4pkl

X-ray diffraction
1.25Å resolution

Bromodomain of Trypanosoma brucei BDF2 With IBET-151

Released:

Function and Biology Details

Biochemical function:
  • not assigned
Biological process:
  • not assigned
Cellular component:
  • not assigned

Structure analysis Details

Assembly composition:
monomeric (preferred)
PDBe Complex ID:
PDB-CPX-174390 (preferred)
Entry contents:
1 distinct polypeptide molecule
Macromolecule:
Bromo domain-containing protein Chains: A, B
Molecule details ›
Chains: A, B
Length: 119 amino acids
Theoretical weight: 13.5 KDa
Source organism: Trypanosoma brucei brucei TREU927
Expression system: Escherichia coli
UniProt:
  • Canonical: Q38AM1 (Residues: 9-123; Coverage: 51%)
Gene name: Tb10.6k15.3240
Sequence domains: Bromodomain
Structure domains: Bromodomain-like

Ligands and Environments

No modified residues

Experiments and Validation Details

Entry percentile scores
X-ray source: NSLS BEAMLINE X29A
Spacegroup: P212121
Unit cell:
a: 55.869Å b: 62.091Å c: 62.117Å
α: 90° β: 90° γ: 90°
R-values:
R R work R free
0.17 0.169 0.179
Expression system: Escherichia coli