CHEBI:62434 - EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor

Main ChEBI Ontology Automatic Xrefs Reactions Pathways Models
ChEBI Name EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor
ChEBI ID CHEBI:62434
Definition An EC 2.7.10.* (protein-tyrosine kinase) inhibitor that interferes with the action of receptor protein-tyrosine kinase (EC 2.7.10.1).
Stars This entity has been manually annotated by the ChEBI Team.
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ChEBI Ontology
Outgoing EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434) is a EC 2.7.10.* (protein-tyrosine kinase) inhibitor (CHEBI:76817)
EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434) is a tyrosine kinase inhibitor (CHEBI:38637)
Incoming 1-(3-{5-[4-(aminomethyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)urea (CHEBI:90541) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
1-[4-(3-amino-1H-indazol-4-yl)phenyl]-3-o-tolylurea (CHEBI:131947) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
2,5-dihydroxycinnamic acid methyl ester (CHEBI:84089) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
3,21-dioxoolean-18-en-28-oic acid (CHEBI:65798) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
N-{4-[(3-bromophenyl)amino]quinazolin-6-yl}but-2-ynamide (CHEBI:90180) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
rac-crizotinib (CHEBI:77563) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
AEE788 (CHEBI:40629) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
alectinib (CHEBI:90936) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
alectinib hydrochloride (CHEBI:62268) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
AMG-925 (CHEBI:145537) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
ASP-3026 (CHEBI:167650) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
AZD3463 (CHEBI:167653) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
BAY-826 (CHEBI:192483) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
BMS-754807 (CHEBI:88339) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
brivanib (CHEBI:167686) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
brivanib alaninate (CHEBI:167656) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
ceritinib (CHEBI:78432) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
CP-724714 (CHEBI:167658) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
crenolanib (CHEBI:145365) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
crizotinib (CHEBI:64310) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
DDR1-IN-1 (CHEBI:189867) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
DDR1-IN-2 (CHEBI:191410) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
DMH4 (CHEBI:229963) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
ebselen (CHEBI:77543) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
entrectinib (CHEBI:195558) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
fruquintinib (CHEBI:229221) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
gilteritinib (CHEBI:145372) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
Ki11502 (CHEBI:133397) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
lenvatinib (CHEBI:85994) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
lenvatinib mesylate (CHEBI:85995) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
linifanib (CHEBI:91435) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
lorlatinib (CHEBI:143117) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
orantinib (CHEBI:91088) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
