Literature for angiotensin IV (M01.011 inhibitor)

Summary Literature

(Topics flags: T Target, P Specificity, I Inhibitor, K Knockout, V Review. To select only the references relevant to a single topic, click the link above. See explanation.)

    2013
  1. Loyens,E., De Bundel,D., Demaegdt,H., Chai,S.Y., Vanderheyden,P., Michotte,Y., Gard,P. and Smolders,I.
    Antidepressant-like effects of oxytocin in mice are dependent on the presence of insulin-regulated aminopeptidase
    Int J Neuropsychopharmacol16, 1153-1163. PubMed  Europe PubMed DOI  K  I
  2. Nikolaou,A., Eynde,I.V., Tourwe,D., Vauquelin,G., Toth,G., Mallareddy,J.R., Poglitsch,M., Van Ginderachter,J.A. and Vanderheyden,P.M.
    [3H]IVDE77, a novel radioligand with high affinity and selectivity for the insulin-regulated aminopeptidase
    Eur J Pharmacol702, 93-102. PubMed  Europe PubMed DOI  I
  3. 2012
  4. Andersson,H. and Hallberg,M.
    Discovery of inhibitors of insulin-regulated aminopeptidase as cognitive enhancers
    Int J Hypertens2012, 789671-789671. PubMed  Europe PubMed DOI  I
  5. Demaegdt,H., De Backer,J.P., Lukaszuk,A., Toth,G., Szemenyei,E., Tourwe,D. and Vauquelin,G.
    Angiotensin IV displays only low affinity for native insulin-regulated aminopeptidase (IRAP)
    Fundam Clin Pharmacol26, 194-197. PubMed  Europe PubMed DOI  I
  6. 2011
  7. Albiston,A.L., Diwakarla,S., Fernando,R.N., Mountford,S.J., Yeatman,H.R., Morgan,B., Pham,V., Holien,J.K., Parker,M.W., Thompson,P.E. and Chai,S.Y.
    Identification and development of specific inhibitors for insulin-regulated aminopeptidase as a new class of cognitive enhancers
    Br J Pharmacol164, 37-47. PubMed  Europe PubMed DOI  I
  8. Andersson,H., Demaegdt,H., Johnsson,A., Vauquelin,G., Lindeberg,G., Hallberg,M., Erdelyi,M., Karlen,A. and Hallberg,A.
    Potent macrocyclic inhibitors of insulin-regulated aminopeptidase (IRAP) by olefin ring-closing metathesis
    J Med Chem54, 3779-3792. PubMed  Europe PubMed DOI  I
  9. 2010
  10. Albiston,A.L., Fernando,R.N., Yeatman,H.R., Burns,P., Ng,L., Daswani,D., Diwakarla,S., Pham,V. and Chai,S.Y.
    Gene knockout of insulin-regulated aminopeptidase: loss of the specific binding site for angiotensin IV and age-related deficit in spatial memory
    Neurobiol Learn Mem93, 19-30. PubMed  Europe PubMed DOI  K  I
  11. Andersson,H., Demaegdt,H., Vauquelin,G., Lindeberg,G., Karlen,A., Hallberg,M., Erdelyi,M. and Hallberg,A.
    Disulfide cyclized tripeptide analogues of angiotensin IV as potent and selective inhibitors of insulin-regulated aminopeptidase (IRAP)
    J Med Chem53, 8059-8071. PubMed  Europe PubMed DOI  I
  12. Beyer,C.E., Dwyer,J.M., Platt,B.J., Neal,S., Luo,B., Ling,H.P., Lin,Q., Mark,R.J., Rosenzweig-Lipson,S. and Schechter,L.E.
    Angiotensin IV elevates oxytocin levels in the rat amygdala and produces anxiolytic-like activity through subsequent oxytocin receptor activation
    Psychopharmacology (Berl)209, 303-311. PubMed  Europe PubMed DOI  I
  13. 2008
  14. Chai,S.Y., Yeatman,H.R., Parker,M.W., Ascher,D.B., Thompson,P.E., Mulvey,H.T. and Albiston,A.L.
