Literature for fumagillin (M24.002 inhibitor)

(Topics flags: S Structure, K Knockout, I Inhibitor. To select only the references relevant to a single topic, click the link above. See explanation.)

2011
1. Ma,A.C., Fung,T.K., Lin,R.H., Chung,M.I., Yang,D., Ekker,S.C. and Leung,A.Y.
   Methionine aminopeptidase 2 is required for HSC initiation and proliferation
   Blood118, 5448-5457. PubMed  Europe PubMed DOI  I
2009
2. Alvarado,J.J., Nemkal,A., Sauder,J.M., Russell,M., Akiyoshi,D.E., Shi,W., Almo,S.C. and Weiss,L.M.
   Structure of a microsporidian methionine aminopeptidase type 2 complexed with fumagillin and TNP-470
   Mol Biochem Parasitol168, 158-167. PubMed  Europe PubMed DOI  S  I
3. Arico-Muendel,C.C., Benjamin,D.R., Caiazzo,T.M., Centrella,P.A., Contonio,B.D., Cook,C.M., Doyle,E.G., Hannig,G., Labenski,M.T., Searle,L.L., Lind,K., Morgan,B.A., Olson,G., Paradise,C.L., Self,C., Skinner,S.R., Sluboski,B., Svendsen,J.L., Thompson,C.D., Westlin,W. and White,K.F.
   Carbamate analogues of fumagillin as potent, targeted inhibitors of methionine aminopeptidase-2
   J Med Chem52, 8047-8056. PubMed  Europe PubMed DOI  I
4. Chen,X., Xie,S., Bhat,S., Kumar,N., Shapiro,T.A. and Liu,J.O.
   Fumagillin and fumarranol interact with P. falciparum methionine aminopeptidase 2 and inhibit malaria parasite growth in vitro and in vivo
   Chem Biol16, 193-202. PubMed  Europe PubMed DOI  I
2004
5. [YEAR:9-8-2004]Asami,Y., Kakeya,H., Onose,R., Chang,Y.H., Toi,M. and Osada,H.
   RK-805, an endothelial-cell-growth inhibitor produced by Neosartorya sp., and a docking model with methionine aminopeptidase-2
   Tetrahedron60, 7085-7091. DOI  I
6. [YEAR:8-10-2004]Boxem,M., Tsai,C.W., Zhang,Y., Saito,R.M. and Liu,J.O.
   The C. elegans methionine aminopeptidase 2 analog map-2 is required for germ cell proliferation
   FEBS Lett576, 245-250. PubMed  Europe PubMed DOI  K  I
7. [YEAR:5-3-2004]Brdlik,C.M. and Crews,C.M.
   A single amino acid residue defines the difference in ovalicin sensitivity between type I and II methionine aminopeptidases
   J Biol Chem279, 9475-9480. PubMed  Europe PubMed DOI  I
8. [YEAR:1-5-2004]Kim,S., LaMontagne,K., Sabio,M., Sharma,S., Versace,R.W., Yusuff,N. and Phillips,P.E.
   Depletion of methionine aminopeptidase 2 does not alter cell response to fumagillin or bengamides
   Cancer Res64, 2984-2987. PubMed  Europe PubMed DOI  I
2000
9. [YEAR:3-1-2000]Han,C.K., Ahn,S.K., Choi,N.S., Hong,R.K., Moon,S.K., Chun,H.S., Lee,S.J., Kim,J.W., Hong,C.I., Kim,D., Yoon,J.H. and No,K.T.
   Design and synthesis of highly potent fumagillin analogues from homology modeling for a human MetAP-2
   Bioorg Med Chem Lett10, 39-43. PubMed  Europe PubMed DOI  I
10. Wang,J., Lou,P. and Henkin,J.
    Selective inhibition of endothelial cell proliferation by fumagillin is not due to differential expression of methionine aminopeptidases
    J Cell Biochem77, 465-473. PubMed  Europe PubMed DOI  I
1998
11. [YEAR:22-12-1998]Griffith,E.C., Su,Z., Niwayama,S., Ramsay,C.A., Chang,Y.H. and Liu,J.O.
    Molecular recognition of angiogenesis inhibitors fumagillin and ovalicin by methionine aminopeptidase 2
    Proc Natl Acad Sci U S A95, 15183-15188. PubMed  Europe PubMed DOI  I
12. [YEAR:13-11-1998]Liu,S., Widom,J., Kemp,C.W., Crews,C.M. and Clardy,J.
    Structure of human methionine aminopeptidase-2 complexed with fumagillin
    Science282, 1324-1327. PubMed  Europe PubMed  S  I
13. [YEAR:13-10-1998]Lowther,W.T., McMillen,D.A., Orville,A.M. and Matthews,B.W.
    The anti-angiogenic agent fumagillin covalently modifies a conserved active-site histidine in the Escherichia coli methionine aminopeptidase
    Proc Natl Acad Sci U S A95, 12153-12157. PubMed  Europe PubMed DOI  I
1997
14. Sin,N., Meng,L., Wang,M.Q., Wen,J.J., Bornmann,W.G. and Crews,C.M.
    The anti-angiogenic agent fumagillin covalently binds and inhibits the methionine aminopeptidase, MetAP-2
    Proc Natl Acad Sci U S A94, 6099-6103. PubMed  Europe PubMed DOI  I