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PDBsum entry 5b5t
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Hydrolase/hydrolase inhibitor
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PDB id
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5b5t
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References listed in PDB file
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Key reference
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Title
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Phosphonate-Based irreversible inhibitors of human γ-Glutamyl transpeptidase (ggt). Ggstop is a non-Toxic and highly selective inhibitor with critical electrostatic interaction with an active-Site residue lys562 for enhanced inhibitory activity.
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Authors
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A.Kamiyama,
M.Nakajima,
L.Han,
K.Wada,
M.Mizutani,
Y.Tabuchi,
A.Kojima-Yuasa,
I.Matsui-Yuasa,
H.Suzuki,
K.Fukuyama,
B.Watanabe,
J.Hiratake.
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Ref.
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Bioorg Med Chem Lett, 2016,
24,
5340-5352.
[DOI no: ]
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PubMed id
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Abstract
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No abstract given.
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