    Development of cognitive enhancers based on inhibition of insulin-regulated aminopeptidase
    BMC Neurosci9 Suppl 2, S14-S14. PubMed  Europe PubMed DOI  T  I
  15. Cohen,M., Wuillemin,C., Chai,S.Y. and Bischof,P.
    Effects of ligands or substrate of insulin-regulated aminopeptidase (IRAP) on trophoblast invasion
    J Pept Sci14, 883-887. PubMed  Europe PubMed DOI  I
  16. Demaegdt,H., Smitz,L., De Backer,J.P., Le,M.T., Bauwens,M., Szemenyei,E., Toth,G., Michotte,Y., Vanderheyden,P. and Vauquelin,G.
    Translocation of the insulin-regulated aminopeptidase to the cell surface: detection by radioligand binding
    Br J Pharmacol154, 872-881. PubMed  Europe PubMed DOI  I
  17. Stragier,B., De Bundel,D., Sarre,S., Smolders,I., Vauquelin,G., Dupont,A., Michotte,Y. and Vanderheyden,P.
    Involvement of insulin-regulated aminopeptidase in the effects of the renin-angiotensin fragment angiotensin IV: a review
    Heart Fail Rev13, 321-337. PubMed  Europe PubMed DOI  V  I
  18. Ye,S., Chai,S.Y., Lew,R.A., Ascher,D.B., Morton,C.J., Parker,M.W. and Albiston,A.L.
    Identification of modulating residues defining the catalytic cleft of insulin-regulated aminopeptidase
    Biochem Cell Biol86, 251-261. PubMed  Europe PubMed DOI  P  I
  19. 2007
  20. Fernando,R.N., Luff,S.E., Albiston,A.L. and Chai,S.Y.
    Sub-cellular localization of insulin-regulated membrane aminopeptidase, IRAP to vesicles in neurons
    J Neurochem102, 967-976. PubMed  Europe PubMed DOI  I
  21. Stragier,B., Demaegdt,H., De Bundel,D., Smolders,I., Sarre,S., Vauquelin,G., Ebinger,G., Michotte,Y. and Vanderheyden,P.
    Involvement of insulin-regulated aminopeptidase and/or aminopeptidase N in the angiotensin IV-induced effect on dopamine release in the striatum of the rat
    Brain Res1131, 97-105. PubMed  Europe PubMed DOI  I
  22. Ye,S., Chai,S.Y., Lew,R.A. and Albiston,A.L.
    Insulin-regulated aminopeptidase: analysis of peptide substrate and inhibitor binding to the catalytic domain
    Biol Chem388, 399-403. PubMed  Europe PubMed DOI  I
  23. 2004
  24. [YEAR:1-10-2004]Demaegdt,H., Vanderheyden,P., De Backer,J.P., Mosselmans,S., Laeremans,H., Le,M.T., Kersemans,V., Michotte,Y. and Vauquelin,G.
    Endogenous cystinyl aminopeptidase in Chinese hamster ovary cells: characterization by [125I]Ang IV binding and catalytic activity
    Biochem Pharmacol68, 885-892. PubMed  Europe PubMed DOI  I
  25. 2003
  26. Lew,R.A., Mustafa,T., Ye,S., McDowall,S.G., Chai,S.Y. and Albiston,A.L.
    Angiotensin AT4 ligands are potent, competitive inhibitors of insulin regulated aminopeptidase (IRAP)
    J Neurochem86, 344-350. PubMed  Europe PubMed DOI  I
  27. 2001
  28. [YEAR:28-12-2001]Albiston,A.L., McDowall,S.G., Matsacos,D., Sim,P., Clune,E., Mustafa,T., Lee,J., Mendelsohn,F.A., Simpson,R.J., Connolly,L.M. and Chai,S.Y.
    Evidence that the angiotensin IV (AT(4)) receptor is the enzyme insulin-regulated aminopeptidase
    J Biol Chem276, 48623-48626. PubMed  Europe PubMed DOI  I