PD-153035 (CHEBI:91076) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
PD-153035 hydrochloride (CHEBI:91075) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
PD-166866 (CHEBI:156259) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
PD158780 (CHEBI:92843) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
PD173074 (CHEBI:63448) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
PDGF receptor tyrosine kinase inhibitor III (CHEBI:143127) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
pexidartinib (CHEBI:145373) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
PQIP (CHEBI:90536) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
quizartinib (CHEBI:90217) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
repotrectinib (CHEBI:229220) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
sapitinib (CHEBI:132986) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
SB 431542 (CHEBI:91108) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
semaxanib (CHEBI:91083) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
SU11652 (CHEBI:132084) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
sunitinib (CHEBI:38940) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
tandutinib (CHEBI:90237) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
tesevatinib (CHEBI:167674) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
TTT-3002 (CHEBI:88219) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
vatalanib (CHEBI:90620) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
vatalanib succinate (CHEBI:90623) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
xestospongin C (CHEBI:131784) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
ZM 323881 hydrochloride (CHEBI:91182) has role EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
c-Met tyrosine kinase inhibitor (CHEBI:90199) is a EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor (CHEBI:62434)
Synonyms Sources
AATK inhibitor ChEBI
AATYK inhibitor ChEBI
AATYK2 inhibitor ChEBI
AATYK3 inhibitor ChEBI
ACH inhibitor ChEBI
ALK inhibitor ChEBI
ALK inhibitors ChEBI
anaplastic lymphoma kinase inhibitor ChEBI
anaplastic lymphoma kinase inhibitors ChEBI
ARK inhibitor ChEBI
ATP:[protein]-L-tyrosine O-phosphotransferase (receptor-type) inhibitor ChEBI
ATP:[protein]-L-tyrosine O-phosphotransferase (receptor-type) inhibitors ChEBI
AXL inhibitor ChEBI
Bek inhibitor ChEBI
Bfgfr inhibitor ChEBI
BRT inhibitor ChEBI
Bsk inhibitor ChEBI
C-FMS inhibitor ChEBI
CAK inhibitor ChEBI
CCK4 inhibitor ChEBI
CD115 inhibitor ChEBI
CD135 inhibitor ChEBI
CDw135 inhibitor ChEBI
Cek1 inhibitor ChEBI
Cek10 inhibitor ChEBI
Cek11 inhibitor ChEBI
Cek2 inhibitor ChEBI
Cek3 inhibitor ChEBI
Cek5 inhibitor ChEBI
Cek6 inhibitor ChEBI
Cek7 inhibitor ChEBI
CFD1 inhibitor ChEBI
CKIT inhibitor ChEBI
CSF1R inhibitor ChEBI
DAlk inhibitor ChEBI
DDR1 inhibitor ChEBI
DDR2 inhibitor ChEBI
Dek inhibitor ChEBI
DKFZp434C1418 inhibitor ChEBI
Drosophila Eph kinase inhibitor ChEBI
DRT inhibitor ChEBI
DTK inhibitor ChEBI
Ebk inhibitor ChEBI
EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitors ChEBI
EC 2.7.10.1 inhibitor ChEBI
EC 2.7.10.1 inhibitors ChEBI
ECK inhibitor ChEBI
EDDR1 inhibitor ChEBI
Eek inhibitor ChEBI
EGFR inhibitor ChEBI
Ehk2 inhibitor ChEBI
Ehk3 inhibitor ChEBI
Elk inhibitor ChEBI
EPH inhibitor ChEBI
EPHA1 inhibitor ChEBI
EPHA2 inhibitor ChEBI
EPHA6 inhibitor ChEBI
EPHA7 inhibitor ChEBI
EPHA8 inhibitor ChEBI
EPHB1 inhibitor ChEBI
EPHB2 inhibitor ChEBI
EPHB3 inhibitor ChEBI
EPHB4 inhibitor ChEBI
EphB5 inhibitor ChEBI
ephrin-B3 receptor tyrosine kinase inhibitor ChEBI
