Literature for PL-100 (A02.001 inhibitor)

Summary Structure Literature

(Topics flags: I Inhibitor, V Review. To select only the references relevant to a single topic, click the link above. See explanation.)

    2013
  1. Asahchop,E.L., Oliveira,M., Quashie,P.K., Moisi,D., Martinez-Cajas,J.L., Brenner,B.G., Tremblay,C.L. and Wainberg,M.A.
    In vitro and structural evaluation of PL-100 as a potential second-generation HIV-1 protease inhibitor
    J Antimicrob Chemother68, 105-112. PubMed  Europe PubMed DOI  I
  2. 2010
  3. Jones,K.L., Holloway,M.K., Su,H.P., Carroll,S.S., Burlein,C., Touch,S., Distefano,D.J., Sanchez,R.I., Williams,T.M., Vacca,J.P. and Coburn,C.A.
    Epsilon substituted lysinol derivatives as HIV-1 protease inhibitors
    Bioorg Med Chem Lett20, 4065-4068. PubMed  Europe PubMed DOI  I
  4. 2008
  5. Dandache,S., Coburn,C.A., Oliveira,M., Allison,T.J., Holloway,M.K., Wu,J.J., Stranix,B.R., Panchal,C., Wainberg,M.A. and Vacca,J.P.
    PL-100, a novel HIV-1 protease inhibitor displaying a high genetic barrier to resistance: an in vitro selection study
    J Med Virol80, 2053-2063. PubMed  Europe PubMed DOI  I
  6. Gulnik,S.V. and Eissenstat,M.
    Approaches to the design of HIV protease inhibitors with improved resistance profiles
    Curr Opin HIV AIDS3, 633-641. PubMed  Europe PubMed DOI  V  I
  7. 2007
  8. Dandache,S., Sevigny,G., Yelle,J., Stranix,B.R., Parkin,N., Schapiro,J.M., Wainberg,M.A. and Wu,J.J.
    In vitro antiviral activity and cross-resistance profile of PL-100, a novel protease inhibitor of human immunodeficiency virus type 1
    Antimicrob Agents Chemother51, 4036-4043. PubMed  Europe PubMed DOI  I
  9. 2006
  10. [YEAR:24-4-2006]Stranix,B.R., Lavallee,J.F., Sevigny,G., Yelle,J., Perron,V., LeBerre,N., Herbart,D. and Wu,J.J.
    Lysine sulfonamides as novel HIV-protease inhibitors: Nepsilon-acyl aromatic alpha-amino acids
    Bioorg Med Chem Lett16, 3459-3462. PubMed  Europe PubMed DOI  I