bu-2743E
BU-32 (proteasome inhibitor)
buckwheat peptidase inhibitor I
BUSI-I inhibitor
butabindide
BX528 (M14.009 inhibitor)
Bz-Arg-His-D-Asp-CH2Cl
Bz-Lys-Lys-Arg-H
Bz-Nle-Lys-Arg-Arg-H
Bz-Nle-Lys-Arg-boronic acid
Bz-Phe-P(O)(OH)-CH(R)-Phe-OH
Bz-Phe-P(O)(OH)-CH(R)-Phe-Val-Val-NH2
Bz-Phe-P(O)(OH)-CH(R)-Pro-Val-Val-NH2
BzLLLCOCHO
C1 inhibitor
CA074
CA074-Me
CAA0225 (cathepsin L inhibitor)
Calbiochem MMP9/13
calpain inhibitor IV
calpastatin inhibitor unit 1
calpastatin inhibitor unit 2
calpastatin inhibitor unit 3
calpastatin inhibitor unit 4
calpeptin
camostat mesilate
candoxatril
caneCPI-4 cystatin (
Saccharum officinalis
)
captopril
carfilzomib
carmegliptin (DPP4 inhibitor)
carp fetuin (
Cyprinus carpio
)
carrapatin
cathepsin B
cathepsin D inhibitor (Solanaceae)
cathepsin G/chymotrypsin inhibitor (
Apis mellifera
)
cathepsin H propeptide
cathepsin K propeptide
cathepsin L
cathepsin L propeptide
cathepsin S propeptide
cathepsin V propeptide
Cbz-Phe(PO(2)-CH(2))-Ala-Arg-Tyr
CCT (neprilysin inhibitor)
CE-0266 (neutrophil elastase inhibitor)
CE-1037 (neutrophil elastase inhibitor)
centerin
CEP1612
cereal subtilisin-chymotrypsin inhibitor-1
cereal subtilisin-chymotrypsin inhibitor-2
CGH728 (thrombin inhibitor)
CGP 53820 (retropepsin inhibitor)
CGS 24592 (NEP inhibitor)
CGS 26303 (neprilysin/ECE inhibitor)
CGS 30084 (ECE inhibitor)
CGS 34043 (neprilysin/ECE inhibitor)
CGS 35066
CGS 35601
CGS27023A
chagasin
chelonianin inhibitor unit 1
chelonianin inhibitor unit 2
CHF5074 (gamma-secretase modulator)
chimadanin (
Haemaphysalis longicornis
)
chlorambucil
chlorodysinosin A
chloroquine
Chondroitin Sulphate
chymostatin
chymotrypsin inhibitor (
Schizolobium parahyba
)
chymotrypsin inhibitor 2
chymotrypsin inhibitor ECI (
Erythrina variegata
)
chymotrypsin inhibitor I (potato)
chymotrypsin inhibitor SCI-I (
Bombyx mori
)
chymotrypsin/elastase inhibitor (
Ascaris
-type)
cilastatin
cilazapril
cinnamoyl-Lys-Lys-Arg-H
circinamide
CKD-732 (MAP inhibitor)
clasto-lactacystin beta-lactone
ClCH2CO-DL-(N-OH)Leu-Ala-Gly-NH2
ClCH2CO-DL-(N-OH)Leu-OCH3
CLIK-148
CLIK-164
CLIK-195
CLIK-60
CLIK148
clitocybin D (neutrophil elastase inhibitor)
clitocypin
CLT (neprilysin inhibitor)
CmPI-II (
Cenchritis muricatus
)
CMT-3 (MMP-inhibitor)
cnispin
coagulation inhibitor (
Anisakis simplex
)
colligin 1
colligin 2
colostrum trypsin inhibitor (
Bos taurus
)
Compound 1
Compound 10
Compound 10.
Compound 11
Compound 11.
Compound 12
Compound 12.
compound 12a (N-(3-(4-chlorophenyl)-1H-pyrazol-5-yl)-2-mercaptoacetamide)
compound 12b (N-(3-(2-chlorophenyl)-1H-pyrazol-5-yl)-2-mercaptoacetamide)
compound 12c (N-(3-(3-(trifluoromethyl)phenyl)-1H-pyrazol-5-yl)-2-mercaptoacetamide)
compound 12d (N-(3-(4-(trifluoromethyl)phenyl)-1H-pyrazol-5-yl)-2- mercaptoacetamide)
compound 12e (N-(3-(phenyl)-1H-pyrazol-5-yl)- 2-mercaptoacetamide)
compound 12f (N-(3-(2-(trifluoromethyl)phenyl)-1H-pyrazol-5-yl)-2- mercaptoacetamide)
compound 12g (N-(3-(3-chlorophenyl)-1H-pyrazol-5-yl)-2-mercaptoacetamide)
compound 12h (N-(3-(4-fluorophenyl)-1H-pyrazol-5-yl)-2-mercaptoace tamide)
compound 12i (N-(3-(4-bromophenyl)-1H-pyrazol-5-yl)-2- mercaptoacetamide)
compound 12j (N-(3-p-tolyl-1H-pyrazol-5-yl)-2-mercaptoacetamide)
compound 12k (N-(3-(4-methoxyphenyl)-1H-pyrazol-5-yl)-2- mercaptoacetamide)
compound 12l (N-(3-(4-nitrophenyl)-1H-pyrazol-5-yl)-2- mercaptoacetamide)
Compound 13
Compound 14
Compound 15
Compound 16
Compound 17
Compound 18
Compound 19
Compound 2
compound 2 (2,4-dichlorocinnamic hydroxamic acid)
compound 20
Compound 21
Compound 22
compound 22 (GT-1017)
Compound 23
compound 24
Compound 25
Compound 26
Compound 27
Compound 28
Compound 29
compound 3
Compound 3.
Compound 30
Compound 31
Compound 32
Compound 33
Compound 34
Compound 35
Compound 36
Compound 38
compound 3a
compound 3b
compound 3c
compound 3d
compound 3e
compound 3f
compound 3g
compound 3k
compound 3m
compound 3o
compound 3q
compound 3s
Compound 4
Compound 4. (GW4459.)
Compound 41
Compound 45
Compound 46
Compound 4e
Compound 5
compound 5 (N-(3-(4-chlorophenyl)-1H-pyrazol-5-yl)-3-mercaptopropanamide)
Compound 6
Compound 6.
Compound 7
Compound 7.
Compound 8
Compound 8.
