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PDBsum entry 5k4x

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Oxidoreductase PDB id
5k4x
Contents
Protein chain
330 a.a.
Ligands
6Q9
IMP
Waters ×349

References listed in PDB file
Key reference
Title Essential but not vulnerable: indazole sulfonamides targeting inosine monophosphate dehydrogenase as potential leads against mycobacterium tuberculosis.
Authors Y.Park, A.Pacitto, T.Bayliss, L.A.Cleghorn, Z.Wang, T.Hartman, K.Arora, T.R.Ioerger, J.Sacchettini, M.Rizzi, S.Donini, T.L.Blundell, D.B.Ascher, K.Rhee, A.Breda, N.Zhou, V.Dartois, S.R.Jonnala, L.E.Via, V.Mizrahi, O.Epemolu, L.Stojanovski, F.Simeons, M.Osuna-Cabello, L.Ellis, C.J.Mackenzie, A.R.Smith, S.H.Davis, D.Murugesan, K.I.Buchanan, P.A.Turner, M.Huggett, F.Zuccotto, M.J.Rebollo-Lopez, M.J.Lafuente-Monasterio, O.Sanz, G.S.Diaz, J.Lelièvre, L.Ballell, C.Selenski, M.Axtman, S.Ghidelli-Disse, H.Pflaumer, M.Bösche, G.Drewes, G.M.Freiberg, M.D.Kurnick, M.Srikumaran, D.J.Kempf, S.R.Green, P.C.Ray, K.Read, P.Wyatt, C.E.Barry, H.I.Boshoff.
Ref. Acs Infect Dis, 2017, 3, 18-33. [DOI no: 10.1021/acsinfecdis.6b00103]
PubMed id 27704782
Abstract
No abstract given.
PROCHECK
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 Headers

 

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