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Structure of the human neutral amino acid transporter ASCT2 in complex with nanobody 469
Resolution: 2.31 Å
EM Method: Single-particle
Fitted PDBs: 8oud
Q-score: 0.666
Khare S, Villalba MI, Canul-Tec JC, Cajiao AB, Kumar A, Backovic M, Rey FA, Pardon E, Steyaert J, Perez C, Reyes N
Nat Struct Mol Biol (2024) [ Pubmed: 38671230 DOI: doi:10.1038/s41594-024-01295-6 ]
- Sodium ion (22 Da, Ligand)
- Alanine (89 Da, Ligand)
- Nanobody 69 (Complex from Lama glama)
- Neutral amino acid transporter b(0) (56 kDa, Protein from Homo sapiens)
- Alanine serine cysteine transporter 2 (Complex from Homo sapiens)
- Cholesterol hemisuccinate (486 Da, Ligand)
- Water (18 Da, Ligand)
- Complex of human asct2 with nanobody 69 (200 kDa, Complex)
- Nanobody 469 (13 kDa, Protein from Lama glama)
Complex of human ASCT2 with Syncytin-1
Resolution: 2.62 Å
EM Method: Single-particle
Fitted PDBs: 8ouh
Q-score: 0.553
Khare S, Villalba MI, Canul-Tec JC, Cajiao AB, Kumar A, Backovic M, Rey FA, Pardon E, Steyaert J, Perez C, Reyes N
Nat Struct Mol Biol (2024) [ Pubmed: 38671230 DOI: doi:10.1038/s41594-024-01295-6 ]
- Alanine (89 Da, Ligand)
- Syncytin-1 (Complex from Homo sapiens)
- Complex of asct2 with synctin-1 (180 MDa, Complex)
- Syncytin-1 (49 kDa, Protein from Homo sapiens)
- Alanine serine cysteine transporter 2 (Complex from Homo sapiens)
- Neutral amino acid transporter b(0) (58 kDa, Protein from Homo sapiens)
Complex of ASCT2 with Suppressyn
Resolution: 3.39 Å
EM Method: Single-particle
Fitted PDBs: 8oui
Q-score: 0.435
Khare S, Villalba MI, Canul-Tec JC, Cajiao AB, Kumar A, Backovic M, Rey FA, Pardon E, Steyaert J, Perez C, Reyes N
Nat Struct Mol Biol (2024) [ Pubmed: 38671230 DOI: doi:10.1038/s41594-024-01295-6 ]
- Complex of alanine serine cysteine transporter 2 with suppressyn (Complex from Homo sapiens)
- Suppressyn (18 kDa, Protein from Homo sapiens)
- Neutral amino acid transporter b(0) (57 kDa, Protein from Homo sapiens)
- Alanine (89 Da, Ligand)
Heterotrimeric Complex of Human ASCT2 with Syncytin-1
Resolution: 3.5 Å
EM Method: Single-particle
Fitted PDBs: 8ouj
Q-score: 0.339
Khare S, Villalba MI, Canul-Tec JC, Cajiao AB, Kumar A, Backovic M, Rey FA, Pardon E, Steyaert J, Perez C, Reyes N
Nat Struct Mol Biol (2024) [ Pubmed: 38671230 DOI: doi:10.1038/s41594-024-01295-6 ]
- Alanine (89 Da, Ligand)
- Syncytin-1 (Complex from Homo sapiens)
- Syncytin-1 (49 kDa, Protein from Homo sapiens)
- Alanine serine cysteine transporter 2 (Complex from Homo sapiens)
- Complex asct2 with syncytin-1 (180 MDa, Complex)
- Neutral amino acid transporter b(0) (58 kDa, Protein from Homo sapiens)
ACE2-B0AT1 complex bound with glutamine
Resolution: 3.2 Å
EM Method: Single-particle
Fitted PDBs: 8i92
Q-score: 0.452
Li Y, Chen Y, Zhang Y, Shen Y, Xu K, Liu Y, Wang Z, Yan R
Cell Discov (2023) 9 pp. 93-93 [ Pubmed: 37684251 DOI: doi:10.1038/s41421-023-00596-2 ]
- Angiotensin-converting enzyme 2 (95 kDa, Protein from Homo sapiens)
- Sodium-dependent neutral amino acid transporter b(0)at1 (68 kDa, Protein from Homo sapiens)
- Glutamine (146 Da, Ligand)
- Ace2-b0at1 complex bound with glutamine (Complex from Homo sapiens)
- Zinc ion (65 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
ACE2-B0AT1 complex bound with methionine
Resolution: 3.1 Å
EM Method: Single-particle
Fitted PDBs: 8i93
Q-score: 0.474
Li Y, Chen Y, Zhang Y, Shen Y, Xu K, Liu Y, Wang Z, Yan R
