Literature for semagacestat (A22.001 inhibitor)

Summary Literature

(Topics flags: I Inhibitor. To select only the references relevant to a single topic, click the link above. See explanation.)

    2017
  1. Tagami,S., Yanagida,K., Kodama,T.S., Takami,M., Mizuta,N., Oyama,H., Nishitomi,K., Chiu,Y.W., Okamoto,T., Ikeuchi,T., Sakaguchi,G., Kudo,T., Matsuura,Y., Fukumori,A., Takeda,M., Ihara,Y. and Okochi,M.
    Semagacestat is a pseudo-inhibitor of gamma-secretase
    Cell Rep21, 259-273. PubMed  Europe PubMed DOI  I
  2. 2015
  3. De Strooper,B. and Chavez Gutierrez,L.
    Learning by failing: ideas and concepts to tackle gamma-secretases in Alzheimer's disease and beyond
    Annu Rev Pharmacol Toxicol55, 419-437. PubMed  Europe PubMed DOI  I
  4. 2014
  5. De Strooper,B.
    Lessons from a failed gamma-secretase Alzheimer trial
    Cell159, 721-726. PubMed  Europe PubMed DOI  I
  6. 2011
  7. Imbimbo,B.P., Panza,F., Frisardi,V., Solfrizzi,V., D'Onofrio,G., Logroscino,G., Seripa,D. and Pilotto,A.
    Therapeutic intervention for Alzheimer's disease with gamma-secretase inhibitors: still a viable option?
    Expert Opin Investig Drugs20, 325-341. PubMed  Europe PubMed DOI  I
  8. 2010
  9. Ross,J.S. and Imbimbo,B.P.
    Are gamma-secretase inhibitors detrimental for Alzheimer's disease patients?
    J Alzheimers Dis22, 401-404. PubMed  Europe PubMed DOI  I
  10. 2008
  11. Imbimbo,B.P.
    Alzheimer's disease: gamma-secretase inhibitors
    Drug Discov Today Ther Strateg5, 169-175. DOI  I
  12. 2006
  13. [YEAR:11-8-2006]Clarke,E.E., Churcher,I., Ellis,S., Wrigley,J.D., Lewis,H.D., Harrison,T., Shearman,M.S. and Beher,D.
    Intra- or intercomplex binding to the gamma-secretase enzyme. A model to differentiate inhibitor classes
    J Biol Chem281, 31279-31289. PubMed  Europe PubMed DOI  I
  14. [YEAR:28-2-2006]Siemers,E.R., Quinn,J.F., Kaye,J., Farlow,M.R., Porsteinsson,A., Tariot,P., Zoulnouni,P., Galvin,J.E., Holtzman,D.M., Knopman,D.S., Satterwhite,J., Gonzales,C., Dean,R.A. and May,P.C.
    Effects of a gamma-secretase inhibitor in a randomized study of patients with Alzheimer disease
    Neurology66, 602-604. PubMed  Europe PubMed DOI  I