EMBL-EBI | Chemical Biology | ChEBI
Example searches: iron*, InChI=1S/CH4O/c1-2/h2H,1H3, caffeine | Advanced Search
| ChEBI ID | CHEBI:131770 |
| ChEBI Name | EC 3.6.3.49 (channel-conductance-controlling ATPase) inhibitor |
| Stars | |
| Definition | A EC 3.6.3.* (acid anhydride hydrolase catalysing transmembrane movement of substances) inhibitor that interferes with the action of channel-conductance-controlling ATPase (EC 3.6.3.49, also known as cystic fibrosis conductance regulator, CFCR). |
| Secondary ChEBI ID | CHEBI:131771 |
| Last Modified | 19 April 2016 |
| Submitter | Gareth Owen |
| Wikipedia |
|---|
| ChEBI Ontology |
|---|
| Outgoing Relation(s) |
| EC 3.6.3.49 (channel-conductance-controlling ATPase) inhibitor (CHEBI:131770) is a EC 3.6.3.* (acid anhydride hydrolase catalysing transmembrane movement of substances) inhibitor (CHEBI:76895) |
| Incoming Relation(s) |
| bumetanide (CHEBI:3213) has role EC 3.6.3.49 (channel-conductance-controlling ATPase) inhibitor (CHEBI:131770) |
| CFTRinh-172 (CHEBI:131686) has role EC 3.6.3.49 (channel-conductance-controlling ATPase) inhibitor (CHEBI:131770) |
| glyburide (CHEBI:5441) has role EC 3.6.3.49 (channel-conductance-controlling ATPase) inhibitor (CHEBI:131770) |
| Synonyms | Source |
|---|---|
| CFTR inhibitors | ChEBI |
| cystic fibrosis transmembrane conductance regulator inhibitor | ChEBI |
| cystic fibrosis transmembrane conductance regulator inhibitors | ChEBI |
| channel-conductance-controlling ATPase (EC 3.6.3.49) inhibitors | ChEBI |
| CFTR inhibitor | ChEBI |
| cystic fibrosis conductance regulator inhibitors | ChEBI |
| Manual Xrefs | Databases |
|---|---|
| Cystic_fibrosis_transmembrane_conductance_regulator | Wikipedia |