Literature for amastatin (M28.002 inhibitor)

Summary Structure Literature

(Topics flags: S Structure, I Inhibitor, V Review. To select only the references relevant to a single topic, click the link above. See explanation.)

    2017
  1. Nakamura,T., Yamazato,M., Ishida,A. and Ohya,Y.
    Excess of aminopeptidase A in the brain elevates blood pressure via the angiotensin II type 1 and bradykinin B2 receptors without dipsogenic effect
    Int J Hypertens (2017) 2017, 3967595-3967595. PubMed  Europe PubMed DOI  PMC  EPMC  I
  2. 2014
  3. Murata,T., Yoshikawa,M., Watanabe,M., Takahashi,S., Kawaguchi,M., Kobayashi,H. and Suzuki,T.
    Potentiation of [Met5]enkephalin-induced antinociception by mixture of three peptidase inhibitors in rat
    J Anesth (2014) 28, 708-715. PubMed  Europe PubMed DOI  I
  4. 2013
  5. Yang,Y., Liu,C., Lin,Y.L. and Li,F.
    Structural insights into central hypertension regulation by human aminopeptidase A
    J Biol Chem (2013) 288, 25638-25645. PubMed  Europe PubMed DOI  S  I
  6. 2012
  7. Wong,A.H., Zhou,D. and Rini,J.M.
    The X-ray crystal structure of human aminopeptidase N reveals a novel dimer and the basis for peptide processing
    J Biol Chem (2012) 287, 36804-36813. PubMed  Europe PubMed DOI  S  I
  8. 2000
  9. Matsuda,Y., Katayama,M., Hara,I., Sato,H., Tomomasa,H., Iizumi,T., Umeda,T. and Ishikawa,H.
    Inhibitors on an elastase-like enzyme activity catalyzing Suc-Ala-Ala-Pro-Leu-pNA amidolysis in human seminal plasma
    Syst Biology Reprod Med (2000) 44, 1-9. DOI  I
  10. 1993
  11. Kim,H. and Lipscomb,W.N.
    X-ray crystallographic determination of the structure of bovine lens leucine aminopeptidase complexed with amastatin: formulation of a catalytic mechanism featuring a gem-diolate transition state
    Biochemistry (1993) 32, 8465-8478. PubMed  Europe PubMed  S  I
  12. 1991
  13. Nagata,Y., Mizutani,S., Nomura,S., Kurauchi,O., Kasugai,M. and Tomoda,Y.
    Purification and properties of human placental aminopeptidase B
    Enzyme (1991) 45, 165-173. PubMed  Europe PubMed  I
  14. 1986
  15. Powers,J.C. and Harper,J.W.
    Inhibitors of metalloproteases
    (1986) , 219-298.  V  I
  16. 1985
  17. [YEAR:25-10-1985]Wilkes,S.H. and Prescott,J.M.
    The slow, tight binding of bestatin and amastatin to aminopeptidases
    J Biol Chem (25-10-1985) 260, 13154-13162. PubMed  Europe PubMed  I
  18. 1984
  19. Rich,D.H., Moon,B.J. and Harbeson,S.
    Inhibition of aminopeptidases by amastatin and bestatin derivatives. Effect of inhibitor structure on slow-binding processes
    J Med Chem (1984) 27, 417-422. PubMed  Europe PubMed  I
  20. 1983
  21. Sakura,H., Kobayashi,H., Mizutani,S., Sakura,N., Hashimoto,T. and Kawashima,Y.
    Kinetic properties of placental aminopeptidase A: N-terminal degradation of angiotensin II
    Biochem Int (1983) 6, 609-615. PubMed  Europe PubMed  I
  22. 1982
  23. Tobe,H., Morishima,H., Aoyagi,T., Umezawa,H., Nakamura,K., Ishiki,K., Yoshioka,T., Shimauchi,Y. and Inui,T.
    Synthesis and structure-activity relationships of amastatin analogues, inhibitors of aminopeptidase A
    Agric Biol Chem (1982) 46, 1865-1872. DOI  I
  24. 1980
  25. Rich,D.H., Moon,B.J. and Boparai,A.S.
    Synthesis of (2S,3R)-3-amino-2-hydroxy-5-methylhexanoic acid derivatives. Application to the synthesis of amastatin, an inhibitor of aminopeptidases
    J Org Chem (1980) 45, 2288-2290.  I
  26. Tobe,H., Kojima,F., Aoyagi,T. and Umezawa,H.
    Purification by affinity chromatography using amastatin and properties of aminopeptidase A from pig kidney
    Biochim Biophys Acta (1980) 613, 459-468. PubMed  Europe PubMed  I
  27. 1979
  28. Tobe,H., Morishima,H., Naganawa,H., Takita,T., Aoyagi,T. and Umezawa,H.
    Structure and chemical synthesis of amastatin
    Agric Biol Chem (1979) 43, 591-596. DOI  I
  29. 1978
  30. Aoyagi,T., Tobe,H., Kojima,F., Hamada,M., Takeuchi,T. and Umezawa,H.
    Amastatin, an inhibitor of aminopeptidase A, produced by actinomycetes
    J Antibiot (Tokyo) (1978) 31, 636-638. PubMed  Europe PubMed  I