 |
PDBsum entry 3n1v
|
|
|
|
 |
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
 |
|
|
|
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
 |
|
|
|
|
|
|
|
|
|
|
Transferase/transferase inhibitor
|
PDB id
|
|
|
|
3n1v
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
|
References listed in PDB file
|
 |
|
Key reference
|
 |
|
Title
|
 |
Allosteric non-Bisphosphonate fpps inhibitors identified by fragment-Based discovery.
|
 |
|
Authors
|
 |
W.Jahnke,
J.M.Rondeau,
S.Cotesta,
A.Marzinzik,
X.Pellé,
M.Geiser,
A.Strauss,
M.Götte,
F.Bitsch,
R.Hemmig,
C.Henry,
S.Lehmann,
J.F.Glickman,
T.P.Roddy,
S.J.Stout,
J.R.Green.
|
 |
|
Ref.
|
 |
Nat Chem Biol, 2010,
6,
660-666.
|
 |
|
PubMed id
|
 |
|
 |
 |
|
Abstract
|
 |
|
No abstract given.
|
 |
|
Secondary reference #1
|
 |
|
Title
|
 |
Structural basis for the exceptional in vivo efficacy of bisphosphonate drugs.
|
 |
|
Authors
|
 |
J.M.Rondeau,
F.Bitsch,
E.Bourgier,
M.Geiser,
R.Hemmig,
M.Kroemer,
S.Lehmann,
P.Ramage,
S.Rieffel,
A.Strauss,
J.R.Green,
W.Jahnke.
|
 |
|
Ref.
|
 |
Chemmedchem, 2006,
1,
267-273.
|
 |
|
PubMed id
|
 |
|
 |
 |
|
|
 |
|
|
|
|
 |