Compound 9
Compound 9.
compound A (rhodanine dimer)
compound B (rhodanine dimer)
compound C (ketoheterocycle)
compound D (benzoxazinone)
compound E (CF3 peptide)
compound E (gamma-secretase inhibitor)
compound F (imidazole)
compound I (CF3 peptide)
compound inhibitor: I12.001, I12.008
compound inhibitor: I12.007, I12.011, I12.012, I12.013
compound JMF1528
compound JMF1807
compound JMF1810
compound JMF1813
compound JMF1857
compound JMF1859
compound JMF1860
compound JMF1897
compound JMF1900
compound JMF1904
compound yzm16
compound yzm18
compound yzm19
compound yzm38
congopain propeptide
contrapsin
cospin (
Coprinopsis cinerea
)
CP-108,420 (renin inhibitor)
CP-271485 (MMP-12 inhibitor)
CP-544439 (MMP-13 inhibitor)
CP-69,799 (endothiapepsin inhibitor)
CP-72,647 (renin inhibitor)
CP-80794 (renin inhibitor)
CP113972
Cph-Cha-Dap-Glu-Bph-Leu
Cph-Cha-Dbu-Glu-Phe-Cha
Cpp-Ala-Ala
Cpp-Ala-Ala-Phe-pAb
Cpp-Ala-Ala-Tyr-pAb
Cpp-Ala-Pro-Phe-pAb
Cpp-Ala-Pro-Tyr-pAb
Cpp-Leu-Trp (thermolysin inhibitor)
CRA-013783
CRA-2059 (tryptase inhibitor)
CRA-9249 (tryptase inhibitor)
crammer peptidase inhibitor
CrmA viral serpin
CrSPI-1 unit 2 (
Carcinoscorpius rotundicauda
)
crucifer cysteine peptidase inhibitor
cruzipain inhibitor (
Bauhinia bauhinioides
)
cruzipain propeptide
cryptopain-1 (
Cryptosporidium parvum
)
CT1746
CTS-21166 (BACE1 inhibitor)
CU-2010 (plasmin inhibitor)
CVS-3983 (matriptase inhibitor)
cvSI-1 (
Crassostrea virginica
)
cvSI-2 (
Crassostrea virginica
)
cyanopeptolin 954
cyanopeptolin 963 A
cyanostatin A
cyanostatin B
cyclic-imide compound 4l
cyclic-imide compound 6
cyclotheonamide E4 (tryptase inhibitor)
cystatin 4 (
Triticum aestivum
)
cystatin A
cystatin B
cystatin Bm-CPI-2 (
Brugia malayi
)
cystatin C
cystatin D
cystatin E/M
cystatin F
cystatin Hv-CPI1 (
Hordeum vulgare
)
cystatin Hv-CPI10 (
Hordeum vulgare
)
cystatin Hv-CPI11 (
Hordeum vulgare
)
cystatin Hv-CPI13 (
Hordeum vulgare
)
cystatin Hv-CPI2 (
Hordeum vulgare
)
cystatin Hv-CPI3 (
Hordeum vulgare
)
cystatin Hv-CPI5 (
Hordeum vulgare
)
cystatin Hv-CPI6 (
Hordeum vulgare
)
cystatin Hv-CPI8 (
Hordeum vulgare
)
cystatin Hv-CPI9 (
Hordeum vulgare
)
cystatin S
cystatin SA
cystatin SN
cystatin-related epididymal spermatogenic protein
cysteic-leucyl-argininal (calpain inhibitor)
cytin A chain (
Theromyzon tessulatum
)
cytin B chain (
Theromyzon tessulatum
)
cytotoxic T-lymphocyte antigen-2 alpha
cytotoxic T-lymphocyte antigen-2 beta
D-3-[(1-aminoethyl) phosphinyl]-D-2-methylpropionic acid I
D-penicillamine
D-Phe(pNH2)-L-Phe
D-Val-Gly-Arg-CH(2)Cl
dabigatran
DANLME
danoprevir
daphnodorin
DAPT
darunavir
DCI
Dec-Arg-Val-Lys-Arg-CMK
deca-D-Arg-NH2
Decanoyl-LTPTAKAPS-OH
Decanoyl-LTPTAKAPSK-OH
Decanoyl-LTPTAKAPSKI-OH
Decanoyl-LTPTAKAPSKID-OH
Decanoyl-LTPTAKAPSKIDD-OH
Decanoyl-PTAKAPSKIDD-OH
Decanoyl-PTANA-aldehyde
Decanoyl-TAKAPSKIDD-OH
Decanoyl-TPTAKAPSKIDD-OH
decanyol-Arg-Val-Lys-Arg-chloromethylketone
delanzomib
delaprilat
DEPC (diethylpyrocarbonate)
DFK167 (gamma-secretase inhibitor)
DFP
DG-051 (leukotriene A4 hydrolase inhibitor)
DG35-VIII (retropepsin inhibitor)
DIAP1 (
Drosophila melanogaster
)
DIAP2 (
Drosophila melanogaster
)
diazoacetylglycine ethyl ester
diazonium Phe(pNH2)-Phe
diazonium Phe(pNH2)-Phe(pNH2)
diazophenylalanine methylketone Phe (pNH2)CH3
dibenzazepine
diethyldithiocarbamate
diethylpyrocarbonate
dihydroeponemycin
dipeptide 7 (D-Ala-D-Gly(SFp-CHF2)-OH)
dipetalogastin
dipetalogastin inhibitor unit 1
dipetalogastin inhibitor unit 2
dipetalogastin inhibitor unit 3
dipicolinic acid
diprotin
diprotin A
diprotin B
dithiopyridine
dithiothreitol
DL-1-diazo-3-tosylamido-2-heptanone
DL-2-mercaptomethyl-3-guanidinoethylthiopropanoic acid
dl-3-mercapto-2-benzylpropanoylglycine (neprilysin inhibitor)
DMP323 (retropepsin inhibitor)
DMP450 (retropepsin inhibitor)
DnsF (dansyl fluoride)
dodeca-D-Arg-NH2
doxycycline
DPC 333 (ADAM17 inhibitor)
DPC-AB9144-00
DPC423
DTT
DTT (Dithiothreitol.)
DX-9065a
DX600 (ACE2 inhibitor)
Dynorphin A (1-13)
E64
E64d
EACA
ebelactone A
EC27
EC33 (aminopeptidase A inhibitor)
ECAM protein (
Escherichia coli
)
ecotin
EDTA
EF6265 (carboxypeptidase U inhibitor)
Egf1.0 peptidase inhibitor
eglin c
EGTA
EI-1941-1
EI-1941-2 (caspase-1 inhibitor)
elafin
elasnin
elastase inhibitor (
Anemonia sulcata
)
elastase inhibitor (
Triatoma infestans
)
elastase inhibitor MCEI (
Momordica charantia
)
elastatinal
EMD 495235 (factor X inhibitor)
EMD 58265 (renin inhibitor)
enalapril
enapilrilat
endopin 1 (
Bos taurus
)
endopin 2 (
Bos taurus
)
endopin 2C
EP-475 (N-[[L-trans-3-(ethoxycarbonyl)oxiran-2-yl]carbonyl]- L-leucyl-3-methylbutanamide)
Ep475
EPI1 protein inhibitor (
Phytophthora
sp.)