Cell Discov (2023) 9 pp. 93-93 [ Pubmed: 37684251 DOI: doi:10.1038/s41421-023-00596-2 ]
- Sodium-dependent neutral amino acid transporter b(0)at1 (73 kDa, Protein from Homo sapiens)
- Methionine (149 Da, Ligand)
- Angiotensin-converting enzyme 2 (86 kDa, Protein from Homo sapiens)
- Zinc ion (65 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Ace2-b0at1 complex bound with methionine (Complex from Homo sapiens)
ACE2 -Targeting Monoclonal Antibody as Potent and Broad-Spectrum Coronavirus Blocker
Resolution: 3.2 Å
EM Method: Single-particle
Fitted PDBs: 7v61
Q-score: 0.366
Chen Y, Zhang YN, Yan R, Wang G, Zhang Y, Zhang ZR, Li Y, Ou J, Chu W, Liang Z, Wang Y, Chen YL, Chen G, Wang Q, Zhou Q, Zhang B, Wang C
Signal Transduct Target Ther (2021) 6 pp. 315-315 [ DOI: doi:10.1038/s41392-021-00740-y Pubmed: 34433803 ]
- Ace2-b0at1 complex (Complex from Homo sapiens)
- Sodium-dependent neutral amino acid transporter b(0)at1 (73 kDa, Protein from Homo sapiens)
- Water (18 Da, Ligand)
- Zinc ion (65 Da, Ligand)
- 3e8 (23 kDa, Protein from Severe acute respiratory syndrome coronavirus 2)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- 3e8 (49 kDa, Protein from Severe acute respiratory syndrome coronavirus 2)
- Angiotensin-converting enzyme 2 (93 kDa, Protein from Homo sapiens)
Conformation 1 of S-ACE2-B0AT1 ternary complex
Resolution: 8.3 Å
EM Method: Single-particle
Fitted PDBs: 7dwx
Q-score: 0.059
Yan R, Zhang Y, Li Y, Ye F, Guo Y, Xia L, Zhong X, Chi X, Zhou Q
Cell Res (2021) 31 pp. 717-719 [ DOI: doi:10.1038/s41422-021-00490-0 Pubmed: 33737693 ]
- Spike glycoprotein (142 kDa, Protein from Severe acute respiratory syndrome coronavirus 2)
- Leucine (131 Da, Ligand)
- Conformation 1 of s-ace2-b0at1 ternary complex (Complex from Homo sapiens)
- Sodium-dependent neutral amino acid transporter b(0)at1 (73 kDa, Protein from Homo sapiens)
- Water (18 Da, Ligand)
- Zinc ion (65 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- Angiotensin-converting enzyme 2 (93 kDa, Protein from Homo sapiens)
The 2019-nCoV RBD/ACE2-B0AT1 complex
Resolution: 2.9 Å
EM Method: Single-particle
Fitted PDBs: 6m17
Q-score: 0.42
Yan R, Zhang Y, Li Y, Xia L, Guo Y, Zhou Q
Science (2020) 367 pp. 1444-1448 [ Pubmed: 32132184 DOI: doi:10.1126/science.abb2762 ]
- The sars-cov-2 rbd (Complex from Severe acute respiratory syndrome coronavirus 2)
- Ace2-b0at1 (Complex from Homo sapiens)
- Angiotensin-converting enzyme 2 (93 kDa, Protein from Homo sapiens)
- Spike protein s1 (25 kDa, Protein from Severe acute respiratory syndrome coronavirus 2)
- Sodium-dependent neutral amino acid transporter b(0)at1 (73 kDa, Protein from Homo sapiens)
- Water (18 Da, Ligand)
- Zinc ion (65 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)
- The sars-cov-2 rbd/ace2-b0at1 complex (Complex)
- Leucine (131 Da, Ligand)
Resolution: 2.9 Å
EM Method: Single-particle
Fitted PDBs: 6m18
Q-score: 0.489
Yan R, Zhang Y, Li Y, Xia L, Guo Y, Zhou Q
Science (2020) 367 pp. 1444-1448 [ Pubmed: 32132184 DOI: doi:10.1126/science.abb2762 ]
- Ace2-b0at1 complex (Complex from Homo sapiens)
- Angiotensin-converting enzyme 2 (93 kDa, Protein from Homo sapiens)
- 1,2-diacyl-glycerol-3-sn-phosphate (704 Da, Ligand)
- Sodium-dependent neutral amino acid transporter b(0)at1 (73 kDa, Protein from Homo sapiens)
- Water (18 Da, Ligand)
- Zinc ion (65 Da, Ligand)
- 2-acetamido-2-deoxy-beta-d-glucopyranose (221 Da, Ligand)