Structure analysis

Crystal structure of ENL (MLLT1) in complex with compound 12

X-ray diffraction
2Å resolution
Source organism: Homo sapiens
Assembly composition:
monomeric (preferred)
Entry contents: 1 distinct polypeptide molecule

Assemblies

Assembly 1 (preferred)
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Multimeric state: monomeric
Accessible surface area: 8425.89 Å2
Buried surface area: 746.1 Å2
Dissociation area: 109.68 Å2
Dissociation energy (ΔGdiss): -1.81 kcal/mol
Dissociation entropy (TΔSdiss): -0.3 kcal/mol
Symmetry number: 1
PDBe Complex ID: PDB-CPX-169829

Macromolecules

Chain: A
Length: 155 amino acids
Theoretical weight: 18.31 KDa
Source organism: Homo sapiens
Expression system: Escherichia coli BL21(DE3)
UniProt:
  • Canonical: Q03111 (Residues: 1-148; Coverage: 27%)
Gene names: ENL, LTG19, MLLT1, YEATS1
Pfam: YEATS family
InterPro:
CATH: YEATS domain

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