EPI1 protein inhibitor domain 1 (
Phytophthora infestans
)
EPI10 (
Phythophthora infestans
) inhibitor domain 2
EPI10 (
Phythophthora
sp.) inhibitor domain 1
EPIC1 (
Phytophthora infestans
)
EPIC2B (
Phytophthora infestans
)
EPNP
epostatin (DPP II inhibitor)
epoxomicin
eppin-3, inhibitor unit 2
equistatin
equistatin (
Actinia
) inhibitor unit 1
equistatin (
Actinia
) inhibitor unit 2
esophagus cancer-related gene-2
etacrynic acid
etacrynic acid t-butylamide inhibitor (SARS coronavirus main peptidase inhibitor)
eurystatin (POP inhibitor)
F1L protein (vaccinia virus)
factor Xa inhibitor BuXI (
Bauhinia
sp.)
falstatin
FE 999011 (DPP VI inhibitor)
FE999024 (tissue kallikrein inhibitor)
FE999026 (plasma kallikrein inhibitor)
five-domain Kazal-type serine proteinase inhibitor (
Penaeus monodon
) inhibitor unit 2
five-domain Kazal-type serine proteinase inhibitor (
Penaeus monodon
) inhibitor unit 3
five-domain Kazal-type serine proteinase inhibitor (
Penaeus monodon
) inhibitor unit 4
five-domain Kazal-type serine proteinase inhibitor (
Penaeus monodon
) inhibitor unit 5
five-domain Kazal-type serine proteinase inhibitor SPIPm2 (
Penaeus monodon
)
FK-706 (neutrophil elastase inhibitor)
flovagatran (thrombin inhibitor)
fluorosalinosporamide
fluostatin A (DPP III inhibitor)
fluostatin B (DPP III inhibitor)
FM 19 (thrombin inhibitor)
FN-439
fondaparinux
fosinopril
FR136706 (elastase inhibitor)
FR217840 (MMP inhibitor)
FR255031 (MMP inhibitor)
FR901451 (elastase inhibitor)
FR901533 (ECE inhibitor)
fraction IX inhibitor (
Bungarus fasciatus
)
FtTI (
Fagopyrum tataricum
)
fumagillin
furin inhibitor I
furoyl saccharin
FY01 (DPP I inhibitor)
G17905 (factor VIIa inhibitor)
gabexate mesilate
galardin
gamma-pyrone-3-acetic acid (L-741,494) (caspase-1 inhibitor)
gemopatrilat
GEMSA
ghilanten
ghilanten inhibitor unit 1
GI254023X
GL-189 (memapsin-2 inhibitor)
gliotoxin
globomycin
Glp-Asn-Pro-Tyr-Trp-Trp-NHMec (PGP II inhibitor)
Glu-Gly-Arg-CH(2)Cl
Glu-Phe-Arg-CH(2)Cl
Glu-thiol
glutamyl peptidase II inhibitor (bitter gourd)
glutamyl phosphonate (R enantiomer)
Gly-Arg-Gly-Tyr-Ala-Leu-Ala-Ala
Gly-Gly-Tyr(Bzl)-Arg
Gly-Lys-Arg
Gly-Phe-diazomethane (DPP I inhibitor)
Gly-Phe-Gly-semicarbazone
Gly-Pro-Phe-(PO(2)CH(2))-Gly-Pro-Nle
Gly-Pro-Phe-(PO(2)CH(2))-Gly-Pro-Nle (PPI-2)
GPI 5693 (GCP II inhibitor)
grassystatin A
grassystatin B
greglin
GRL-02031 (retropepsin inhibitor)
GRL-8234
GRL-98065 (retropepsin inhibitor)
GRL0617
GS-8374 (retropepsin inhibitor)
guamerin (
Hirudo nipponia
)
GW-311616 (neutrophil elastase inhibitor)
GW0385
GW3333
GW475151
GW640385 (retropepsin inhibitor)
GW796406
GW9471
H-142 (aspartic peptidase inhibitor)
H-boroPheC6H12
H-Glu-(NHO-Bz)-Pyr
H.77 (renin inhibitor)
haemadin
HBY-793 (retropepsin inhibitor)
HcPI (
Hermodice carunculata)
hemalin (
Haemaphysalis longicornis
)
Heparan Sulphate
Heparin
heparin cofactor II
hepatocyte growth factor activator inhibitor 1 inhibitor unit 1
hepatocyte growth factor activator inhibitor 1 inhibitor unit 2
hepatocyte growth factor activator inhibitor 2 inhibitor unit 1
hepatocyte growth factor activator inhibitor 2 inhibitor unit 2
hepatocyte growth factor activator inhibitor type 1
hepatocyte growth factor activator inhibitor type 2
hepta-D-Arg-NH2
hexa-D-Arg-NH2
hirudin
hirustasin
histargin
histidine-rich glycoprotein inhibitor unit 1
HiTI serine peptidase inhibitor (
Haematobia irritans
)
HNSA (aminopeptidase N inhibitor)
homocysteine
HONHCO-CH2-CH(CH2-C6H5)CO-Ile-Ala
HONHCOCH(CH2C6H5)CO-Ala-Gly-NH2
hookworm coagulation inhibitor
Hph-Cha-Dap-Har-Phe-Leu
Hph-Cha-Dbu-Arg-Hph-Cha
Hph-Nva-Dap-Har-Nal-Nva
hPheP[CH(2)]Phe
HPI
HSAc-Phe-Leu
HSCH2CH-(CH2C6H5)CO-Ala-Gly-NH2
HWTX-XI trypsin inhibitor (
Ornithoctonus
sp.)
ICI 186,756 (leukocyte elastase inhibitor)
ICI-200,880 (neutrophil elastase inhibitor)
IDR-803 (MAP inhibitor)
IDR-804 (MAP inhibitor)
IDR-805 (MAP inhibitor)
ILTI trypsin inhibitor (
Inga laurina
)
INCB003619 (ADAM peptidase inhibitor)
indinavir
inducible metallopeptidase inhibitor (
Galleria mellonella
)
inducible serine protease inhibitor 1 (
Galleria mellonella
)
infestin (
Triatoma infestans
)
infestin 1R
infestin 4
inhibitor 49
inhibitor AeTI (
Archidendron ellipticum
)
inhibitor of trypsin and Hageman factor (
Cucurbita maxima
)
inhibitor TgTI (
Toxoplasma gondii
)
intracellular coagulation inhibitor 1 (
Tachypleus
)
intracellular coagulation inhibitor 2 (
Tachypleus
)
intracellular coagulation inhibitor 3 (
Tachypleus
)
iodoacetamide
iodoacetate
IP96
IRS-2 (
Ixodes
sp.)
IseA protein (
Bacillus subtilis
)
ISP2 (
Leishmania
sp.)
ixolaris (
Ixodes scapularis
)
IXP1
JA-2
JCP104
JG-365 (retropepsin inhibitor)
JMV 390-1
JMV1195 (memapsin-2 inhibitor)
JMV2764 (memapsin-2 inhibitor)
JNJ 10329670 (cathepsin S inhibitor)
JNJ 27265732 (leukotriene A4 hydrolase inhibitor)
JNJ-26993135 (leukotriene A4 hydrolase inhibitor)
JTP-4819
JTV-803 (factor Xa inhibitor)
K11002 (cruzipain/rhodesain inhibitor)
K11017 (falcipain-3 inhibitor)
K11777
K2Pt(C2O4)2
K579
KALI-10 (plasma kallikrein inhibitory Kunitz domain.)
