Literature for RXPA380 (M02.004 inhibitor)

Summary Structure Literature

(Topics flags: S Structure, I Inhibitor. To select only the references relevant to a single topic, click the link above. See explanation.)

    2012
  1. Anthony,C.S., Masuyer,G., Sturrock,E.D. and Acharya,K.R.
    Structure based drug design of angiotensin-I converting enzyme inhibitors
    Curr Med Chem19, 845-855. PubMed  Europe PubMed DOI  I
  2. 2011
  3. Akif,M., Schwager,S.L., Anthony,C.S., Czarny,B., Beau,F., Dive,V., Sturrock,E.D. and Acharya,K.R.
    Novel mechanism of inhibition of human angiotensin-I-converting enzyme (ACE) by a highly specific phosphinic tripeptide
    Biochem J436, 53-59. PubMed  Europe PubMed DOI  S  I
  4. 2009
  5. Kroger,W.L., Douglas,R.G., O'Neill,H.G., Dive,V. and Sturrock,E.D.
    Investigating the domain specificity of phosphinic inhibitors RXPA380 and RXP407 in angiotensin-converting enzyme
    Biochemistry48, 8405-8412. PubMed  Europe PubMed DOI  I
  6. 2007
  7. Corradi,H.R., Chitapi,I., Sewell,B.T., Georgiadis,D., Dive,V., Sturrock,E.D. and Acharya,K.R.
    The structure of testis angiotensin-converting enzyme in complex with the C domain-specific inhibitor RXPA380
    Biochemistry46, 5473-5478. PubMed  Europe PubMed DOI  S  I
  8. 2004
  9. Georgiadis,D., Cuniasse,P., Cotton,J., Yiotakis,A. and Dive,V.
    Structural determinants of RXPA380, a potent and highly selective inhibitor of the angiotensin-converting enzyme C-domain
    Biochemistry43, 8048-8054. PubMed  Europe PubMed DOI  I