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PDBsum entry 3n1v

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Transferase/transferase inhibitor PDB id
3n1v
Contents
Protein chain
343 a.a.
Ligands
3N1 ×2
PO4
Waters ×115

References listed in PDB file
Key reference
Title Allosteric non-Bisphosphonate fpps inhibitors identified by fragment-Based discovery.
Authors W.Jahnke, J.M.Rondeau, S.Cotesta, A.Marzinzik, X.Pellé, M.Geiser, A.Strauss, M.Götte, F.Bitsch, R.Hemmig, C.Henry, S.Lehmann, J.F.Glickman, T.P.Roddy, S.J.Stout, J.R.Green.
Ref. Nat Chem Biol, 2010, 6, 660-666.
PubMed id 20711197
Abstract
No abstract given.
Secondary reference #1
Title Structural basis for the exceptional in vivo efficacy of bisphosphonate drugs.
Authors J.M.Rondeau, F.Bitsch, E.Bourgier, M.Geiser, R.Hemmig, M.Kroemer, S.Lehmann, P.Ramage, S.Rieffel, A.Strauss, J.R.Green, W.Jahnke.
Ref. Chemmedchem, 2006, 1, 267-273.
PubMed id 16892359
Abstract
PROCHECK
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 Headers

 

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