Literature for K777 (C01.075 inhibitor)

Summary Structure Literature

(Topics flags: S Structure, T Target, I Inhibitor, E Expression. To select only the references relevant to a single topic, click the link above. See explanation.)

    2020
  1. Jilkova,A., Horn,M. and Mares,M.
    Structural and functional characterization of Schistosoma mansoni cathepsin B1
    Methods Mol Biol2151, 145-158. PubMed  Europe PubMed DOI  E  S  I
  2. 2013
  3. Ndao,M., Nath-Chowdhury,M., Sajid,M., Marcus,V., Mashiyama,S.T., Sakanari,J., Chow,E., Mackey,Z., Land,K.M., Jacobson,M.P., Kalyanaraman,C., McKerrow,J.H., Arrowood,M.J. and Caffrey,C.R.
    A cysteine protease inhibitor rescues mice from a lethal Cryptosporidium parvum infection
    Antimicrob Agents Chemother57, 6063-6073. PubMed  Europe PubMed DOI  I
  4. 2012
  5. Lee,G.M., Balouch,E., Goetz,D.H., Lazic,A., McKerrow,J.H. and Craik,C.S.
    Mapping inhibitor binding modes on an active cysteine protease via nuclear magnetic resonance spectroscopy
    Biochemistry51, 10087-10098. PubMed  Europe PubMed DOI  E  S  I
  6. 2009
  7. Caffrey,C.R. and Steverding,D.
    Kinetoplastid papain-like cysteine peptidases
    Mol Biochem Parasitol167, 12-19. PubMed  Europe PubMed DOI  I
  8. Kerr,I.D., Lee,J.H., Farady,C.J., Marion,R., Rickert,M., Sajid,M., Pandey,K.C., Caffrey,C.R., Legac,J., Hansell,E., McKerrow,J.H., Craik,C.S., Rosenthal,P.J. and Brinen,L.S.
    Vinyl sulfones as antiparasitic agents and a structural basis for drug design
    J Biol Chem284, 25697-25703. PubMed  Europe PubMed DOI  S  I
  9. 2007
  10. [YEAR:9-1-2007]Abdulla,M.H., Lim,K.C., Sajid,M., McKerrow,J.H. and Caffrey,C.R.
    Schistosomiasis mansoni: novel chemotherapy using a cysteine protease inhibitor
    PLoS Medicine4, e14-e14. PubMed  Europe PubMed DOI  T  I
  11. Doyle,P.S., Zhou,Y.M., Engel,J.C. and McKerrow,J.H.
    A cysteine protease inhibitor cures Chagas' disease in an immunodeficient-mouse model of infection
    Antimicrob Agents Chemother51, 3932-3939. PubMed  Europe PubMed DOI  I
  12. Melendez-Lopez,S.G., Herdman,S., Hirata,K., Choi,M.H., Choe,Y., Craik,C., Caffrey,C.R., Hansell,E., Chavez-Munguia,B., Chen,Y.T., Roush,W.R., McKerrow,J., Eckmann,L., Guo,J., Stanley,S.L., Jr. and Reed,S.L.
    Use of recombinant Entamoeba histolytica cysteine proteinase 1 to identify a potent inhibitor of amebic invasion in a human colonic model
    Eukaryot Cell6, 1130-1136. PubMed  Europe PubMed DOI  I
  13. 2006
  14. [YEAR:2-10-2006]Nikolskaia,O.V., de,A.L., Kim,Y.V., Lonsdale-Eccles,J.D., Fukuma,T., Scharfstein,J. and Grab,D.J.
    Blood-brain barrier traversal by African trypanosomes requires calcium signaling induced by parasite cysteine protease
    J Clin Invest116, 2739-2747. PubMed  Europe PubMed DOI  I
  15. 2005
  16. Barr,S.C., Warner,K.L., Kornreic,B.G., Piscitelli,J., Wolfe,A., Benet,L. and McKerrow,J.H.
    A cysteine protease inhibitor protects dogs from cardiac damage during infection by Trypanosoma cruzi
    Antimicrob Agents Chemother49, 5160-5161. PubMed  Europe PubMed DOI  I
  17. 2000
  18. Jacobsen,W., Christians,U. and Benet,L.Z.
    In vitro evaluation of the disposition of a novel cysteine protease inhibitor
    Drug Metab Dispos28, 1343-1351. PubMed  Europe PubMed  I
  19. 1998
  20. [YEAR:17-8-1998]Engel,J.C., Doyle,P.S., Hsieh,I. and McKerrow,J.H.
    Cysteine protease inhibitors cure an experimental Trypanosoma cruzi infection
    J Exp Med188, 725-734. PubMed  Europe PubMed DOI  I