Literature for P5091 (C19.016 inhibitor)

(Topics flags: T Target, I Inhibitor. To select only the references relevant to a single topic, click the link above. See explanation.)

2019
1. Peng,Y., Liu,Y., Gao,Y., Yuan,B., Qi,X., Fu,Y., Zhu,Q., Cao,T., Zhang,S., Yin,L. and Li,X.
   USP7 is a novel deubiquitinase sustaining PLK1 protein stability and regulating chromosome alignment in mitosis
   J Exp Clin Cancer Res38, 468-468. PubMed  Europe PubMed DOI  I
2018
2. Srivastava,M., Suri,C., Singh,M., Mathur,R. and Asthana,S.
   Molecular dynamics simulation reveals the possible druggable hot-spots of USP7
   Oncotarget9, 34289-34305. PubMed  Europe PubMed DOI  I
2017
3. Ali,A., Raja,R., Farooqui,S.R., Ahmad,S. and Banerjea,A.C.
   USP7 deubiquitinase controls HIV-1 production by stabilizing Tat protein
   Biochem J474, 1653-1668. PubMed  Europe PubMed DOI  I
4. Chen,C., Song,J., Wang,J., Xu,C., Chen,C., Gu,W., Sun,H. and Wen,X.
   Synthesis and biological evaluation of thiazole derivatives as novel USP7 inhibitors
   Bioorg Med Chem Lett27, 845-849. PubMed  Europe PubMed DOI  I
5. Wang,F., Wang,L., Wu,J., Sokirniy,I., Nguyen,P., Bregnard,T., Weinstock,J., Mattern,M., Bezsonova,I., Hancock,W.W. and Kumar,S.
   Active site-targeted covalent irreversible inhibitors of USP7 impair the functions of Foxp3+ T-regulatory cells by promoting ubiquitination of Tip60
   PLoS ONE12, e0189744-e0189744. PubMed  Europe PubMed DOI  I
2016
6. Lee,G., Oh,T.I., Um,K.B., Yoon,H., Son,J., Kim,B.M., Kim,H.I., Kim,H., Kim,Y.J., Lee,C.S. and Lim,J.H.
   Small-molecule inhibitors of USP7 induce apoptosis through oxidative and endoplasmic reticulum stress in cancer cells
   Biochem Biophys Res Commun470, 181-186. PubMed  Europe PubMed DOI  I
7. Wang,L., Kumar,S., Dahiya,S., Wang,F., Wu,J., Newick,K., Han,R., Samanta,A., Beier,U.H., Akimova,T., Bhatti,T.R., Nicholson,B., Kodrasov,M.P., Agarwal,S., Sterner,D.E., Gu,W., Weinstock,J., Butt,T.R., Albelda,S.M. and Hancock,W.W.
   Ubiquitin-specific protease-7 inhibition impairs Tip60-dependent Foxp3+ T-regulatory cell function and promotes antitumor immunity
   EBioMedicine13, 99-112. PubMed  Europe PubMed DOI  I
2012
8. Chauhan,D., Tian,Z., Nicholson,B., Kumar,K.G., Zhou,B., Carrasco,R., McDermott,J.L., Leach,C.A., Fulcinniti,M., Kodrasov,M.P., Weinstock,J., Kingsbury,W.D., Hideshima,T., Shah,P.K., Minvielle,S., Altun,M., Kessler,B.M., Orlowski,R., Richardson,P., Munshi,N. and Anderson,K.C.
   A small molecule inhibitor of ubiquitin-specific protease-7 induces apoptosis in multiple myeloma cells and overcomes bortezomib resistance
   Cancer Cell22, 345-358. PubMed  Europe PubMed DOI  I
9. Weinstock,J., Wu,J., Cao,P., Kingsbury,W.D., McDermott,J.L., Kodrasov,M.P., McKelvey,D.M., Suresh Kumar,K.G., Goldenberg,S.J., Mattern,M.R. and Nicholson,B.
   Selective dual inhibitors of the cancer-related deubiquitylating proteases USP7 and USP47
   ACS Med Chem Lett3, 789-792. PubMed  Europe PubMed DOI  I
2011
10. Nicholson,B. and Suresh Kumar,K.G.
    The multifaceted roles of USP7: new therapeutic opportunities
    Cell Biochem Biophys60, 61-68. PubMed  Europe PubMed DOI  T  I