spacer
spacer

PDBsum entry 6tma

Go to PDB code: 
protein ligands metals Protein-protein interface(s) links
Antibiotic PDB id
6tma

 

 

 

 

Loading ...

 
JSmol PyMol  
Contents
Protein chains
231 a.a.
Ligands
_OH ×2
9O8 ×2
Metals
IOD ×2
_ZN ×6
_CL ×4
Waters ×627
PDB id:
6tma
Name: Antibiotic
Title: Vim-2_1dj- triazole inhibitors with promising inhibitor effects against antibiotic resistance metallo-beta-lactamases
Structure: Beta-lactamase class b vim-2. Chain: a, b. Synonym: blavim-2,class b carbapenemase vim-2,metallo beta-lactamase, metallo-beta lactamase protein,metallo-beta-lactamase vim-2,vim-2, vim-2 beta-lactamase,vim-2 class b metallo b-lactamase,vim-2 type metallo-beta-lactamase. Engineered: yes
Source: Pseudomonas aeruginosa. Organism_taxid: 287. Gene: blavim-2, bla vim-2, bla-vim-2, blasvim-2, blavim2, blm, vim- 2, vim-2, paerug_p32_london_17_vim_2_10_11_06255. Expressed in: escherichia coli. Expression_system_taxid: 562
Resolution:
1.50Å     R-factor:   0.158     R-free:   0.194
Authors: H.-K.S.Leiros
Date:
03-Dec-19     Release date:   02-Sep-20    
PROCHECK
Go to PROCHECK summary
 Headers
 References

Protein chains
Q9K2N0  (Q9K2N0_PSEAI) -  beta-lactamase from Pseudomonas aeruginosa
Seq:
Struc:
266 a.a.
232 a.a.
Key:    Secondary structure

 Enzyme reactions 
   Enzyme class: E.C.3.5.2.6  - beta-lactamase.
[IntEnz]   [ExPASy]   [KEGG]   [BRENDA]

      Pathway:
Penicillin Biosynthesis and Metabolism
      Reaction: a beta-lactam + H2O = a substituted beta-amino acid
      Cofactor: Zn(2+)

 

spacer

spacer