Literature for benzamidine (S01.151 inhibitor)

(Topics flags: S Structure, I Inhibitor, V Review. To select only the references relevant to a single topic, click the link above. See explanation.)

2018
1. Pilon,A.M., Campos,W.G., Silva,C.R., Cordeiro,G., Silva,C.R. and Oliveira,M.G.A.
   Protease inhibitory, insecticidal and deterrent effects of the trypsin-inhibitor benzamidine on the velvetbean caterpillar in soybean
   An Acad Bras Cienc (2018) 90, 3475-3482. PubMed  Europe PubMed DOI  I
2016
2. Teo,I., Mayne,C.G., Schulten,K. and Lelievre,T.
   Adaptive multilevel splitting method for molecular dynamics calculation of benzamidine-trypsin dissociation time
   J Chem Theory Comput (2016) 12, 2983-2989. PubMed  Europe PubMed DOI  I
2011
3. Kumar,P., Singh,P. and Singh,J.P.
   Topological descriptor based QSAR study of benzamidine as inhibitor of thrombin
   J Chem Pharm Res (2011) 3, 296-303.  I
2009
4. Shi,Y., Jiao,D., Schnieders,M.J. and Ren,P.
   Trypsin-ligand binding free energy calculation with AMOEBA
   Conf Proc IEEE Eng Med Biol Soc (2009) 2009, 2328-2331. PubMed  Europe PubMed DOI  I
2005
5. [YEAR:12-8-2005]Warejcka,D.J. and Twining,S.S.
   Specific conformational changes of plasminogen induced by chloride ions, 6-aminohexanoic acid and benzamidine, but not the overall openness of plasminogen regulate, production of biologically active angiostatins
   Biochem J (12-8-2005) 392, 703-712. PubMed  Europe PubMed DOI  PMC  EPMC  I
1998
6. [YEAR:1-12-1998]Presnell,S.R., Patil,G.S., Mura,C., Jude,K.M., Conley,J.M., Bertrand,J.A., Kam,C.M., Powers,J.C. and Williams,L.D.
   Oxyanion-mediated inhibition of serine proteases
   Biochemistry (1-12-1998) 37, 17068-17081. PubMed  Europe PubMed DOI  S  I
1993
7. Smalas,A. and Hordvik,A.
   Structure determination and refinement of benzamidine-inhibited trypsin from the North Atlantic salmon (Salmo salar) at 1.82 A resolution
   Acta Crystallogr D Biol Crystallogr (1993) 49, 318-330. PubMed  Europe PubMed DOI  S  I
1991
8. [YEAR:25-10-1991]Banner,D.W. and Hadvary,P.
   Crystallographic analysis at 3.0-A resolution of the binding to human thrombin of four active site-directed inhibitors
   J Biol Chem (25-10-1991) 266, 20085-20093. PubMed  Europe PubMed  I
1990
9. Smalas,A.O., Hordvik,A., Hansen,L.K., Hough,E. and Jynge,K.
   Crystallization and preliminary X-ray crystallographic studies of benzamidine-inhibited trypsin from the North Atlantic salmon (Salmo salar)
   J Mol Biol (1990) 214, 355-358. PubMed  Europe PubMed DOI  I
1986
10. Powers,J.C. and Harper,J.W.
    Inhibitors of serine proteinases
    (1986) , 55-152.  V  I
1980
11. Takahashi,K., Nagasawa,S. and Koyama,J.
    Effect of C1-inhibitor, benzamidine, and heat treatment on the hydrolytic activity of a subcomponent of the first component of human complement, C1s
    Biochim Biophys Acta (1980) 611, 196-204. PubMed  Europe PubMed  I
1978
12. Parrish,R.F., Straus,J.W., Paulson,J.D., Polakoski,K.L., Tidwell,R.R., Geratz,J.D. and Stevens,F.M.
    Structure-activity relationships for the inhibition of acrosin by benzamidine derivatives
    J Med Chem (1978) 21, 1132-1136. PubMed  Europe PubMed  I
1977
13. Zahler,W.L. and Polakoski,K.L.
    Benzamidine as an inhibitor of proacrosin activation in bull sperm
    Biochim Biophys Acta (1977) 480, 461-468. PubMed  Europe PubMed  I
1976
14. Holleman,W.H. and Weiss,L.J.
    The thrombin-like enzyme from Bothrops atrox snake venom. Properties of the enzyme purified by affinity chromatography on p-aminobenzamidine substituted agarose
    J Biol Chem (1976) 251, 1663-1669. PubMed  Europe PubMed  I
1975
15. [YEAR:15-11-1975]Bode,W. and Schwager,P.
    The refined crystal structure of bovine beta-trypsin at 1.8 A resolution. II. Crystallographic refinement, calcium binding site, benzamidine binding site and active site at pH 7.0
    J Mol Biol (15-11-1975) 98, 693-717. PubMed  Europe PubMed  S  I
1974
16. [YEAR:25-2-1974]Krieger,M., Kay,L.M. and Stroud,R.M.
    Structure and specific binding of trypsin: comparison of inhibited derivatives and a model for substrate binding
    J Mol Biol (25-2-1974) 83, 209-230. PubMed  Europe PubMed  I
1973
17. Schleuning,W.D., Schiessler,H. and Fritz,H.
    Highly purified acrosomal proteinase (boar acrosin): isolation by affinity chromatography using benzamidine-cellulose and stabilization
    Hoppe Seylers Z Physiol Chem (1973) 354, 550-554. PubMed  Europe PubMed  I
1972
18. Schmer,G.
    The purification of bovine thrombin by affinity chromatography on benzamidine-agarose
    Hoppe Seylers Z Physiol Chem (1972) 353, 810-814. PubMed  Europe PubMed  I
1970
19. [YEAR:30-6-1970]Geratz,J.D.
    Inhibition of thrombin, plasmin and plasminogen activation by amidino compounds
    Thromb Diath Haemorrh (30-6-1970) 23, 486-499. PubMed  Europe PubMed  I
1969
20. [YEAR:15-12-1969]Geratz,J.D.
    Inhibitory effect of aromatic diamidines on trypsin and enterokinase
    Experientia (15-12-1969) 25, 1254-1255. PubMed  Europe PubMed DOI  I
1968
21. East,E.J. and Trowbridge,C.G.
    Binding of benzamidine and protons to trypsin as measured by difference spectra
    Arch Biochem Biophys (1968) 125, 334-343. PubMed  Europe PubMed  I
22. Markwardt,F., Landmann,H. and Walsmann,P.
    Comparative studies on the inhibition of trypsin, plasmin, and thrombin by derivatives of benzylamine and benzamidine
    Eur J Biochem (1968) 6, 502-506. PubMed  Europe PubMed  I
23. Tanizawa,K., Ishii,S.I. and Kanaoka,Y.
    Trypsin substrates derived from benzamidine: application to active site titration and isolation of acyl-enzyme intermediate
    Biochem Biophys Res Commun (1968) 32, 893-897. PubMed  Europe PubMed  I
1966
24. [YEAR:15-2-1966]Geratz,J.D.
    p-Aminobenzamidine as inhibitor of trypsinogen activation
    Experientia (15-2-1966) 22, 73-74. PubMed  Europe PubMed DOI  I