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PDBsum entry 5lof

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Apoptosis/inhibitor PDB id
5lof
Contents
Protein chain
514 a.a.
Ligands
GLC-GLC
70R
Waters ×183

References listed in PDB file
Key reference
Title The mcl1 inhibitor s63845 is tolerable and effective in diverse cancer models.
Authors A.Kotschy, Z.Szlavik, J.Murray, J.Davidson, A.L.Maragno, G.Le toumelin-Braizat, M.Chanrion, G.L.Kelly, J.N.Gong, D.M.Moujalled, A.Bruno, M.Csekei, A.Paczal, Z.B.Szabo, S.Sipos, G.Radics, A.Proszenyak, B.Balint, L.Ondi, G.Blasko, A.Robertson, A.Surgenor, P.Dokurno, I.Chen, N.Matassova, J.Smith, C.Pedder, C.Graham, A.Studeny, G.Lysiak-Auvity, A.M.Girard, F.Gravé, D.Segal, C.D.Riffkin, G.Pomilio, L.C.Galbraith, B.J.Aubrey, M.S.Brennan, M.J.Herold, C.Chang, G.Guasconi, N.Cauquil, F.Melchiore, N.Guigal-Stephan, B.Lockhart, F.Colland, J.A.Hickman, A.W.Roberts, D.C.Huang, A.H.Wei, A.Strasser, G.Lessene, O.Geneste.
Ref. Nature, 2016, 538, 477-482. [DOI no: 10.1038/nature19830]
PubMed id 27760111
Abstract
No abstract given.
PROCHECK
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