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Literature for inhibitor I52.001: tick anticoagulant peptide (Ornithodorus sp.)

Summary Alignment Sequences Sequence features Distribution Structure Literature Inhibits

(Topics flags: S Structure. To select only the references relevant to a single topic, click the link above. See explanation.)

    2024
  1. De Filippis,V., Acquasaliente,L., Pierangelini,A. and Marin,O.
    Chemical Synthesis and Structure-Activity Relationship Studies of the Coagulation Factor Xa Inhibitor Tick Anticoagulant Peptide from the Hematophagous Parasite Ornithodoros moubata
    Biomimetics (Basel) (2024) 9 PubMed  Europe PubMed DOI  PMC  EPMC
    2. 2011
  2. Chang,J.Y.
    Distinct folding pathways of two homologous disulfide proteins: bovine pancreatic trypsin inhibitor and tick anticoagulant peptide
    Antioxid Redox Signal (2011) 14, 127-135. PubMed  Europe PubMed DOI
    3. 2004
  3. [YEAR:30-3-2004]Rezaie,A.R.
    Kinetics of factor Xa inhibition by recombinant tick anticoagulant peptide: both active site and exosite interactions are required for a slow- and tight-binding inhibition mechanism
    Biochemistry (30-3-2004) 43, 3368-3375. PubMed  Europe PubMed DOI
    4. 2000
  4. Chang,J.Y. and Ballatore,A.
    Structure and heterogeneity of the one- and two-disulfide folding intermediates of tick anticoagulant peptide
    J Protein Chem (2000) 19, 299-310. PubMed  Europe PubMed DOI
  5. St Charles,R., Padmanabhan,K., Arni,R.V., Padmanabhan,K.P. and Tulinsky,A.
    Structure of tick anticoagulant peptide at 1.6 A resolution complexed with bovine pancreatic trypsin inhibitor
    Protein Sci (2000) 9, 265-272. PubMed  Europe PubMed DOI  PMC  EPMC  S
    6. 1999
  6. Wei,A., Smallwood,A., Alexander,R.S., Duke,J., Ross,H., Rosenfeld,S.A. and Chang,C.H.
    Crystallization and preliminary X-ray diffraction data of the complex of recombinant tick anticoagulant peptide (rTAP) and bovine factor Xa
    Acta Crystallogr D Biol Crystallogr (1999) 55, 862-864. PubMed  Europe PubMed DOI
    7. 1998
  7. Cook,J.C., Schultz,L.D., Huang,J., George,H.A., Herber,W.K., Ip,C., Joyce,J.G., Mao,S.S., Markus,H.Z., Miller,W.J., Sardana,M.K. and Lehman,E.D.
    Expression and purification of recombinant tick anticoagulant peptide (Y1W/D10R) double mutant secreted by Saccharomyces cerevisiae
    Protein Expr Purif (1998) 13, 291-300. PubMed  Europe PubMed DOI
  8. Joubert,A.M., Louw,A.I., Joubert,F. and Neitz,A.W.
    Cloning, nucleotide sequence and expression of the gene encoding factor Xa inhibitor from the salivary glands of the tick, Ornithodoros savignyi
    Exp Appl Acarol (1998) 22, 603-619. PubMed  Europe PubMed DOI
  9. Wei,A., Alexander,R.S., Duke,J., Ross,H., Rosenfeld,S.A. and Chang,C.H.
    Unexpected binding mode of tick anticoagulant peptide complexed to bovine factor Xa
    J Mol Biol (1998) 283, 147-154. PubMed  Europe PubMed DOI  S
    10. 1997
  10. [YEAR:7-1-1997]Betz,A., Vlasuk,G.P., Bergum,P.W. and Krishnaswamy,S.
    Selective inhibition of the prothrombinase complex: factor Va alters macromolecular recognition of a tick anticoagulant peptide mutant by factor Xa
    Biochemistry (7-1-1997) 36, 181-191. PubMed  Europe PubMed DOI
  11. [YEAR:3-1-1997]Chang,J.Y.
    A two-stage mechanism for the reductive unfolding of disulfide-containing proteins
    J Biol Chem (3-1-1997) 272, 69-75. PubMed  Europe PubMed
    12. 1996
  12. [YEAR:10-9-1996]Chang,J.Y.
    The disulfide folding pathway of tick anticoagulant peptide (TAP), a Kunitz-type inhibitor structurally homologous to BPTI
    Biochemistry (10-9-1996) 35, 11702-11709. PubMed  Europe PubMed DOI
  13. Gaspar,A.R., Joubert,A.M., Crause,J.C. and Neitz,A.W.
    Isolation and characterization of an anticoagulant from the salivary glands of the tick, Ornithodoros savignyi (Acari: Argasidae)
    Exp Appl Acarol (1996) 20, 583-598. PubMed  Europe PubMed
  14. [YEAR:15-11-1996]van de Locht,A., Stubbs,M.T., Bode,W., Friedrich,T., Bollschweiler,C., Hoffken,W. and Huber,R.
    The ornithodorin-thrombin crystal structure, a key to the TAP enigma?
    EMBO J (15-11-1996) 15, 6011-6017. PubMed  Europe PubMed  PMC  EPMC  S