KALI-13 (plasma kallikrein inhibitory Kunitz domain.)
KALI-30 (plasma kallikrein inhibitory Kunitz domain.)
KALI-38 (plasma kallikrein inhibitory Kunitz domain.)
KALI-42 (plasma kallikrein inhibitory Kunitz domain.)
KALI-46 (plasma kallikrein inhibitory Kunitz domain.)
KALI-48 (plasma kallikrein inhibitory Kunitz domain.)
KALI-8 (plasma kallikrein inhibitory Kunitz domain.)
KALI-D (plasma kallikrein inhibitory Kunitz domain.)
KALI-DV (plasma kallikrein inhibitory Kunitz domain.)
KALI-DY (plasma kallikrein inhibitory Kunitz domain.)
KALI-E (plasma kallikrein inhibitory Kunitz domain.)
KALI-EV (plasma kallikrein inhibitory Kunitz domain.)
KALI-EY (plasma kallikrein inhibitory Kunitz domain.)
KALI-P (plasma kallikrein inhibitory Kunitz domain.)
KALI-PV (plasma kallikrein inhibitory Kunitz domain.)
KALI-PY (plasma kallikrein inhibitory Kunitz domain.)
kallistatin
Kazal inhibitor CCTI (
Caiman crocodylus
)
KB-R7785
kelatorphan
kempopeptin A
kempopeptin B
keto-ACE
kexstatin I
kininogen
kininogen inhibitor unit 2
kininogen inhibitor unit 3
KMI-008 (memapsin-2 inhibitor)
KMI-260 (memapsin-2 inhibitor)
KMI-358 (memapsin-2 inhibitor)
KMI-360 (memapsin-2 inhibitor)
KMI-370 (memapsin-2 inhibitor)
KMI-420 (memapsin-2 inhibitor)
KMI-429 (memapsin-2 inhibitor)
KMI-570 (memapsin-2 inhibitor)
KMI-684 (memapsin-2 inhibitor)
KNI-10006 (plasmepsin inhibitor)
KNI-10127 (HTLV-1 retropepsin inhibitor)
KNI-10161 (HTLV-1 retropepsin inhibitor)
KNI-10166 (HTLV-1 retropepsin inhibitor)
KNI-10516 (HTLV-1 retropepsin inhibitor)
KNI-577 (retropepsin inhibitor)
KPC-4 peptidase propeptide
KRI-1314 (renin inhibitor)
Kunitz cysteine peptidase inhibitor 1 (plant)
Kunitz serine peptidase inhibitor (
Delonix regia
)
Kunitz subtilisin inhibitor (Fabaceae-type)
kynostatin-272
KYT-1 (gingipain inhibitor)
KYT-36 (gingipain inhibitor)
L-1-diazo-3-tosylamido-4-phenyl-2-butanone
L-1-tosylamido-2-phenylethylchloromethylketone
L-363,564 (renin inhibitor)
L-375,378
L-658,758
L-659,286 (leukocyte elastase inhibitor)
L-680,833 (leukocyte elastase inhibitor)
L-681,176
L-682,679 (retropepsin inhibitor)
L-683,845 (leukocyte elastase inhibitor)
L-685,434 (retropepsin inhibitor)
L-685,458
L-694,458 (neutrophil elastase inhibitor)
L-873724
L-arginine compound 5q
L-arginine compound 5s
L-lysine compound C20
L-lysine compound C7
lactacystin
lactoyl-Glu-Sta-Ala-Sta-NH2
lactoyl-Lys-Sta-Ala-Sta-NH2
lapstatin
latex serine peptidase inhibitor (
Papaya carica
)
latexin
LCZ696 (neprilysin inhibitor)
LDN-57444 (UCHL-1 inhibitor)
leech metallocarboxypeptidase inhibitor
Lentinus peptidase inhibitor
Leu-CH2Cl
Leu-PheCH2C1
leucinal
leucinethiol
leuhistin
leupeptin
linagliptin
lisinopril
lisinopril-Trp
LK-733 (thrombin inhibitor)
lopinavir
LP-130
LP-149 (FIV retropepsin inhibitor)
LSEAL peptide (calpain inhibitor)
lupin Bowman-Birk trypsin inhibitor
LY2434074 (BACE1 inhibitor)
LY312340 (PSA inhibitor)
LY411575
lyngbyastatin 4
lyngbyastatins 10
lyngbyastatins 8
lyngbyastatins 9
LYP (aminopeptidase N inhibitor)
Lys-Arg
Lys-Lys-Arg
Lys-Thr-Glu-Glu-Ile-Ser-Val-Val-Sta-Val-Ala-Glu-Phe
Lys-Thr-Lys-Val-Leu-Val-Val-Gln-Pro-Lys
lysinethiol
M826 (caspase-3 inhibitor)
M867 (caspase-3 inhibitor)
macrocyclic squash trypsin inhibitor (
Momordica cochinchinensis
)
macrocypin 1
macrocypin 3
macrocypin 4
madanin 1 (
Haemaphysalis longicornis
)
maize trypsin/factor XIIa inhibitor
mannan-binding protein (MBP-A)
marimastat
marinostatin
matlystatin A
matlystatin B
MCoCI chymotrypsin inhibitor (
Momordica cochinchinensis
)
MD1 (signal peptidase I inhibitor)
MD2 (signal peptidase I inhibitor)
MD3 (signal peptidase I inhibitor)
MDL104903 calpain inhibitor
MDL28170
MDL73347 (aminopeptidase inhibitor)
melagatran
MeOSuc-Ala-Ala-Pro-Val-CH(2)Cl
metallocarboxypeptidase A inhibitor (
Ascaris suum
)
metallopeptidase inhibitor (snake venom)
metallopeptidase inhibitor (
Erwinia
)
methoxysuccinyl-Ala-Ala-Pro-Phe-chloromethyl ketone
methyl 2-(4-
4-[(2-thiiranylpropyl)sulfonyl]phenoxy
phenyl)acetate
methyl methanethiosulfanate (MMTS)
MG-262
MG115
MG132
MHC II invariant chain p41 form
micropeptin 103
micropeptin EI964
micropeptin EI992
microviridin J
MK-0674 (cathepsin K inhibitor)
MK-1256 (cathepsin K inhibitor)
MLN-4760
MLN273 (proteasome inibitor)
MLN519
MLN9708 (proteasome inibitor)
MMI-166
MMP408 (MMP-12 inhibitor)
MMPSI (caspase 3/7- inhibitor)
MNRC-5
moexipril (ACE inhibitor)
MR-889 (neutrophil elastase inhibitor)
MRK-560 (gamma-secretase inhibitor)
MRT12113
MUGB
murinoglobulin 1
mustard trypsin inhibitor-2
MUTMAC
Mu–Phe–Hph