EPHT inhibitor ChEBI
EPHT2 inhibitor ChEBI
EPHT3 inhibitor ChEBI
EPHX inhibitor ChEBI
ERBB inhibitor ChEBI
ERBB1 inhibitor ChEBI
ERBB2 inhibitor ChEBI
ERBB3 inhibitor ChEBI
ERBB4 inhibitor ChEBI
ERK inhibitor ChEBI
Eyk inhibitor ChEBI
FGFR1 inhibitor ChEBI
FGFR2 inhibitor ChEBI
FGFR3 inhibitor ChEBI
FGFR4 inhibitor ChEBI
FLG inhibitor ChEBI
FLK1 inhibitor ChEBI
FLK2 inhibitor ChEBI
FLT1 inhibitor ChEBI
FLT2 inhibitor ChEBI
FLT3 inhibitor ChEBI
FLT4 inhibitor ChEBI
FMS inhibitor ChEBI
Fv2 inhibitor ChEBI
HBGFR inhibitor ChEBI
HEK11 inhibitor ChEBI
HEK2 inhibitor ChEBI
HEK3 inhibitor ChEBI
HEK5 inhibitor ChEBI
HEK6 inhibitor ChEBI
HEP inhibitor ChEBI
HER2 inhibitor ChEBI
HER3 inhibitor ChEBI
HER4 inhibitor ChEBI
HGFR inhibitor ChEBI
HSCR1 inhibitor ChEBI
HTK inhibitor ChEBI
IGF1R inhibitor ChEBI
INSR inhibitor ChEBI
INSRR inhibitor ChEBI
insulin receptor protein-tyrosine kinase inhibitor ChEBI
IR inhibitor ChEBI
IRR inhibitor ChEBI
JTK12 inhibitor ChEBI
JTK13 inhibitor ChEBI
JTK14 inhibitor ChEBI
JWS inhibitor ChEBI
K-SAM inhibitor ChEBI
KDR inhibitor ChEBI
KGFR inhibitor ChEBI
KIA0641 inhibitor ChEBI
KIAA1079 inhibitor ChEBI
KIAA1459 inhibitor ChEBI
Kil inhibitor ChEBI
Kin15 inhibitor ChEBI
Kin16 inhibitor ChEBI
KIT inhibitor ChEBI
KLG inhibitor ChEBI
LTK inhibitor ChEBI
MCF3 inhibitor ChEBI
Mdk1 inhibitor ChEBI
Mdk2 inhibitor ChEBI
Mdk5 inhibitor ChEBI
MEhk1 inhibitor ChEBI
MEN2A/B inhibitor ChEBI
Mep inhibitor ChEBI
MER inhibitor ChEBI
MERTK inhibitor ChEBI
Mlk1 inhibitor ChEBI
Mlk2 inhibitor ChEBI
Mrk inhibitor ChEBI
MST1R inhibitor ChEBI
MTC1 inhibitor ChEBI
MUSK inhibitor ChEBI
Myk1 inhibitor ChEBI
N-SAM inhibitor ChEBI
NEP inhibitor ChEBI
NET inhibitor ChEBI
Neu inhibitor ChEBI
neurite outgrowth regulating kinase inhibitor ChEBI
NGL inhibitor ChEBI
NOK inhibitor ChEBI
nork inhibitor ChEBI
novel oncogene with kinase-domain inhibitor ChEBI
Nsk2 inhibitor ChEBI
NTRK1 inhibitor ChEBI
NTRK2 inhibitor ChEBI
NTRK3 inhibitor ChEBI
NTRK4 inhibitor ChEBI
NTRKR1 inhibitor ChEBI
NTRKR2 inhibitor ChEBI
NTRKR3 inhibitor ChEBI
Nuk inhibitor ChEBI
NYK inhibitor ChEBI
PCL inhibitor ChEBI
PDGFR inhibitor ChEBI
PDGFRA inhibitor ChEBI
PDGFRB inhibitor ChEBI
PHB6 inhibitor ChEBI
PTK inhibitor ChEBI
PTK3 inhibitor ChEBI
PTK7 inhibitor ChEBI
receptor protein tyrosine kinase inhibitor ChEBI
receptor protein-tyrosine kinase (EC 2.7.10.1) inhibitor ChEBI
receptor protein-tyrosine kinase (EC 2.7.10.1) inhibitors ChEBI
receptor protein-tyrosine kinase inhibitor ChEBI
receptor protein-tyrosine kinase inhibitors ChEBI
RET inhibitor ChEBI
RON inhibitor ChEBI
ROR1 inhibitor ChEBI
ROR2 inhibitor ChEBI
ROS1 inhibitor ChEBI
RSE inhibitor ChEBI
RTK inhibitor ChEBI
RYK inhibitor ChEBI
SEA inhibitor ChEBI
Sek2 inhibitor ChEBI
Sek3 inhibitor ChEBI
Sek4 inhibitor ChEBI
Sfr inhibitor ChEBI
SKY inhibitor ChEBI
STK inhibitor ChEBI
STK1 inhibitor ChEBI
TEK inhibitor ChEBI
TIE inhibitor ChEBI
TIE1 inhibitor ChEBI
TIE2 inhibitor ChEBI
TIF inhibitor ChEBI
TKT inhibitor ChEBI
TRK inhibitor ChEBI
TRKA inhibitor ChEBI
TRKB inhibitor ChEBI
TRKC inhibitor ChEBI
TRKE inhibitor ChEBI
TYK1 inhibitor ChEBI
TYRO10 inhibitor ChEBI
Tyro11 inhibitor ChEBI
TYRO3 inhibitor ChEBI
Tyro5 inhibitor ChEBI
Tyro6 inhibitor ChEBI
TYRO7 inhibitor ChEBI
UFO inhibitor ChEBI
VEGFR1 inhibitor ChEBI
VEGFR2 inhibitor ChEBI
VEGFR3 inhibitor ChEBI
Vik inhibitor ChEBI
YK1 inhibitor ChEBI
Yrk inhibitor ChEBI
Manual Xref Database
Anaplastic_lymphoma_kinase Wikipedia
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Last Modified
12 April 2024