    15. 1995
  15. Lim-Wilby,M.S., Hallenga,K., De Maeyer,M., Lasters,I., Vlasuk,G.P. and Brunck,T.K.
    NMR structure determination of tick anticoagulant peptide (TAP)
    Protein Sci (1995) 4, 178-186. PubMed  Europe PubMed DOI  PMC  EPMC  S
  16. [YEAR:18-4-1995]Mao,S.S., Huang,J., Welebob,C., Neeper,M.P., Garsky,V.M. and Shafer,J.A.
    Identification and characterization of variants of tick anticoagulant peptide with increased inhibitory potency toward human factor Xa
    Biochemistry (18-4-1995) 34, 5098-5103. PubMed  Europe PubMed
  17. [YEAR:18-5-1995]Sanyal,G., Marquis-Omer,D., Waxman,L., Mach,H., Ryan,J.A., O'Brien Gress,J. and Middaugh,C.R.
    Spectroscopic characterization of tick anticoagulant peptide
    Biochim Biophys Acta (18-5-1995) 1249, 100-108. PubMed  Europe PubMed DOI
    18. 1994
  18. [YEAR:26-9-1994]Antuch,W., Guntert,P., Billeter,M., Hawthorne,T., Grossenbacher,H. and Wuthrich,K.
    NMR solution structure of the recombinant tick anticoagulant protein (rTAP), a factor Xa inhibitor from the tick Ornithodoros moubata
    FEBS Lett (26-9-1994) 352, 251-257. PubMed  Europe PubMed DOI  S
    19. 1993
  19. Lehman,E.D., Joyce,J.G., Freymeyer,D.K., Bailey,F.J., Herber,W.K. and Miller,W.J.
    A novel process for the large-scale purification of recombinant tick anticoagulant peptide using perfusion chromatography
    Biotechnology (N Y) (1993) 11, 207-212. PubMed  Europe PubMed DOI
  20. [YEAR:1-7-1993]Vlasuk,G.P.
    Structural and functional characterization of tick anticoagulant peptide (TAP): a potent and selective inhibitor of blood coagulation factor Xa
    Thromb Haemost (1-7-1993) 70, 212-216. PubMed  Europe PubMed
    21. 1992
  21. [YEAR:8-12-1992]Dunwiddie,C.T., Neeper,M.P., Nutt,E.M., Waxman,L., Smith,D.E., Hofmann,K.J., Lumma,P.K., Garsky,V.M. and Vlasuk,G.P.
    Site-directed analysis of the functional domains in the factor Xa inhibitor tick anticoagulant peptide: identification of two distinct regions that constitute the enzyme recognition sites
    Biochemistry (8-12-1992) 31, 12126-12131. PubMed  Europe PubMed DOI
  22. [YEAR:16-6-1992]Jordan,S.P., Mao,S.S., Lewis,S.D. and Shafer,J.A.
    Reaction pathway for inhibition of blood coagulation factor Xa by tick anticoagulant peptide
    Biochemistry (16-6-1992) 31, 5374-5380. PubMed  Europe PubMed DOI
  23. [YEAR:14-2-1992]Lehman,E.D., Schaefer,T.F., Przysiecki,C.T., Joyce,J.G., Bailey,F.J., Schulman,C.A., Burke,C.J., Ramjit,H.G. and Miller,W.J.
    Large-scale purification and characterization of recombinant tick anticoagulant peptide
    J Chromatogr (14-2-1992) 574, 225-235. PubMed  Europe PubMed DOI
    24. 1991
  24. [YEAR:25-7-1991]Sardana,M., Sardana,V., Rodkey,J., Wood,T., Ng,A., Vlasuk,G.P. and Waxman,L.
    Determination of disulfide bond pairs and stability in recombinant tick anticoagulant peptide
    J Biol Chem (25-7-1991) 266, 13560-13563. PubMed  Europe PubMed
  25. [YEAR:4-3-1991]Vlasuk,G.P., Ramjit,D., Fujita,T., Dunwiddie,C.T., Nutt,E.M., Smith,D.E. and Shebuski,R.J.
    Comparison of the in vivo anticoagulant properties of standard heparin and the highly selective factor Xa inhibitors antistasin and tick anticoagulant peptide (TAP) in a rabbit model of venous thrombosis
    Thromb Haemost (4-3-1991) 65, 257-262. PubMed  Europe PubMed
    26. 1990
  26. [YEAR:18-12-1990]Jordan,S.P., Waxman,L., Smith,D.E. and Vlasuk,G.P.
    Tick anticoagulant peptide: kinetic analysis of the recombinant inhibitor with blood coagulation factor Xa
    Biochemistry (18-12-1990) 29, 11095-11100. PubMed  Europe PubMed DOI
  27. [YEAR:15-10-1990]Neeper,M.P., Waxman,L., Smith,D.E., Schulman,C.A., Sardana,M., Ellis,R.W., Schaffer,L.W., Siegl,P.K. and Vlasuk,G.P.
    Characterization of recombinant tick anticoagulant peptide. A highly selective inhibitor of blood coagulation factor Xa
    J Biol Chem (15-10-1990) 265, 17746-17752. PubMed  Europe PubMed
  28. [YEAR:4-5-1990]Waxman,L., Smith,D.E., Arcuri,K.E. and Vlasuk,G.P.
    Tick anticoagulant peptide (TAP) is a novel inhibitor of blood coagulation factor Xa
    Science (4-5-1990) 248, 593-596. PubMed  Europe PubMed

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