Literature for peptidase S01.236: kallikrein-related peptidase 6

(References are filtered for relevance to Inhibitor. To remove the filter click here. See explanation.)

2020

De Vita,E., Smits,N., van den Hurk,H., Beck,E.M., Hewitt,J., Baillie,G., Russell,E., Pannifer,A., Hamon,V., Morrison,A., McElroy,S.P., Jones,P., Ignatenko,N.A., Gunkel,N. and Miller,A.K.
Synthesis and structure-activity relationships of N-(4-benzamidino)-oxazolidinones: potent and selective inhibitors of kallikrein-related peptidase 6
ChemMedChem15, 79-95. PubMed Europe PubMed DOI I

2018

De Vita,E., Schuler,P., Lovell,S., Lohbeck,J., Kullmann,S., Rabinovich,E., Sananes,A., Hessling,B., Hamon,V., Papo,N., Hess,J., Tate,E.W., Gunkel,N. and Miller,A.K.
Depsipeptides featuring a neutral P1 are potent inhibitors of kallikrein-related peptidase 6 with on-target cellular activity
J Med Chem61, 8859-8874. PubMed Europe PubMed DOI I
Soualmia,F., Bosc,E., Amiri,S.A., Stratmann,D., Magdolen,V., Darmoul,D., Reboud-Ravaux,M. and El Amri,C.
Insights into the activity control of the kallikrein-related peptidase 6: small-molecule modulators and allosterism
Biol Chem399, 1073-1078. PubMed Europe PubMed DOI I

2012

Arnold,S., Pampalakis,G., Kantiotou,K., Silva,D., Cortez,C., Missailidis,S. and Sotiropoulou,G.
One round of SELEX for the generation of DNA aptamers directed against KLK6
Biol Chem393, 343-353. PubMed Europe PubMed DOI I
Liang,G., Chen,X., Aldous,S., Pu,S.F., Mehdi,S., Powers,E., Xia,T. and Wang,R.
Human kallikrein 6 inhibitors with a para-amidobenzylanmine P1 group identified through virtual screening
Bioorg Med Chem Lett22, 2450-2455. PubMed Europe PubMed DOI S I
Liang,G., Chen,X., Aldous,S., Pu,S.F., Mehdi,S., Powers,E., Giovanni,A., Kongsamut,S., Xia,T., Zhang,Y., Wang,R., Gao,Z., Merriman,G., McLean,L.R. and Morize,I.
Virtual screening and X-ray crystallography for human kallikrein 6 inhibitors with an amidinothiophene P1 group
ACS Med Chem Lett3, 159-164. PubMed Europe PubMed DOI S I