Mu–Phe–Lys
MVT-101 (retropepsin inhibitor)
MW167
myeloid and erythroid nuclear termination stage-specific protein (
Gallus gallus
)
myxoma virus serpin serp-1
myxoma virus serpin serp2
N, N, N’-tetrakis(2-pyridylmethyl) ethylenediamine (TPEN)
N-(2-chloroethyl)-N-methylphenylalanine
N-(hydroxyacetyl)-L-Phe
N-alkoxy-arylsulfonamide (retropepsin inhibitor)
N-bromoacetyl-D-Leu-Gly
N-bromoacetyl-N-methyl-L-Phe
N-chloroacetyl-N-hydroxy-alpha-Phe-O-methylamide
N-chloroacetyl-N-hydroxy-beta-L-Phe-N-methylamide
N-cinnamoyl-l-aspartic acid compound 8c
N-diazoacetyl-N’-(2,4-dinitrophenyl)-ethylenediamine
N-iodoacetyl-valine-phenylalanine-amide (IVF)
N-methoxyphenylalanine glycylnitrile
N-methylmaleimide
N-phenylmaleimide
N-[(L-trans-3-carbamoyloxiran-2-yl)carbonyl]-L-leucyl- 3-methylbutanamide
N-[(R)-2-benzyl-5-cyano-4-oxopentanoyl]-L-Phe
N-[N-(cyanoacetyl)-L-Phe]-L-Phe
N-[[L-trans-(hydroxylamino)oxiran-2-yl]carbonyl]-Lleucyl- 3-methylbutanamide
N-[[L-trans-(methylcarbonyl)oxiran-2-yl]carbonyl]-Lleucyl- 3-methylbutanamide
N-[[L-trans-3-(ethoxycarbonyl)oxiran-2-yl]carbonyl]- L-leucyl-3-methylbutanamide
N-[[L-trans-3-(hydroxymethyl)oxiran-2-yl]carbonyl]- L-leucyl-3-methylbutanamide
nafamostat mesilate
Nal-Cha-Dap-Glu-Nal-Nva
Nal-Cha-Lys-Aph-Btr-Nle
Nal-Cha-Met-Glu-Phg-Cha
Nal-Nle-Dbu-Glu-Hph-Nva
Nal-Val-Met-Har-Tyr-Nva
NAPAP
napsagatran
nazumamide A (thrombin-inhibitor)
NC2213 (MetAP2 inhibitor)
NcPI-S protein (
Neospora caninum
)
Nedd8 aldehyde
Nedd8 vinyl sulfone
nelfinavir
NEM
neuroserpin
Nip-Leu-Leu-LeuVS-Me
NK3201
nona-D-Arg-NH2
nostopeptin BN920
NPGB
NSC 632839 (isopeptidase inhibitor)
NVP-AHW700-NX (gamma-secretase inhibitor)
NVP-DPP728
O-(hydroxyacetyl)-L-beta-phenyllactic acid
O-[(1S)-aminoethylhydroxyphosphinyl]-D-lactic acid
O. microlepidotus inhibitor (OMI)
octa-D-Arg-NH2
odanacatib
OH-TCI trypsin/chymotrypsin inhibitor (
Ophiophagus hannah
)
OM00-3
OM99-1
OM99-2
omapatrilat
onchocystatin
ONO-4817
ONO-6818
Ono-EI-600 (elastase inhibitor)
ONO3307
opiorphin
oprin
ornithodorin inhibitor unit 1
oryctin (
Oryctes rhinoceros
)
oryzacystatin II
oscillapeptin
oscillarin (thrombin inhibitor)
OST-4077 (cathepsin K inhibitor)
Osteocalcin
otamixaban (factor Xa inhibitor)
ovalicin
ovocalyxin-32
ovocystatin
ovoinhibitor inhibitor unit 1
ovoinhibitor inhibitor unit 2
ovoinhibitor inhibitor unit 3
ovoinhibitor inhibitor unit 4
ovoinhibitor inhibitor unit 5
ovoinhibitor inhibitor unit 6
ovoinhibitor inhibitor unit 7
ovomacroglobulin
ovomucoid
ovomucoid inhibitor unit 1
ovomucoid inhibitor unit 2
ovomucoid inhibitor unit 3
P-1946 (retropepsin inhibitor)
p-bromophenacyl bromide
p-chloromercuriphenylsulfonic acid
p-hydroxymercuribenzoate
P-Leu-Phe
p-nitrophenyl N2-acetyl-N1-benzylcarbazate (chymotrypsin titrant)
p-S8 peptide
p35 homologue (Amsacta moorei entomopoxvirus)
P9941 (retropepsin inhibitor)
paecilopeptin
papain
papain inhibitor (
Prosopis
-type)
papaya cystatin
PAPI-I inhibitor unit 1
PAQ-22 (cytosol alanyl aminopeptidase inhibitor)
paragonial peptide D (
Drosophila funebris
)
PB8 (SYLKKLCGTVLGGPK)
PC18 (aminopeptidase N inhibitor)
PCMB
Pcp24 (Ala-Tyr-His-Asn-Gly-Ala-Ala)
Pcp25 (EFRATYHNGAEYYAAAL)
Pcp26 (DMSPEEFRATYHNGAEYYAAAL)
Pcp27 (NPYATFGVTRFSDMSPEEFRATYHNGAEYYAAAL)
Pcp33 (EEFRSRYHNGAAAHFAAAEE)
PD 163594 (caspase-1 inhibitor)
PD151746
pentenocin B
penthalaris (
Ixodes scapularis
)
pepstatin
peptidase A inhibitor 1 (
Pleurotus ostreatus
)
peptidase B inhibitor (fungus)
peptidase inhibitor (
Tachypleus
)
peptidase inhibitor 3 (rodent)
peptidase inhibitor 5 (
Anemonia sulcata
)
peptidase inhibitor LGPI (Orthoptera) inhibitor unit 2
peptidase inhibitor LMPI (Orthoptera) inhibitor unit 1
PF-00356231 (MMP-12 inhibitor)
PF-734200 (DPP4 inhibitor)
PF3491390 (pancaspase inhibitor)
Phe-LeuCH2C1
Phe-Tyr-Val-Phe-Sta-Ala-Met-Thr-NH2
phebestin
PheCh2Br
PheCH2C1
phenacein
phenacetyl-Arg-Lys-Arg-H
phenacetyl-Cit-Lys-Arg-H
phenacetyl-hArg-Lys-Arg-H
phenacetyl-Lys-Arg-Arg-H
phenacetyl-Lys-hArg-Arg-H
phenacetyl-Lys-Lys-Arg-H
phenacetyl-Lys-Orn-Arg-H
phenacetyl-Orn-Lys-Arg-H
phenoxyacetyl-Lys-Lys-Arg-H
phenylacetyl-Arg-Val-Arg-4-amidinobenzylamide (furin inhibitor)
Phenylalanyl-ureido-citrullinyl-valinyl-cycloarginal
phenylalanylglycinal
phenylpropanoyl-Lys-Lys-Arg-H
phepropeptin A
phepropeptin B
phepropeptin C
phepropeptin D
phevalin
phosphatidylethanolamine-binding protein
phosphodiepryl 08
phosphodiepryl 21
phosphodiepryl 33
phosphoramidon
Phosphoryl-Leu-Trp
phthalhydrazide 24
PHX1149 (DPP IV inhibitor)
phytocystatin
phytocystatin (
Actinidia
sp.)
