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EMD-16557
Mouse serotonin 5-HT3A receptor in complex with PZ-1939
EMD-16557
Single-particle3.0 Å
Deposition: 26/01/2023Map released: 11/10/2023
Last modified: 09/07/2025
Sample Organism:
Mus musculus
Sample: Mouse serotonin 5-HT3A receptor in complex with PZ-1922
Fitted models: 8cc7
Deposition Authors: Lopez-Sanchez U
,
Nury H
Sample: Mouse serotonin 5-HT3A receptor in complex with PZ-1922
Fitted models: 8cc7
Deposition Authors: Lopez-Sanchez U
,
Nury H
Superiority of the Triple-Acting 5-HT 6 R/5-HT 3 R Antagonist and MAO-B Reversible Inhibitor PZ-1922 over 5-HT 6 R Antagonist Intepirdine in Alleviation of Cognitive Deficits in Rats.
Grychowska K ,
Lopez-Sanchez U ,
Vitalis M ,
Canet G ,
Satala G ,
Olejarz-Maciej A ,
Golebiowska J,
Kurczab R ,
Pietrus W ,
Kubacka M,
Moreau C ,
Walczak M ,
Blicharz-Futera K ,
Bento O ,
Bantreil X ,
Subra G ,
Bojarski AJ ,
Lamaty F ,
Becamel C ,
Zussy C,
Chaumont-Dubel S ,
Popik P ,
Nury H ,
Marin P ,
Givalois L ,
Zajdel P
(2023) J Med Chem , 66 , 14928 - 14947
,
Lopez-Sanchez U ,
Vitalis M ,
Canet G ,
Satala G ,
Olejarz-Maciej A ,
Golebiowska J,
Kurczab R ,
Pietrus W ,
Kubacka M,
Moreau C ,
Walczak M ,
Blicharz-Futera K ,
Bento O ,
Bantreil X ,
Subra G ,
Bojarski AJ ,
Lamaty F ,
Becamel C ,
Zussy C,
Chaumont-Dubel S ,
Popik P ,
Nury H ,
Marin P ,
Givalois L ,
Zajdel P
(2023) J Med Chem , 66 , 14928 - 14947
Grant Support:
- European Research Council (ERC): PentaBrain (European Union)