5l8j

X-ray diffraction
1.68Å resolution

Aurora-A kinase domain in complex with vNAR-D01 S93R

Released:

Function and Biology Details

Structure analysis Details

Assembly composition:
hetero dimer (preferred)
PDBe Complex ID:
PDB-CPX-127235 (preferred)
Entry contents:
2 distinct polypeptide molecules
Macromolecules (2 distinct):
Aurora kinase A Chain: A
Molecule details ›
Chain: A
Length: 285 amino acids
Theoretical weight: 32.96 KDa
Source organism: Homo sapiens
Expression system: Escherichia coli BL21(DE3)
UniProt:
  • Canonical: O14965 (Residues: 122-403; Coverage: 70%)
Gene names: AIK, AIRK1, ARK1, AURA, AURKA, AYK1, BTAK, IAK1, STK15, STK6
Sequence domains: Protein kinase domain
Structure domains:
Ig-like domain-containing protein Chain: B
Molecule details ›
Chain: B
Length: 117 amino acids
Theoretical weight: 12.84 KDa
Source organism: Orectolobus maculatus
Expression system: Escherichia coli BL21(DE3)
UniProt:
  • Canonical: Q8JJ25 (Residues: 1-108; Coverage: 95%)
Sequence domains: Immunoglobulin V-set domain
Structure domains: Immunoglobulins

Ligands and Environments

3 bound ligands:
1 modified residue:

Experiments and Validation Details

Entry percentile scores
X-ray source: DIAMOND BEAMLINE I04-1
Spacegroup: P21212
Unit cell:
a: 91.23Å b: 111.12Å c: 41.62Å
α: 90° β: 90° γ: 90°
R-values:
R R work R free
0.201 0.199 0.231
Expression system: Escherichia coli BL21(DE3)