Structure for danoprevir (S29.001 inhibitor)

Summary Structure Literature

 

TERTIARY STRUCTURE DATA
Comment Resolution PDB PDBe SCOP CATH PDBSum Proteopedia Reference
hepacivirin ( hepatitis C virus)
Arg155Lys variant; complex with danoprevir 1.16 Å 3SU0 3SU0 3SU0 3SU0 3SU0 3SU0
Asp168Ala variant; complex with danoprevir 1.40 Å 3SU1 3SU1 3SU1 3SU1 3SU1 3SU1
Ala156Thr variant; complex with danoprevir 1.50 Å 3SU2 3SU2 3SU2 3SU2 3SU2 3SU2
Tyr56His/Asp168Ala double mutant; complex with danoprevir 1.80 Å 6C2N 6C2N 6C2N 6C2N 6C2N 6C2N