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Literature for actinonin (M01.001 inhibitor)

Summary Structure Literature

(Topics flags: S Structure, A Assay, I Inhibitor. To select only the references relevant to a single topic, click the link above. See explanation.)

    2019
  1. Chepurnova Dcapital A,C., Samoilova capital IE,C., Verin capital A,C., Fesenko,A.G., Anisimov capital A,C.A.C. and Korotaeva,A.A.
    Inhibition of meprins reduces pulmonary edema in LPS-induced acute lung damage
    Bull Exp Biol Med (2019) 166, 719-721. PubMed  Europe PubMed DOI  I
    2. 2018
  2. Kim,B., Lee,H.J., Im,N.R., Lee,D.Y., Kang,C.Y., Park,I.H., Lee,S.H., Lee,S.H., Baek,S.K. and Kim,T.H.
    Effect of matrix metalloproteinase inhibitor on disrupted E-cadherin after acid exposure in the human nasal epithelium
    Laryngoscope (2018) 128, E1-E1. PubMed  Europe PubMed DOI  I
  3. Schulze,A., Wermann,M., Demuth,H.U., Yoshimoto,T., Ramsbeck,D., Schlenzig,D. and Schilling,S.
    Continuous assays for meprin alpha and beta using prolyl tripeptidyl aminopeptidase (PtP) from Porphyromonas gingivalis
    Anal Biochem (2018) 559, 11-16. PubMed  Europe PubMed DOI  A  I
    4. 2017
  4. Leipoldt,F., Santos-Aberturas,J., Stegmann,D.P., Wolf,F., Kulik,A., Lacret,R., Popadic,D., Keinhorster,D., Kirchner,N., Bekiesch,P., Gross,H., Truman,A.W. and Kaysser,L.
    Warhead biosynthesis and the origin of structural diversity in hydroxamate metalloproteinase inhibitors
    Nat Commun (2017) 8, 1965-1965. PubMed  Europe PubMed DOI  PMC  EPMC  I
    5. 2015
  5. Ganji,R.J., Reddi,R., Gumpena,R., Marapaka,A.K., Arya,T., Sankoju,P., Bhukya,S. and Addlagatta,A.
    Structural basis for the inhibition of M1 family aminopeptidases by the natural product actinonin: crystal structure in complex with E. coli aminopeptidase N
    Protein Sci (2015) 24, 823-831. PubMed  Europe PubMed DOI  S  I
    6. 2011
  6. Addison,M.L., Minnion,J.S., Shillito,J.C., Suzuki,K., Tan,T.M., Field,B.C., Germain-Zito,N., Becker-Pauly,C., Ghatei,M.A., Bloom,S.R. and Murphy,K.G.
    A role for metalloendopeptidases in the breakdown of the gut hormone, PYY3-36
    Endocrinology (2011) 152, 4630-4640. PubMed  Europe PubMed DOI  I
  7. Sina,A., Lord-Dufour,S., Roy,R. and Annabi,B.
    Pharmacological targeting of MT1-MMP by actinonin in brain tumours
    Bio Trib Mag (2011) 38, 39-45. DOI  I
  8. Wang,Z., Herzog,C., Kaushal,G.P., Gokden,N. and Mayeux,P.R.
    Actinonin, a meprin a inhibitor, protects the renal microcirculation during sepsis
    Shock (2011) 35, 141-147. PubMed  Europe PubMed DOI  I
    9. 2009
  9. Gao,P., Guo,R.W., Chen,J.F., Chen,Y., Wang,H., Yu,Y. and Huang,L.
    A meprin inhibitor suppresses atherosclerotic plaque formation in ApoE-/- mice
    Atherosclerosis (2009) 207, 84-92. PubMed  Europe PubMed DOI  I
  10. Sina,A., Lord-Dufour,S. and Annabi,B.
    Cell-based evidence for aminopeptidase N/CD13 inhibitor actinonin targeting of MT1-MMP-mediated proMMP-2 activation
    Cancer Lett (2009) 279, 171-176. PubMed  Europe PubMed DOI  I
    11. 2008
  11. Takayama,J., Takaoka,M., Yamamoto,S., Nohara,A., Ohkita,M. and Matsumura,Y.
    Actinonin, a meprin inhibitor, protects ischemic acute kidney injury in male but not in female rats
    Eur J Pharmacol (2008) 581, 157-163. PubMed  Europe PubMed DOI  I
    12. 2005
  12. Matters,G.L., Manni,A. and Bond,J.S.
