Structure-activity relationship data for a series of N-(phenylmehtyl)-2-(1H-pyrazol-4-yl)acetamide and N-(phenylmethyl)2-(4-isoxazolyl) acetamide antagonists of the P2X7 receptor (Supplementary Bioactivity Data for publication CHEMBL1157114)
Supplementary bioactivity data for the GlaxoSmithKline (GSK) publication Bioorg. Med. Chem. Lett. 2010, 20, 3161-3164 (ChEMBL Doc ID: CHEMBL1157114): pIC50 values for 54 compounds that have been tested in the ethidium bromide release assay (ChEMBL Assay ID: CHEMBL1103860) described in reference 24 of the aforementioned publication. All compounds have been tested at least four times and have been reported as being active in all test occasions.