pinA Lon peptidase inhibitor (phage T4)
pinostrobin
piperastatin A
PIQ-22 (alanyl aminopeptidase inhibitor)
PKSI-527
PL-100 (retropepsin inhibitor)
PL250 (M01.005 inhibitor)
PL302 (aminopeptidae A inhibitor)
plasma kallikrein inhibitor (
Oxyuranus
sp.)
plasmin inhibitor
plasminogen activator inhibitor 2
plasminogen activator inhibitor-1
plasminostreptin
PLG-NHOH (Pro-Leu-Gly-NHOH)
PMPA
PMSF
Pol 647 (adamalysin inhibitor)
Pol 656 (adamalysin inhibitor)
polyhedral metallacarborane (retropepsin inhibitor)
Portland variant
poststatin
potato Kunitz-type trypsin inhibitor
potato metallocarboxypeptidase inhibitor
potato multicystatin inhibitor unit 1
potato multicystatin inhibitor unit 2
potato multicystatin inhibitor unit 3
potato multicystatin inhibitor unit 4
potato multicystatin inhibitor unit 5
potato multicystatin inhibitor unit 6
potato multicystatin inhibitor unit 7
potato multicystatin inhibitor unit 8
potato peptidase inhibitor I
potato peptidase inhibitor II inhibitor unit 1
PPACK
PPI-2458 (MetAP-2 inhibitor)
PR-047
PR39 peptide (proteasome inhibitor)
pralnacasan
pregnancy-zone protein
Prinomastat
pro-eosinophil major basic protein
Pro-Ile
Pro-Leu-Gly-NHOH
Pro-Phe-(PO(2)CH(2))-Gly-Pro
Pro-Phe-(PO(2)CH(2))-Leu-Pro-NH2
probestin
prodipine (DPP4 inhibitor)
prohisin
propioxatin A
propioxatin B
proSAAS
protease nexin-1
protease nexin-2
protein C inhibitor
protein Z-dependent peptidase inhibitor
proteinase inhibitor A (
Sagittaria sagittifolia
)
proteinase inhibitor B (
Sagittaria sagittifolia
)
PRT2005
PRT2253
PT-100
PTL11028 (Der p 1 inhibitor)
puromycin
PwSERPIN (
Paragonimus westermani
)
pyrimidinetrione compound 12
pyrimidinetrione compound 14
pyrimidinetrione compound 15
pyrimidinetrione compound 18
pyrimidinetrione compound 26
pyrimidinetrione compound 28
pyrimidinetrione compound 29
pyrimidinetrione compound 3
pyrimidinetrione compound 30
pyrimidinetrione compound 31
pyrimidinetrione compound 32
pyrimidinetrione compound 33
pyrimidinetrione compound 34
pyrimidinetrione compound 35
pyrimidinetrione compound 36
pyrimidinetrione compound 37
pyrimidinetrione compound 8
pyrimidinetrione compound 9
pyrizinostatin (pyroglutamyl peptidase inhibitor)
quisqualic acid
R-3032 (cathepsin B inhibitor)
R-94138 (matrixin inhibitor)
ragi seed trypsin/alpha-amylase inhibitor
ramipril
rape trypsin inhibitor
razaxaban (factor Xa inhibitor)
RB 101(S)
RB 105
RB25 (neprilysin inhibitor)
RB3007 (neprilysin/aminopeptidase N inhibitor)
RB3014 (alanyl aminopeptidase inhibitor)
RECK protein inhibitor unit 1
recursterol (chymotrypsin inhibitor)
relacatib
rhodniin inhibitor unit 1
rhodniin inhibitor unit 2
rice Bowman-Birk inhibitor inhibitor unit 1
rice Bowman-Birk trypsin inhibitor inhibitor unit 2
ritonavir
rivaroxaban
RK-805 (MetAP2 inhibitor)
Ro 28-2653
Ro 32-7315
RO1 (retropepsin inhibitor)
RO200-1770
RPR120844 (factor Xa inhibitor)
RPR209685 (factor Xa inhibitor)
rupintrivir
RWJ-355871 (cathepsin G/chymase inhibitor)
RWJ-445167 (thrombin and factor Xa inhibitor)
RWJ-56423 (tryptase inhibitor)
RXP03 (MMP inhibitor)
RXP407
RXP407 (M02.001 inhibitor)
RXPA380
RXPA380 (M02.004 inhibitor)
S-2209 (proteasome inhibitor)
S-3304 (MMP inhibitor)
S-nitrosothiol compound (unassigned)
S17092
S18326
SA898 (TOP inhibitor)
saccharopepsin inhibitor
salarin
salinosporamide A
salinosporamide B
saquinavir
sarcocystatin
savignin (
Ornithodoros savignyi
)
saxagliptin
SB 331750
SB-3CT
SB-553484 (cathepsin K inhibitor)
SB203238 (retropepsin inhibitor)
SC-22716 (leukotriene A4 hydrolase inhibitor)
SC-57461A (leukotriene A4 hydrolase inhibitor)
SC68896 (proteasome inhibitor)
SCH 32615 (neprilysin inhibitor)
SCH 34826
SCH 42354
SCH47896 (neprilysin inhibitor)
SCH6
ScNPI inhibitor (
Streptomyces caespitosus
)
scyptolin (pancreatic elastase inhibitor)
SD146 (retropepsin inhibitor)
SDZ 224-015 (caspase-1 inhibitor)
SDZ283-910 (retropepsin inhibitor)
secretogranin V
secretory leukocyte peptidase inhibitor
secretory leukocyte peptidase inhibitor domain 1
secretory leukocyte peptidase inhibitor domain 2
semagacestat
sepimostat mesilate
Ser-Lys-Lys-Arg
serine carboxypeptidase Y inhibitor (
Saccharomyces cerevisiae
)
serine peptidase inhibitor II (
Capsicum
-type)
serpin 4 (
Drosophila melanogaster
)
serpin B1
serpin B12
serpin B13
serpin B6
serpin B8
serpin B9
serpin Emu (
Echinococcus multilocularis
)
serpin Iris (
Ixodes ricinus
)
serpin Necrotic (
Drosophila melanogaster
)
serpin SPI-3 (orthopoxvirus)
serpin SPI-C1 (
Mus musculus
)
serpin SPI2
serpin SPN27A (
Drosophila melanogaster
)
serpin srp-2 (
Caenorhabditis elegans
)
serpin srp-3 (
Caenorhabditis elegans
)
serpin SRP-6 (
Caenorhabditis elegans
)
serpin-4 (
Manduca sexta
)
serpin-5 (
Drosophila melanogaster
)
serpin-6 (
Manduca sexta
)
serpina3n
serpinb3b (
Mus musculus
)
serralysin inhibitor (
Serratia
sp.)
sialorphin
sialostatin L (
Ixodes scapularis
)
SIL-1 inhibitor (
Streptomyces cacaoi
)
SIL-10 inhibitor (
Streptomyces thermotolerans
)
SIL-12 inhibitor (
Streptomyces hygroscopicus
)
SIL-13 inhibitor (
Streptomyces galbus
)
SIL-14 inhibitor (
Streptomyces cyaneus
)
SIL-15 inhibitor (
Streptomyces bikiniensis
)
SIL-2 inhibitor (
Streptomyces
sp.)
