Structure analysis

Src kinase in complex with a quinazoline inhibitor

X-ray diffraction
2.2Å resolution
Source organism: Homo sapiens
Assembly composition:
monomeric (preferred)
Entry contents: 1 distinct polypeptide molecule

Assemblies

Assembly 1 (preferred)
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Multimeric state: monomeric
Accessible surface area: 21983.85 Å2
Buried surface area: 909.54 Å2
Dissociation area: 454.77 Å2
Dissociation energy (ΔGdiss): 2.29 kcal/mol
Dissociation entropy (TΔSdiss): 5.63 kcal/mol
Symmetry number: 1
PDBe Complex ID: PDB-CPX-146379

Macromolecules

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