EMD-53260
Inward-occluded structure of human GABA transporter 3 bound to substrate GABA
EMD-53260
Single-particle3.2 Å
Deposition: 25/03/2025Map released: 04/03/2026
Last modified: 04/03/2026
Sample Organism:
Homo sapiens
Sample: Human GABA transporter 3 bound to substrate GABA
Fitted models: 9qo9
Deposition Authors: Mortensen JS
,
Bavo F,
Jensen MH
,
Pedersen APS
,
Storm JP,
Pape T
,
Frolund B,
Wellendorph P
,
Shahsavar A
Sample: Human GABA transporter 3 bound to substrate GABA
Fitted models: 9qo9
Deposition Authors: Mortensen JS
,
Bavo F,
Jensen MH
,
Pedersen APS
,
Storm JP,
Pape T
,
Frolund B,
Wellendorph P
,
Shahsavar A
Structural basis for selective inhibition of human GABA transporter GAT3.
Mortensen JS
,
Bavo F,
Jensen MH
,
Pedersen APS
,
Storm JP,
Pape T
,
Frolund B,
Wellendorph P
,
Shahsavar A
(2026) Nat Commun , 17 , 1774 - 1774
,
Bavo F,
Jensen MH
,
Pedersen APS
,
Storm JP,
Pape T
,
Frolund B,
Wellendorph P
,
Shahsavar A
(2026) Nat Commun , 17 , 1774 - 1774
Grant Support:
- Lundbeckfonden: R368-2021-522 (Denmark)
- Novo Nordisk Foundation: NNF21OC0067835 (Denmark)
- Novo Nordisk Foundation: NFF20OC0065017 (Denmark)
- Other government: 1026-00335B (Denmark)
