Literature for DSR-12727 (S09.003 inhibitor)

Summary Literature

(Topics flags: I Inhibitor. To select only the references relevant to a single topic, click the link above. See explanation.)

    2011
  1. Nishio,Y., Kimura,H., Sawada,N., Sugaru,E., Horiguchi,M., Ono,M., Furuta,Y., Sakai,M., Masui,Y., Otani,M., Hashizuka,T., Honda,Y., Deguchi,J., Nakagawa,T. and Nakahira,H.
    2-({6-[(3R)-3-amino-3-methylpiperidine-1-yl]-1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydro-5H-pyrrolo[3,2-d]pyrimidine-5-yl}methyl)-4-fluorobenzonitrile (DSR-12727): A potent, orally active dipeptidyl peptidase IV inhibitor without mechanism-based inactivation of CYP3A
    Bioorg Med Chem (2011) 19, 5490-5499. PubMed  Europe PubMed DOI  I