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PDBsum entry 3qlh
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Transferase,hydrolase/inhibitor
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PDB id
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3qlh
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References listed in PDB file
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Key reference
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Title
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Synthesis, Activity, And structural analysis of novel α-Hydroxytropolone inhibitors of human immunodeficiency virus reverse transcriptase-Associated ribonuclease h.
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Authors
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S.Chung,
D.M.Himmel,
J.K.Jiang,
K.Wojtak,
J.D.Bauman,
J.W.Rausch,
J.A.Wilson,
J.A.Beutler,
C.J.Thomas,
E.Arnold,
S.F.Le grice.
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Ref.
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J Med Chem, 2011,
54,
4462-4473.
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PubMed id
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Abstract
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No abstract given.
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Secondary reference #1
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Title
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Structure of HIV-1 reverse transcriptase with the inhibitor beta-Thujaplicinol bound at the rnase h active site.
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Authors
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D.M.Himmel,
K.A.Maegley,
T.A.Pauly,
J.D.Bauman,
K.Das,
C.Dharia,
A.D.Clark,
K.Ryan,
M.J.Hickey,
R.A.Love,
S.H.Hughes,
S.Bergqvist,
E.Arnold.
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Ref.
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Structure, 2009,
17,
1625-1635.
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PubMed id
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Secondary reference #2
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Title
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Crystal engineering of HIV-1 reverse transcriptase for structure-Based drug design.
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Authors
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J.D.Bauman,
K.Das,
W.C.Ho,
M.Baweja,
D.M.Himmel,
A.D.Clark,
D.A.Oren,
P.L.Boyer,
S.H.Hughes,
A.J.Shatkin,
E.Arnold.
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Ref.
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Nucleic Acids Res, 2008,
36,
5083-5092.
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PubMed id
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Secondary reference #3
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Title
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Sensitivity of xenotropic murine leukemia virus-Relat retrovirus reverse transcriptase-Associated ribonucul to alpha-Hydroxytropolone inhibitors
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Authors
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S.Chung,
D.M.Himmel,
J jiang,
B.Scarth,
Y.Wang,
J.W.Rauschv.Kewalramani,
E.Arnold,
M gotte,
J.A.Beutler,
C.R.Thomass.F.J.Le grice.
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Ref.
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TO BE PUBLISHED ...
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