Structure for telaprevir (S29.001 inhibitor)

Summary Structure Literature

 

TERTIARY STRUCTURE DATA
Comment Resolution PDB PDBe SCOP CATH PDBSum Proteopedia Reference
hepacivirin ( hepatitis C virus)
complex with telaprevir 1.40 Å 3SV6 3SV6 3SV6 3SV6 3SV6 3SV6
Arg155Lys variant; complex with telaprevir 1.55 Å 3SV7 3SV7 3SV7 3SV7 3SV7 3SV7
Asp168Ala variant; complex with telaprevir 2.50 Å 3SV8 3SV8 3SV8 3SV8 3SV8 3SV8
Ala156Thr variant; complex with telaprevir 1.60 Å 3SV9 3SV9 3SV9 3SV9 3SV9 3SV9