EMBL-EBI | Chemical Biology | ChEBI
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| ChEBI ID | CHEBI:77748 |
| ChEBI Name | EC 3.6.3.44 (xenobiotic-transporting ATPase) inhibitor |
| Stars | |
| Definition | An EC 3.6.3.* (acid anhydride hydrolase catalysing transmembrane movement of substances) inhibitor that interferes with the action of xenobiotic-transporting ATPase (EC 3.6.3.44). |
| Last Modified | 7 December 2016 |
| Submitter | Gareth Owen |
| Wikipedia |
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| ChEBI Ontology |
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| Outgoing Relation(s) |
| EC 3.6.3.44 (xenobiotic-transporting ATPase) inhibitor (CHEBI:77748) is a EC 3.6.3.* (acid anhydride hydrolase catalysing transmembrane movement of substances) inhibitor (CHEBI:76895) |
| Incoming Relation(s) |
| dexverapamil (CHEBI:77734) has role EC 3.6.3.44 (xenobiotic-transporting ATPase) inhibitor (CHEBI:77748) |
| dexverapamil hydrochloride (CHEBI:77739) has role EC 3.6.3.44 (xenobiotic-transporting ATPase) inhibitor (CHEBI:77748) |
| itraconazole (CHEBI:6076) has role EC 3.6.3.44 (xenobiotic-transporting ATPase) inhibitor (CHEBI:77748) |
| norverapamil (CHEBI:132050) has role EC 3.6.3.44 (xenobiotic-transporting ATPase) inhibitor (CHEBI:77748) |
| quinidine (CHEBI:28593) has role EC 3.6.3.44 (xenobiotic-transporting ATPase) inhibitor (CHEBI:77748) |
| verapamil (CHEBI:9948) has role EC 3.6.3.44 (xenobiotic-transporting ATPase) inhibitor (CHEBI:77748) |
| Synonyms | Source |
|---|---|
| steroid-transporting ATPase inhibitor | ChEBI |
| P-glycoprotein inhibitor | ChEBI |
| EC 3.6.3.44 (xenobiotic-transporting ATPase) inhibitors | ChEBI |
| multidrug-resistance protein inhibitor | ChEBI |
| MDR protein inhibitor | ChEBI |
| EC 3.6.3.44 inhibitors | ChEBI |
| Manual Xrefs | Databases |
|---|---|
| Xenobiotic-transporting_ATPase | Wikipedia |