SIL-3 inhibitor (
Streptomyces coelicolor
)
SIL-4 inhibitor (
Streptomyces lavendulae
)
SIL-5 inhibitor (
Streptomyces fradiae
)
SIL-7 inhibitor (
Streptomyces ambofaciens
)
SIL-8 inhibitor (
Streptomyces virginiae
)
sitagliptin
sivelestat
Sizzled protein (
Xenopus laevis
)
SJA6017
SKF 107457 (retropepsin inhibitor)
SKF 108738 (retropepsin inhibitor)
skin protein 1 (
Phyllomedusa sauvagii
)
SLV306 (neprilysin/ECE inhibitor)
SM-19712 (ECE inhibitor)
snake venom cystatin (
Bitis
sp.)
SNJ-1715 (calpain inhibitor)
SNJ-1757 (calpain inhibitor)
SNJ-1945
SO2(C6H4)NHCO(C6H4)(CH2)4CH3
soybean Kunitz trypsin inhibitor
SPF-32629 (chymase inhibitor)
SPINK1
SPINK2
SPINK5 g.p. (
Homo sapiens
)
SPINK5 inhibitor unit 15
SPINK5 inhibitor unit 6
SPINK6
SPINK9
spinorphin
spirapril
spiropyrrolidine compound 1
spiropyrrolidine compound 10a
spiropyrrolidine compound 10b
spiropyrrolidine compound 11
spiropyrrolidine compound 12
spiropyrrolidine compound 13
spiropyrrolidine compound 14
spiropyrrolidine compound 15
spiropyrrolidine compound 16
spiropyrrolidine compound 17
spiropyrrolidine compound 18
spiropyrrolidine compound 19
spiropyrrolidine compound 20
spiropyrrolidine compound 21
spiropyrrolidine compound 22
spiropyrrolidine compound 23
spiropyrrolidine compound 24
spiropyrrolidine compound 25
spiropyrrolidine compound 26
spiropyrrolidine compound 4
spleen trypsin inhibitor I (
Bos taurus
)
sporamin
spumigin E
SQ 14,603 (carboxypeptidase A inhibitor)
SQ 24,798 (carboxypeptidase B inhibitor)
SQ 28,603
SQ-28603 (neprilysin inhibitor)
squamous cell carcinoma antigen 1
squamous cell carcinoma antigen 2
SR 26831 (leukocyte elastase inhibitor)
SRPN2 (
Anopheles gambiae
)
SsCEI (
Sulfolobus
sp.)
SSR182289A (thrombin inhibitor)
SSR69071
staphostatin A
staphostatin B
Streptomyces metallopeptidase inhibitor
streptomyces subtilisin inhibitor
streptopain inhibitor (
Streptococcus pyogenes
)
SUAM 1221 (POP inhibitor)
SUB1 peptidase propeptide
substance P
subtilisin inhibitor I (Fabaceae)
subtilisin propeptide
subtilisin-chymotrypsin inhibitor CI-1A (barley)
Suc-Ala-Ala-Pro-Phe-CH(2)Cl
sulfonyl hydroxamate inhibitor of metallopeptidase (unassigned)
SUMO1-vinyl methyl ester
SUMO3-vinyl methyl ester
SUN13834 (chymase inhibitor)
sunflower cyclic trypsin inhibitor
sunflower multicystatin inhibitor unit 1
survivin
SWDPm subtilisin inhibitor (
Penaeus monodon
)
syringolin A
T-kininogen
T-kininogen inhibitor unit 2
T-kininogen inhibitor unit 3
T06126 (4-(4-(5-methyl-3-phenylisoxazol-4-yl)thiazol-2-yl)piperidine-1-carboxamide)
talopeptin
tamarind Kunitz trypsin inhibitor (
Tamarindus indica
)
TAPI
TAPI-2
TBODA (prolyl aminopeptidase inhibitor)
TdPI tryptase inhibitor (
Rhipicephalus appendiculatus
)
TEI-8362 (neutrophil elastase inhibitor)
TEI-E548 (chymase inhibitor)
telaprevir
temocapril
teprotide
tessulin
testican 3
testican-1
tetracycline derivative (unassigned)
tetraethylene pentamine
tetraethylene-pentamine
Tetraethylenepentamine
textilinin-1 (
Pseudonaja textilis
)
TF7I-C (plasma kallikrein inhibitory Kunitz domain.)
therin
thermopin (
Thermobifida fusca
)
theromin (
Theromyzon tessulatum
)
Thiobendazole
thiorphan
thrombin inhibitor (
Glossina morsitans
)
thrombostasin (
Haematobia irritans
)
thymopentin (neprilysin inhibitor)
thysanone (rhinovirus picornain 3C inhibitor)
tick anticoagulant peptide (
Ornithodorus
sp.)
tick carboxypeptidase inhibitor (
Haemaphysalis longicornis
)
tick carboxypeptidase inhibitor (
Rhipicephalus bursa
)
timp-1
timp-2
timp-3
timp-4
timp-DM (
Drosophila melanogaster
)
tipranavir
tissue factor pathway inhibitor-1
tissue factor pathway inhibitor-1 inhibitor unit 1
tissue factor pathway inhibitor-1 inhibitor unit 2
tissue factor pathway inhibitor-2
tissue factor pathway inhibitor-2 inhibitor unit 1
Tk-serpin (
Thermococcus kodakaraensis
)
TL-3
TLCK
TMC-95
TMC240 (retropepsin inhibitor)
TMC435350
TMI-1
TMI-2 (TACE inhibitor)
TmSPN48 (
Tenebrio molitor
)
TNP-470
tobacco peptidase inhibitor II inhibitor unit 1
tomato peptidase inhibitor I
tomato peptidase inhibitor II inhibitor unit 1
Tos-Leu-CH2Cl
toxostatin-1 (
Toxoplasma gondii
)
TP-110 (proteasome inhibitor)
TPCK
trandolaprilat
tranexamic acid
triabin
trypsin inhibitor (
Acacia confusa
)
trypsin inhibitor (
Enterolobium contortisiliquum
)
trypsin inhibitor (
Mirabilis jalapa
)
trypsin inhibitor (
Rana areolata
)
trypsin inhibitor BDTI-II (
Bryonia dioica
)
trypsin inhibitor CMeTI-B (
Cucumis melo
)
trypsin inhibitor CMTI-I (
Cucurbita maxima
)
trypsin inhibitor CMTI-II (
Cucumis melo
)
trypsin inhibitor CMTI-III (
Cucurbita maxima
)
trypsin inhibitor CPTI (
Cucurbita pepo
)
trypsin inhibitor CSTI-IIb (
Cucumis sativus
)
trypsin inhibitor CSTI-IV (
Cucumis sativus
)
trypsin inhibitor CVTI-I (Cucurbitaceae)
trypsin inhibitor EETI-II (
Ecballium elaterium
)
trypsin inhibitor LCTI (
Luffa cylindrica
)
trypsin inhibitor MCTI-1 (
Momordica charantia
)
trypsin inhibitor MCTI-A (
Momordica charantia
)
trypsin inhibitor MCTI-II (
Momordica charantia
)
trypsin inhibitor MCTI-III (
Momordica charantia
)
trypsin inhibitor MRTI-I (
Momordica repens
)
trypsin inhibitor PtTI (
Populus tremuloides
and similar)
trypsin inhibitor STI1 (
Streptomyces coelicolor
)
trypsin inhibitor TGTI-I (
Luffa cylindrica
)
trypsin inhibitor TGTI-II (
Luffa cylindrica
)
trypsin inhibitor TTII (
Trichosanthes kirilowii
)
trypsin/subtilisin inhibitor (
Amaranthus
sp.)