    Inhibitors of polyamine biosynthesis decrease the expression of the metalloproteases meprin alpha and MMP-7 in hormone-independent human breast cancer cells
    Clin Exp Metastasis (2005) 22, 331-339. PubMed  Europe PubMed DOI  I
    13. 2002
  13. [YEAR:26-7-2002]Guilloteau,J.P., Mathieu,M., Giglione,C., Blanc,V., Dupuy,A., Chevrier,M., Gil,P., Famechon,A., Meinnel,T. and Mikol,V.
    The crystal structures of four peptide deformylases bound to the antibiotic actinonin reveal two distinct types: a platform for the structure-based design of antibacterial agents
    J Mol Biol (26-7-2002) 320, 951-962. PubMed  Europe PubMed DOI  S  I
    14. 2000
  14. [YEAR:15-2-2000]Chen,D.Z., Patel,D.V., Hackbarth,C.J., Wang,W., Dreyer,G., Young,D.C., Margolis,P.S., Wu,C., Ni,Z.J., Trias,J., White,R.J. and Yuan,Z.
    Actinonin, a naturally occurring antibacterial agent, is a potent deformylase inhibitor
    Biochemistry (15-2-2000) 39, 1256-1262. PubMed  Europe PubMed DOI  I
  15. Matsuda,Y., Katayama,M., Hara,I., Sato,H., Tomomasa,H., Iizumi,T., Umeda,T. and Ishikawa,H.
    Inhibitors on an elastase-like enzyme activity catalyzing Suc-Ala-Ala-Pro-Leu-pNA amidolysis in human seminal plasma
    Syst Biology Reprod Med (2000) 44, 1-9. DOI  I
    16. 1994
  16. Wolz,R.L.
    A kinetic comparison of the homologous proteases astacin and meprin A
    Arch Biochem Biophys (1994) 310, 144-151. PubMed  Europe PubMed DOI  I
    17. 1992
  17. [YEAR:3-11-1992]Tieku,S. and Hooper,N.M.
    Inhibition of aminopeptidases N, A and W. A re-evaluation of the actions of bestatin and inhibitors of angiotensin converting enzyme
    Biochem Pharmacol (3-11-1992) 44, 1725-1730. PubMed  Europe PubMed DOI  I
    18. 1985
  18. Umezawa,H., Aoyagi,T., Tanaka,T., Suda,H., Okuyama,A., Naganawa,H., Hamada,M. and Takeuchi,T.
    Production of actinonin, an inhibitor of aminopeptidase M, by actinomycetes
    J Antibiot (Tokyo) (1985) 38, 1629-1630. PubMed  Europe PubMed  I
    19. 1975
  19. Anderson,N.H., Ollis,W.D., Thorpe,J.E. and Ward,A.D.
    Studies concerning the antibiotic actinonin. Part II. Total synthesis of actinonin and some structural analogues by the isomaleimide method
    J Chem Soc [Perkin 1] (1975) , 825-830. PubMed  Europe PubMed  I
  20. Broughton,B.J., Chaplen,P., Freeman,W.A., Warren,P.J., Wooldridge,K.R. and Wright,D.E.
    Studies concerning the antibiotic actinonin. Part VIII. Structure-activity relationships in the actinonin series
    J Chem Soc [Perkin 1] (1975) 1975, 857-860. PubMed  Europe PubMed  I
  21. Devlin,J.P., Ollis,W.D. and Thorpe,J.E.
    Studies concerning the antibiotic actinon. Part V. Synthesis of structural analogues of actinonin by the anhydride-ester method
    J Chem Soc [Perkin 1] (1975) 1975, 846-848. PubMed  Europe PubMed  I
  22. Gordon,J.J., Devlin,J.P., East,A.J., Ollis,W.D., Wright,D.E. and Ninet,L.
    Studies concerning the antibiotic actinonin. Part I. The constitution of actinonin. A natural hydroxamic acid with antibiotic activity
    J Chem Soc [Perkin 1] (1975) 1975, 819-825. PubMed  Europe PubMed  I
    23. 1969
  23. Attwood,M.M.
    An investigation into the mode of action of actinonin
    J Gen Microbiol (1969) 55, 209-216. PubMed  Europe PubMed  I
    24. 1962
  24. [YEAR:18-8-1962]Gordon,J.J., Kelly,B.K. and Miller,G.A.
    Actinonin: an antibiotic substance produced by an actinomycete
    Nature (18-8-1962) 195, 701-702. PubMed  Europe PubMed DOI  I

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