tryptase inhibitor (
Hirudo medicinalis
)
TTP889 (factor IXa inhibitor)
turkinh1 (
Meleagris gallopavo
)
TY-51076 (chymase inhibitor)
TY-51184 (chymase inhibitor)
TY-51469 (chymase inhibitor)
tynorphin
tyropeptin A
tyrostatin
U 71038 (renin inhibitor)
U-81749 (retropepsin inhibitor)
UAMC00039 (DPPII inhibitor)
ubiquitin aldehyde
ubiquitin vinyl sulfone
Ucf-101 (HtrA2 inhibitor)
UIC-PI
UK 156,406
UK-356,202 (urokinase inhibitor)
UK-396082 (carboxypeptidase U inhibitor)
undeca-D-Arg-NH2
upain-1 (uPA inhibitor)
Val-pyrrolidide
vanadate
vaniprevir
variegin (
Amblyomma variegatum
)
vildagliptin
VRT-018858 (caspase-1 inhibitor)
VX-166 (caspase inhibitor)
VX-765 (caspase-1 inhibitor)
WAY-281418 (TACE inhibitor)
WFIKKN peptidase inhibitor inhibitor unit 3
wheat subtilisin/chymotrypsin inhibitor
wheat trypsin/alpha-amylase inhibitor
winged-bean chymotrypsin inhibitor
WRR483 (histolysain inhibitor)
WRR605
WRSI5 trypsin inhibitor
WS75624 A (endothelin converting enzyme inhibitor)
WS75624 B (endothelin converting enzyme inhibitor)
WX-FX4 (factor Xa inhibitor)
WX-UK1 (urokinase inhibitor)
XIAP caspase inhibitor
XM323 (retropepsin inhibitor)
Y-40613 (chymase inhibitor)
Y1 (Arg-Val-Ser-Met-Ile-Lys-Asn-Arg)
YM-60828 (factor Xa inhibitor)
YM-96765 (factor Xa inhibitor)
YO-2 (plasmin inhibitor)
YS-980 (ACE inhibitor)
YU102 (Ac-Gly-Pro-Phe-Leu-epoxyketone)
Z-(L,D)Phe-(PO(2)CH(2))(L,D)Ala-Arg-Met
Z-(L,D)Phe-(PO(2)CH(2))(L,D)Ala-Arg-Phe
Z-(L,D)Phe-(PO(2)CH(2))(L,D)Ala-Arg-Xaa
Z-321 (POP inhibitor)
Z-AEVD-FMK (caspase-10 inhibitor)
Z-Ala-Ala-aza-Asn-epoxycarboxylate ethyl ester
Z-Ala-Ala-Pro-Phe-chloromethyl ketone
z-Ala-Ile-boronic acid
Z-Ala-Pro-Phe-chloromethylketone
z-DEVD-cmk
Z-DEVD-FMK
Z-FA-FMK
Z-Glu-Tyr
Z-Gly-Pro-Phe-Leu-Ala
Z-IETD-FMK
Z-Ile-Glu(OtBu)-Ala-Leu-H
Z-Ile-His-Phe-P(O)(OH)-CH(R)-Phe-Val-Val-NH2
Z-LEHD-FMK (caspase-9 inhibitor)
Z-Leu-Leu-LeuVS
Z-Leu-Leu-Nle-H
Z-Leu-Leu-Phe-H
Z-Leu-Leu-Tyr-FMK
Z-Leu-Tyr-chloromethyl ketone
Z-Lys-Lys-Arg-H
Z-Phe
Z-Phe-(PO(2)CH(2))-Ala-Lys-Ser (PPI-1)
Z-Phe-(PO(2)CH(2))-Ala-Lys-Tyr
Z-Phe-(PO(2)CH(2))-Ala-Lys-Tyr (PPI-0)
Z-Phe-Ala-chloromethyl ketone
Z-Phe-Ala-CHN2
Z-Phe-Ala-diazomethane
Z-Phe-Arg-2,4,6-dimethylbenzoyloxymethyl ketone
Z-Phe-Arg-diazomethane
Z-Phe-D-Leu-Ala-Ala
Z-Phe-Gly-Asn-His-OBz
Z-Phe-Gly-NHO-Bz
Z-Phe-Leu
Z-Phe-Leu-Ala
Z-Phe-Lys-2,4,6-trimethylbenzoyloxymethyl ketone
Z-Phe-Lys-chloromethyl ketone
Z-Phe-P(O)(OH)-CH(R)-Pip-Val-Val-NH2
Z-Phe-P(O)(OH)-CH(R)-Pro-Val-Val-NH2
Z-Phe-Phe-diazomethane
Z-Phe-Tyr(OBut)-CHN(2)
Z-PnLD-al (Z-Pro-norLeu-Asp-aldehyde)
Z-Pro (prolidase inhibitor)
Z-Ser-Ser-Gln-Nle-(boro)-Leu (KLK3 inhibitor)
Z-VAD-FMK
Z-VDVAD-FMK (caspase-2 inhibitor)
Z-YVAD-FMK
Z13752A (ACE/neprilysin inhibitor)
ZD-0892 (neutrophil elastase inhibitor)
ZD-8321 (neutrophil elastase inhibitor)
zincon
Zincov
Zincov (pseudolysin inhibitor)
ZJ-43 (glutamate carboxypeptidase II inhibitor)
ZK-807834
zVAD-fmk
zVAM-fmk
Z–Phe–Arg–CH2F
Ancylostoma caninum
anticoagulant peptide c2
Bauhinia
-type trypsin inhibitor
Bombyx
-type cysteine peptidase inhibitor
Erythrina
-type trypsin/tissue plasminogen activator inhibitor
Leucaena
-type trypsin inhibitor (Fabaceae)
Veronica
trypsin inhibitor
Order results by :
MEROPS Identifier
Recommended name